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3-{3-[(dimethylamino)methyl]-3-hydroxypiperidine-1-carbonyl}-2-methyl-4,5,6,7-tetrahydro-1H-indol-4-one
2-hydroxy-1-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
N-[(3S,4R)-1-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
1-(2-{methyl[(1-propyl-1H-imidazol-2-yl)methyl]amino}ethyl)piperidin-2-one
1-[1-(3-fluoropropyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
1-{4-[(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)methyl]phenyl}pyrrolidin-2-one
1-{7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-3-(1,2-oxazinan-2-yl)propan-1-one
N-[2-hydroxy-3-(piperazin-1-yl)propyl]-3-(1H-pyrazol-1-yl)benzamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-5-[(dimethylsulfamoyl)amino]-1-methyl-2-(2-methylpropyl)-1H-1,3-benzodiazole-7-carboxamide
N-({3-[3-(dimethylamino)propoxy]-4-methoxyphenyl}methyl)-4-fluoro-N-(pyridin-3-ylmethyl)benzamide
[1-(5-{[(2-ethylpyrimidin-5-yl)methyl]amino}-5,6,7,8-tetrahydroquinazolin-2-yl)piperidin-4-yl]methanol
1-{1-[(2-chloro-4-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-3-(2-methylphenyl)piperidine
7-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]-1,2,3,4-tetrahydroquinoxalin-2-one
(2S,4R)-1-(cyclohexylmethyl)-N-ethyl-4-[2-(pyridin-3-yl)acetamido]pyrrolidine-2-carboxamide
ethyl 4-[4-(5-carbamoylpyridin-2-yl)piperazin-1-yl]piperidine-1-carboxylate
2-(2-methoxyethyl)-8-[4-methyl-6-(methylamino)pyrimidin-2-yl]-2,8-diazaspiro[5.5]undecan-3-one
ethyl 1-(3-methylbutyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
{[1-(2-methoxyethyl)-2-(3-methylbutanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)(propan-2-yl)amine
8-[5-(1H-imidazol-1-ylmethyl)pyridin-2-yl]quinoline
3-[(1H-imidazol-2-ylmethyl)(methyl)sulfamoyl]-N-(3-methylbutan-2-yl)benzamide
2-[(3aR,6aS)-octahydropyrrolo[3,4-c]pyrrole-2-carbonyl]-4-chloro-1-methyl-1H-pyrrole
4-{[4-(aminomethyl)-1H-1,2,3-triazol-1-yl]methyl}-N-(2H-1,3-benzodioxol-5-yl)piperidine-1-carboxamide
1-[5-(2,4-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]piperidin-3-ol
({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)(methyl){[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}amine
N-(furan-2-ylmethyl)-2-methyl-2,8-diazaspiro[4.5]decane-8-carboxamide
N-(2-{[7-(pyridine-3-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]amino}ethyl)acetamide
N-(oxolan-2-ylmethyl)-3-[1-(3,3,5,5-tetramethylcyclohexyl)piperidin-4-yl]propanamide
4-[2-(pyrrolidin-1-yl)ethyl]-1-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)-1,4-diazepan-5-one
4-(2-{1-[1-(2-fluorophenyl)cyclopropanecarbonyl]piperidin-2-yl}ethyl)morpholine
4-[5-cyclobutyl-3-(oxolan-3-yl)-1H-1,2,4-triazol-1-yl]benzene-1-sulfonamide
{[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]amine
2-[(4-chlorophenyl)methyl]-8-(1H-imidazol-2-ylmethyl)-2,8-diazaspiro[4.5]decan-3-one
4-methyl-6-(quinolin-8-yl)pyrimidin-2-amine
5-[3-(2-methylphenoxymethyl)piperidine-1-carbonyl]-1H-indole
2-{3-[1-(1,4-dioxan-2-ylmethyl)-1H-pyrazol-3-yl]phenyl}-1,3-thiazole
N-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-N-methyl-2-(2-oxopyrrolidin-1-yl)propanamide
2-(oxolan-2-ylmethyl)-4-[3-(thiomorpholine-4-carbonyl)piperidin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
2-cyclopropyl-N,4-dimethyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]pyrimidine-5-carboxamide
methyl[3-(1-methyl-1H-pyrazol-4-yl)propyl]({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)amine
7-fluoro-3-methyl-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-1-benzofuran-2-carboxamide
1-{[4-(dimethylamino)oxan-4-yl]methyl}-3-(1-phenyl-1H-pyrazol-5-yl)urea
N-{[2-(methoxymethyl)-4-methyl-1,3-thiazol-5-yl]methyl}-2-(morpholin-4-yl)benzamide
5-benzyl-4-(cyclopropylmethyl)-1-(3-methoxyphenyl)piperazin-2-one
2-[2-(furan-2-yl)-4-(1,2,3,6-tetrahydropyridin-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]acetic acid
methyl 4-({[2-(3-carbamoylpiperidin-1-yl)ethyl]carbamoyl}amino)-2-chlorobenzoate
4-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}-N-ethyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]benzamide
3-(1,3-benzothiazol-2-yl)-1-{3-[(3,4-dimethoxyphenyl)amino]piperidin-1-yl}propan-1-one
3-[(2-hydroxyethyl)({[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl})amino]-1λ6-thiolane-1,1-dione
5-{1-[(2-hydroxy-3-methoxyphenyl)methyl]piperidin-4-yl}-5-(2-methylpropyl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
N-{1-oxo-1-[3-oxo-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-9-yl]pentan-2-yl}acetamide