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4-chloro-2-{[4-cyclohexyl-3-(2-hydroxyethyl)piperazin-1-yl]methyl}phenol
3-(2-phenylethyl)-8-[(2S)-pyrrolidine-2-carbonyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(4aR,7aS)-1-ethyl-4-[(3-phenoxyphenyl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
8-(1-benzothiophene-5-carbonyl)-2-ethyl-2,8-diazaspiro[4.5]decan-3-one
N-(2-ethoxyethyl)-3-{[1-(pyrimidin-4-yl)ethyl]sulfamoyl}benzamide
N-(3-hydroxy-2,2-dimethylpropyl)-N-methyl-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
methyl 2-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}pyridine-3-carboxylate
N-benzyl-3-[1-(1-ethylpiperidine-2-carbonyl)piperidin-4-yl]-N-methylpropanamide
(3ar,6ar)-N-[2-(3-benzyl-1,2,4-oxadiazol-5-yl)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
1-(pyridin-3-ylmethyl)-4-[4-(pyrrolidine-1-carbonyl)pyridin-2-yl]-1,4-diazepane
1-[1'-(2,5-dimethylfuran-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanamide
3-methyl-N-{[4-(3-methylpiperidin-1-yl)phenyl]methyl}-1-propyl-1H-pyrazole-4-carboxamide
1-[6-methyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-N-[(3-methyloxetan-3-yl)methyl]piperidin-4-amine
(1R,3S)-7-(4-chloro-1-methyl-1H-pyrazole-3-carbonyl)-7-azaspiro[3.5]nonane-1,3-diol
N-[2-(ethylsulfanyl)ethyl]-2-methylimidazo[1,2-a]pyridine-6-carboxamide
N-cyclopropyl-1-[1-(2,6-dihydroxybenzoyl)piperidin-4-yl]piperidine-4-carboxamide
1-methyl-4-({3-[4-(trifluoromethyl)phenyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)-1H-pyrazole
4-[(2-hydroxyethyl)sulfamoyl]-N-[1-(pyrazin-2-yl)propan-2-yl]benzamide
(2S,4R)-N-[2-(3-fluorophenyl)ethyl]-4-[(4-fluorophenyl)sulfanyl]-1-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
1-[3-(azetidine-1-sulfonyl)benzoyl]-3-(methoxymethyl)piperidine
5-(azepane-1-carbonyl)-1-(2-methylpropyl)-4-oxo-N-{[3-(trifluoromethyl)phenyl]methyl}-1,4-dihydropyridine-3-carboxamide
N-{[5-(2-acetylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-methoxy-2-phenylacetamide
1-{2-hydroxy-3-[3-({methyl[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]amino}methyl)phenoxy]propyl}piperidin-4-ol
4-{1-[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazole-4-carbonyl]azetidin-3-yl}pyridine
1-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecan-4-yl]-2-(1H-1,2,4-triazol-1-yl)propan-1-one
8-(furan-3-ylmethyl)-1-(2-methylpropyl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-{1-[(2-methylphenyl)methyl]-4-{[2-(prop-2-en-1-yloxy)phenyl]methyl}piperazin-2-yl}ethan-1-ol
N-ethyl-N-(2-hydroxyethyl)-1-[(3-methoxyphenyl)methyl]-6-oxopiperidine-3-carboxamide
{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}({[4-(1H-imidazol-1-yl)phenyl]methyl})methylamine
3-(2-oxo-2-{4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidin-1-yl}ethyl)-1,3-oxazolidin-2-one
3-{imidazo[1,2-a]pyridin-2-yl}-N-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]propanamide
5-chloro-4,6-dimethyl-2-oxo-N-[phenyl(pyridin-4-yl)methyl]-1,2-dihydropyridine-3-carboxamide
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N,1-dimethyl-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
N-(2-{4-[(1-methyl-1H-pyrazol-4-yl)methyl]morpholin-2-yl}ethyl)thiophene-3-carboxamide
1-[4-methyl-2-({[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}amino)pyrimidin-5-yl]ethan-1-one
(1S,5R)-6-[(2-chloro-4-fluorophenyl)methyl]-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-(2-ethoxybutyl)-2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-amine
1-{4-[3-(3-methoxybenzoyl)piperidin-1-yl]piperidin-1-yl}ethan-1-one
(1R,5S,8S)-3-[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]-3-azabicyclo[3.2.1]octan-8-ol
2-methoxy-N-{1-[1-(pyrazin-2-yl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
1-methyl-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1H-imidazole-5-carboxamide
N-(2-methylpropyl)-N-[(2E)-3-phenylprop-2-en-1-yl]-2-(1H-1,2,4-triazol-3-yl)benzamide
2-{1-methyl-5-[2-(morpholin-4-yl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}-1,2,3,4-tetrahydroisoquinoline
4-(4-ethoxyphenyl)-3-(3,3,3-trifluoropropyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
5-(2-{3-[(4-fluorophenyl)amino]piperidin-1-yl}-2-oxoethyl)-2,6-dimethyl-3,4-dihydropyrimidin-4-one
N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-amine
N-methyl-4-(2-oxopyrrolidin-1-yl)-N-[1-(pyridin-3-yl)propyl]butanamide
4-[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]pyrrolidin-2-one