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3-(3-methoxy-4-methylphenyl)-1-[2-(trifluoromethyl)morpholin-4-yl]propan-1-one
1-methyl-N-(3-methylbutyl)-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-[(3R,7S,8aS)-3-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[2-(trifluoromethyl)phenyl]urea
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-(pyridin-4-ylmethyl)piperidine-4-carboxamide
2-(4-chloro-2-methylphenoxy)-1-[1-(pyridin-4-ylmethyl)-3-(pyrrolidine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]ethan-1-one
5-{[2-(methoxymethyl)piperidin-1-yl]methyl}-2-phenylpyrimidine
N,N-dimethyl-5-(2-oxo-6-phenyl-1,2-dihydropyridine-3-carbonyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-3-carboxamide
5-{[benzyl(methyl)amino]methyl}-N-[(2R)-1-hydroxy-3-methylbutan-2-yl]-1,2-oxazole-3-carboxamide
N-[2-(ethanesulfonyl)ethyl]-2-fluoro-5-sulfamoylbenzamide
1-(1-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-1-oxopropan-2-yl)pyrrolidin-2-one
2-amino-N-[2-methoxy-2-(thiophen-2-yl)ethyl]-6-methylpyrimidine-4-carboxamide
4-(4-methoxyphenoxy)-1-(1H-pyrrole-3-carbonyl)piperidine
6-(aminomethyl)-N-[(1-cyclopropanecarbonylpiperidin-3-yl)methyl]-2-methylpyrimidin-4-amine
methyl(oxan-2-ylmethyl)[(2-phenyl-1H-imidazol-4-yl)methyl]amine
(2S,4S)-1-acetyl-N-ethyl-4-[3-(1-methyl-1H-pyrrol-2-yl)propanamido]pyrrolidine-2-carboxamide
1-[4-({[(1-methylpiperidin-4-yl)methyl](2-phenylethyl)amino}methyl)thiophen-2-yl]ethan-1-one
1-(2-methylphenyl)-4-[4-(1H-pyrazol-4-yl)butanoyl]piperazin-2-one
1-[5-(2,6-dimethylphenoxymethyl)-1,2-oxazole-3-carbonyl]-4-phenylpiperidine
N-(3-chloro-4-methoxyphenyl)-3-[1-(2,2-dimethyl-4-oxo-3,4-dihydro-2H-pyran-6-carbonyl)piperidin-3-yl]propanamide
(1S,6R)-9-{[4-(2-methylpropyl)phenyl]methyl}-3,9-diazabicyclo[4.2.1]nonan-4-one
1-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)-4-(pyrimidin-2-yl)-1,4-diazepane
6-methyl-4-oxo-N-{[4-(pyrrolidin-1-ylmethyl)phenyl]methyl}-1,4-dihydropyridine-3-carboxamide
9-{3-methoxy-4-[(1-methylpiperidin-4-yl)oxy]benzoyl}-6-oxa-9-azaspiro[4.5]decane
4,6-dimethyl-2-{3-[4-(2-methylphenyl)piperazin-1-yl]piperidin-1-yl}pyridine-3-carbonitrile
(1S,5R)-3-[(3,5-dichloropyridin-4-yl)methyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonane
1-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-methyl-2-phenylpropan-1-one
(4-{[methyl(2-phenylpropyl)amino]methyl}oxan-4-yl)methanol
2-(3-methoxypropyl)-1-(thiophene-3-sulfonyl)piperidine
N-[(2-fluorophenyl)methyl]-3-[(3S,4R)-1-(2-methylpropyl)-4-(morpholin-4-yl)piperidin-3-yl]propanamide
N-(3-ethyl-4-methyl-1-phenyl-1H-pyrazol-5-yl)furan-3-carboxamide
(3R,4R)-4-(morpholin-4-yl)-1-[(3-phenoxyphenyl)methyl]piperidin-3-ol
2-methyl-N-{5-[2-(4-methylphenoxy)ethyl]-1,3,4-thiadiazol-2-yl}-1H-imidazole-4-carboxamide
2-{5-[(2,4-dimethoxyphenyl)methyl]-3-(pyridin-4-yl)-1H-1,2,4-triazol-1-yl}acetic acid
N,1,3-trimethyl-N-[3-(oxolan-2-yl)propyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
3-(4-hydroxyphenyl)-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-1H-pyrazole-5-carboxamide
2-(5-acetylthiophen-3-yl)-N-cyclopentyl-N-(thiophen-3-ylmethyl)acetamide
N-(propan-2-yl)-1-[(1s,4s)-4-(4-methoxybenzenesulfonamido)cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
2-amino-N-[2-fluoro-4-(6-methoxypyridin-3-yl)phenyl]acetamide
(1s,4s)-4-[(1R,3R,5S)-3-(4-fluoro-3-methylphenyl)-8-azabicyclo[3.2.1]octane-8-carbonyl]cyclohexan-1-ol
N-{[(3S,4S)-3-hydroxy-1-[(2E)-3-phenylprop-2-enoyl]piperidin-4-yl]methyl}furan-2-carboxamide
4-amino-N-(2-methoxyethyl)-N-(thiophen-2-ylmethyl)pyridine-2-carboxamide
2,3-dimethyl-5-{2-methyl-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl}benzene-1-sulfonamide
N-methyl-N-[1-(3-phenylpropyl)piperidin-3-yl]-3-(propan-2-yl)-1,2-oxazole-5-carboxamide
N-({2-[4-(furan-3-amido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-5-methyl-3-phenyl-1,2-oxazole-4-carboxamide
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-{1-[2-(methylsulfanyl)benzoyl]piperidin-4-yl}propanamide
(1S,5R)-1,3,3-trimethyl-6-[2-(phenoxymethyl)-1,3-oxazole-4-carbonyl]-6-azabicyclo[3.2.1]octane
6-(azocane-1-carbonyl)-2-[(3,4-dimethoxyphenyl)methyl]-1,3-benzoxazole
methyl 5-[(3-carbamoylpiperidine-1-carbonyl)amino]-2-chlorobenzoate
1-{3-[4-(5-chloropyridin-2-yl)piperazin-1-yl]-3-oxopropyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-(1H-1,3-benzodiazol-2-ylmethyl)-3H,4H-thieno[3,2-d]pyrimidin-4-one