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N-(1-{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}pyrrolidin-3-yl)acetamide
3-chloro-4-({1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]piperidin-4-yl}oxy)-N-(2-methoxyethyl)benzamide
N-[(1S,2R)-2-(cycloheptylamino)cyclobutyl]-2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]acetamide
3-{2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]acetamido}-N-(1,3-thiazol-2-yl)propanamide
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)-4-(1H-1,2,4-triazol-1-yl)butanamide
methyl 2-{4-[(5-methyl-1,3,4-thiadiazol-2-yl)carbamoyl]-2-oxopiperazin-1-yl}acetate
1-(1-methylpiperidine-2-carbonyl)-4-[3-(trifluoromethyl)phenyl]piperazine
1-(azocan-1-yl)-3-(2-methoxy-4-{[methyl(1,2-oxazol-3-ylmethyl)amino]methyl}phenoxy)propan-2-ol
(3S,4S)-1-(2,3-dimethylquinoxaline-6-carbonyl)-4-(1H-imidazol-2-yl)pyrrolidine-3-carboxylic acid
4-{1-[(2,3-dimethoxyphenyl)methyl]-1H-imidazol-2-yl}-3-methoxyphenol
5-{2-[3-(1H-imidazol-2-yl)piperidin-1-yl]-2-oxoethyl}-3-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[(8-methoxy-2H-chromen-3-yl)methyl]-4-(pyrrolidine-1-carbonyl)piperidine
1-[(1-{6-[(pentan-2-yl)amino]pyridine-3-carbonyl}piperidin-4-yl)methyl]pyrrolidin-2-one
2-(4-fluorophenyl)-N-(oxolan-2-ylmethyl)-N-({3-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)acetamide
1-methyl-1'-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
1-cyclohexyl-3-[2-(methylsulfanyl)ethyl]-5-[3-(1H-pyrazol-1-yl)propyl]-1H-1,2,4-triazole
5-[2-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-oxoethyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
(2S,4R)-4-amino-N,N-diethyl-1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}pyrrolidine-2-carboxamide
N-cycloheptyl-4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}benzamide
2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]-1-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
5-acetyl-N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-N-methylthiophene-3-carboxamide
1-(4-{[(2R)-hexan-2-yl]amino}-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
1-(2-oxo-2-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethyl)-1,2-dihydropyrimidin-2-one
methyl 4-[(4-{4-methyl-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)methyl]benzoate
2-amino-6-(3,4-difluorophenyl)-4-{2-[(propan-2-yl)amino]pyrimidin-5-yl}pyridine-3-carbonitrile
3-(4-hydroxyphenyl)-N-[3-(1H-indol-1-yl)propyl]-1H-pyrazole-5-carboxamide
4-hydroxy-N-[1-phenyl-2-(pyrrolidin-1-yl)ethyl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide
methyl 4-methyl-3-({[2-(1-methyl-1H-pyrazol-5-yl)ethyl]carbamoyl}amino)benzoate
1-[(2-methoxyphenyl)methyl]-4-({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)piperazine
1-cyclopropyl-N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-5-oxopyrrolidine-3-carboxamide
2-{1-[3-(4-methoxyphenyl)-1H-pyrazole-5-carbonyl]piperidin-2-yl}pyridine
5-({4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}methyl)-N-(oxolan-2-ylmethyl)pyrimidin-2-amine
(3aS,6aR)-5-[(1-ethyl-1H-pyrazol-4-yl)methyl]-3-[3-(4-fluorophenyl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
5-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-1-(2-fluorophenyl)-3-methyl-1H-1,2,4-triazole
N-[4-({3-[5-(4-fluorophenyl)-2-methylpyrimidin-4-yl]piperidin-1-yl}methyl)phenyl]acetamide
N-(oxolan-2-ylmethyl)-N-({3-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)propanamide
4-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidine-1-carbonyl]-1-(propan-2-yl)pyrrolidin-2-one
N-cyclopentyl-3-acetamido-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)propanamide
3-{2-[2-(4-fluorophenyl)pyrrolidin-1-yl]-2-oxoethyl}-3-(2-methylphenyl)-1-(pyridin-3-ylmethyl)pyrrolidine-2,5-dione
N-[3-(4-methoxyphenyl)propyl]-6-(4-methyl-1,4-diazepan-1-yl)pyridine-3-carboxamide
ethyl 1-(2-amino-1,3-benzothiazole-5-carbonyl)-4-(3-phenylpropyl)piperidine-4-carboxylate
2-(dimethylamino)-2-(3-fluorophenyl)-1-{4-[2-(morpholin-4-yl)ethyl]piperazin-1-yl}ethan-1-one
1,3-dimethyl-5-(2-{3-[(2-methylphenyl)methoxy]azetidin-1-yl}-2-oxoethyl)imidazolidine-2,4-dione
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-3-methylpentanamide
9-[3-(2-ethoxyethoxy)benzoyl]-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
(1R,5S)-6-{[2-(3,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-6-azabicyclo[3.2.1]octane
3-(1H-imidazol-1-ylmethyl)-1-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}piperidine
2-[(3R,4S)-3-amino-4-phenylpyrrolidin-1-yl]-1-(morpholin-4-yl)ethan-1-one
N-[2-(2-fluorophenyl)ethyl]-2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]acetamide
1-[4-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethan-1-one