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2-{[6-(4-cyclohexylpiperazin-1-yl)pyridazin-3-yl]oxy}-N-[2-(2-fluorophenyl)ethyl]acetamide
4-fluoro-N-(oxolan-2-ylmethyl)-N-({3-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)benzene-1-sulfonamide
3-(cyclopropylmethyl)-1-[4-(1H-1,2,4-triazol-1-yl)butanoyl]piperidine-3-carboxylic acid
1-benzyl-8-[(5-chloro-2-hydroxyphenyl)methyl]-3-(2-methoxyethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
6-(methylsulfanyl)-2-[3-(4H-1,2,4-triazol-4-yl)benzoyl]-1,2,3,4-tetrahydroisoquinoline
3-(2H-1,3-benzodioxol-5-yl)-5-{spiro[2.4]heptane-1-carbonyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
8-fluoro-4-oxo-N-(pyridin-3-ylmethyl)-1,4-dihydroquinoline-2-carboxamide
1-(2-oxo-2-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethyl)-1,2-dihydropyrimidin-2-one
5-(methoxymethyl)-N-[4-(5-methyl-4-{[3-(1H-1,2,4-triazol-1-yl)propanamido]methyl}-1,3-oxazol-2-yl)phenyl]thiophene-2-carboxamide
2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-4-yl)-N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]acetamide
7-[(3S)-3-phenylbutanoyl]-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
(1R,5S)-3-(1-ethyl-5-methyl-1H-pyrazole-4-carbonyl)-3,8-diazabicyclo[3.2.1]octane
1-{[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}-2-methyl-1,4-diazepan-5-one
3-(3-chloro-4-propoxyphenyl)-1-[(1S,2S)-2-hydroxycyclohexyl]urea
2-methyl-6-{1-[2-(1H-pyrazol-1-yl)benzoyl]piperidin-3-yl}pyrimidin-4-ol
2-[3-(methoxymethyl)-5-oxo-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-1-yl]-N-methyl-N-(1,3-thiazol-2-ylmethyl)acetamide
2-methyl-1-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-(4-methylphenyl)piperazine
N-[(2-methoxyphenyl)methyl]-N-(pyridin-4-ylmethyl)oxane-4-carboxamide
N-{6-ethyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-1-(oxolan-2-ylmethyl)piperidin-4-amine
N-[2-(dimethylamino)-2-(furan-2-yl)ethyl]-4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzamide
[(3R,4R)-4-[(dimethylamino)methyl]-1-(4-ethyl-2-methyl-1,3-thiazole-5-carbonyl)pyrrolidin-3-yl]methanol
(3aR,6aS)-5-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(4-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}phenyl)methanol
(4aR,8aR)-2-cyclobutanecarbonyl-7-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}-decahydro-2,7-naphthyridin-4a-ol
3-(2-amino-4-methyl-6-{[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]amino}pyrimidin-5-yl)propanoic acid
1-(4-{[4-(2,8-dimethylquinoline-4-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperazin-1-yl)ethan-1-one
4-[4-(thiophen-2-ylmethyl)piperazin-1-yl]-2-{[3-(trifluoromethyl)phenyl]methyl}-2,3-dihydro-1H-isoindole-1,3-dione
{[2-cyclopropylmethanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}[(1-ethyl-1H-imidazol-2-yl)methyl]methylamine
2-[1-(3,5-dimethyl-1-benzofuran-2-carbonyl)piperidin-3-yl]-1,3-benzoxazole
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-2-(ethylamino)pyrimidine-5-carboxamide
4-[(4-ethoxyphenyl)methyl]-3-[2-(1,2-oxazolidin-2-yl)-2-oxoethyl]piperazin-2-one
6-fluoro-N-[1-(6-methylpyridin-3-yl)ethyl]-2-(1H-pyrazol-4-yl)quinoline-4-carboxamide
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-3-methoxy-5-methylthiophene-2-carboxamide
(2S)-2-phenyl-2-{4-phenyl-5-[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-1H-imidazol-1-yl}ethan-1-ol
1-({1-[(3-methylquinoxalin-2-yl)methyl]pyrrolidin-3-yl}methyl)-3-(propan-2-yl)urea
ethyl 1-[3-(2-phenylethyl)-1,2-oxazole-5-carbonyl]piperidine-2-carboxylate
(1R,3s,6r,8S)-N-benzyl-4-azatricyclo[4.3.1.13,8]undecane-4-sulfonamide
2-(1H-pyrazol-3-yl)-5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridine
1-methyl-N-[(5-methylpyrazin-2-yl)methyl]piperidine-2-carboxamide
2-(2,3-dihydro-1H-inden-1-yl)-N-[(1-hydroxycyclohexyl)methyl]acetamide
1-(3-methoxypropyl)-8-(2-phenylethyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-methyl-2-{5-[1-(propan-2-yl)pyrrolidin-3-yl]-1,2,4-oxadiazol-3-yl}pyridine
4-[3-(piperidine-1-carbonyl)pyrazine-2-carbonyl]piperazine-2-carboxylic acid
3-(3-fluorophenyl)-5-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
2-(3-hydroxyphenyl)-2-(3-oxo-4-phenylpiperazin-1-yl)acetic acid
2-{1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)benzoyl]pyrrolidin-2-yl}pyridine
N-(1-{2-oxo-2-[1-(propan-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]ethyl}-1H-pyrazol-4-yl)-2H-1,3-benzodioxole-5-carboxamide
methyl[(5-phenyl-1,2-oxazol-3-yl)methyl]{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}amine
2-[4-cyclohexyl-3-(2-hydroxyethyl)piperazin-1-yl]ethan-1-ol
2-methyl-5-[4-(2-{3-methyl-2-oxo-2H,3H-imidazo[1,2-a]pyridin-3-yl}acetyl)piperazin-1-yl]-2,3-dihydropyridazin-3-one