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N-(3-methylbutyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-(2-methoxyethyl)-4-(1H-pyrazol-3-yl)-N-(pyridin-4-ylmethyl)benzamide
ethyl 2-(2-{[1-methyl-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-yl]amino}ethyl)-1,3-thiazole-4-carboxylate
2-(3,6-dimethylpyrazin-2-yl)-5-[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridine
2-{[2-(4-chlorophenyl)morpholin-4-yl]methyl}-5-methoxypyridin-4-ol
(2S)-2-[2-(2-fluoro-4,5-dimethoxyphenyl)-1H-imidazol-1-yl]-4-(methylsulfanyl)butan-1-ol
7-[(3-methoxyphenyl)methyl]-2-(6-methylpyridine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
2-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]acetic acid
N-[3-(cyclohexyloxy)propyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
N-(3,5-dimethoxyphenyl)-3-[1-(oxan-4-yl)piperidin-3-yl]propanamide
3-chloro-2-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1H-indole
1-(1-ethyl-3,5-dimethyl-1H-pyrazole-4-carbonyl)-4-(2-methylphenyl)-1,4-diazepane
2-(oxan-4-yl)-1-{2-[5-(piperidine-1-carbonyl)thiophen-2-yl]pyrrolidin-1-yl}ethan-1-one
4-{1-[4-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)phenyl]piperidin-4-yl}-1,4-diazepane-1-carbaldehyde
{3-cyclobutanecarbonyl-9-[(5-methylthiophen-2-yl)methyl]-3,9-diazaspiro[5.5]undecan-1-yl}methanol
1-(1-methyl-1H-imidazole-2-carbonyl)-4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
4-(1-{[4-(butan-2-yloxy)-3-chloro-5-methoxyphenyl]methyl}azetidin-3-yl)morpholine
1-methyl-5-{1-[4-(methylsulfanyl)phenyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}-1H-pyrazole
5-(2-methylpropyl)-1'-(1,2-oxazole-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-{[1-(2-cyclohexylethyl)-3-hydroxy-2-oxopiperidin-3-yl]methyl}piperazin-2-one
4-{[1-(4-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1-methyl-1H-pyrazole
4-{[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-1H-imidazol-1-yl]methyl}-2-(propan-2-yl)-1,3-thiazole
3-phenyl-1-(4-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)propan-1-ol
1-(cyclohexylmethyl)-N,N-dimethyl-5-{[(5-methylfuran-2-yl)methyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-{1-[(3,4-difluorophenyl)methyl]-4-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl}ethan-1-ol
(3S,4R)-1-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-4-methyl-3-(2-methylpropyl)piperidin-4-ol
5-{2-[1-tert-butyl-3-(oxolan-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1,2-oxazol-3-ol
(1S,5R)-6-[(1-methyl-1H-imidazol-2-yl)methyl]-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
2-{[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl](thiophen-3-ylmethyl)amino}butan-1-ol
2-({[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}amino)-6-methylpyridine-3-carbonitrile
N-{[1-(1,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)piperidin-3-yl]methyl}-4-fluorobenzamide
2-[(4aR,6R,8aS)-8a-(methoxymethyl)-6-(morpholin-4-yl)-decahydroisoquinolin-2-yl]-6-methylpyridine-3-carbonitrile
N-(6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
2-({4-[2-(pyridin-4-yl)ethyl]piperazin-1-yl}methyl)pyridine-3-carboxylic acid
4-{[(butan-2-yl)(thiophen-3-ylmethyl)amino]methyl}-N-methylbenzene-1-sulfonamide
1-[5-(2-chloro-4-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]-4,4-dimethylpiperidine
N-(3-chloro-4-methoxyphenyl)-6-[(3-ethoxy-4-hydroxyphenyl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
ethyl 4-(oxan-2-ylmethyl)-1-phenylmethanesulfonylpiperidine-4-carboxylate
2-{3-[(4-aminopiperidin-1-yl)methyl]phenyl}-6-(2-chlorophenyl)-3,4-dihydropyrimidin-4-one
2-[(2,6-dichlorophenyl)methyl]-4-hydroxy-N-methyl-N-(1-methylpyrrolidin-3-yl)pyrimidine-5-carboxamide
[3-(cyclopropylmethyl)-1-{[6-(trifluoromethyl)pyridin-3-yl]methyl}piperidin-3-yl]methanol
5-({2-[4-(1H-imidazol-1-yl)phenyl]-1H-imidazol-1-yl}methyl)-1,3-dimethyl-2,3-dihydro-1H-1,3-benzodiazol-2-one
8-[(benzylcarbamoyl)methyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-2-(4-fluorophenyl)piperidine
N-[(1-methylpiperidin-2-yl)methyl]-3-(4-methylthiophen-2-yl)-5-(morpholine-4-sulfonyl)benzamide
N,1-dimethyl-N-(1,2-oxazol-5-ylmethyl)-6-(2-phenylethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-ethyl-3-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}propanamide
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-[({[1-(propan-2-yl)cyclopropyl]methyl}amino)methyl]piperidin-2-one
(3S,4R)-N,N-dimethyl-4-propyl-1-(pyridine-3-sulfonyl)pyrrolidin-3-amine
3-(1-{6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}piperidin-3-yl)propan-1-ol