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3-({[1-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)piperidin-3-yl]oxy}methyl)pyridine
2-methyl-6-({5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-4H-pyran-4-one
ethyl 4-{5-cyclopropyl-1-[4-(3-fluoro-4-methoxyphenyl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl}piperazine-1-carboxylate
1-[(3,4-difluorophenyl)methyl]-3-hydroxy-3-({[2-(morpholin-4-yl)ethyl]amino}methyl)piperidin-2-one
2-{[4-(1-propyl-1H-imidazol-2-yl)-1H-1,2,3-triazol-1-yl]methyl}-3,4-dihydroquinazolin-4-one
2-hydroxy-3-methyl-1-[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]butan-1-one
4-{1-[(5-fluoro-2-methylphenyl)methyl]-1H-imidazol-2-yl}-1-(2-methoxyethyl)piperidine
methyl 3-{[1-(2-cyclohexylethyl)-1H-1,2,3-triazol-4-yl]formamido}propanoate
N-[2-(pyridin-3-yloxy)ethyl]-1-[4-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)phenyl]piperidin-4-amine
2-cyclopropyl-5-[2-(trifluoromethyl)morpholine-4-carbonyl]-3,4-dihydropyrimidin-4-one
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
4-{1-[(2,4-dimethoxyphenyl)carbamoyl]piperidin-3-yl}benzoic acid
2-benzyl-8-(9H-purin-6-yl)-2,8-diazaspiro[4.5]decan-3-one
4-{[2-(4-fluorophenyl)pyrrolidin-1-yl]methyl}-2-(propan-2-yl)pyrimidine
4-(hydroxymethyl)-1-[5-(oxolan-2-yl)thiophene-2-carbonyl]piperidin-4-ol
6-[1-(1-benzofuran-2-sulfonyl)piperidin-4-yl]-3,4-dihydropyrimidin-4-one
2-(morpholin-4-yl)-N-{4-[2-(pyridin-4-yl)-1H-imidazol-1-yl]phenyl}acetamide
N-(1-{7-[(2,3-difluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-phenoxyacetamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-2-methoxy-N-(pentan-3-yl)pyrimidine-5-carboxamide
3-(3,4-dimethoxybenzoyl)-1-[(3-phenyl-1H-pyrazol-4-yl)methyl]piperidine
N-[(2R,4R,6S)-2-tert-butyl-6-(2,4,5-trimethylphenyl)oxan-4-yl]acetamide
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-N5-(2-phenoxyethyl)piperidine-3,5-dicarboxamide
(3R,4R)-4-ethyl-1-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]piperidine-3,4-diol
2-{1-[(3-chloro-5-fluorophenyl)methyl]pyrrolidin-2-yl}-5-fluoro-1H-1,3-benzodiazole
3-(2-phenoxyethyl)-1-(quinoxalin-2-yl)piperidine-3-carboxylic acid
1-(pyridin-2-ylmethyl)-N-[(2,4,5-trimethoxyphenyl)methyl]piperidin-3-amine
(2S,4R)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-[(3-chlorophenyl)methyl]-4-(cyclooctylamino)pyrrolidine-2-carboxamide
ethyl 4-[(4-chlorophenyl)methyl]-1-[(4S,6R)-6-methyl-2-sulfanylidene-1,3-diazinane-4-carbonyl]piperidine-4-carboxylate
3-{1-[1-(2,3-dihydro-1-benzofuran-5-carbonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}pyridine
N-[(4-fluorophenyl)methyl]-2-hydroxy-N-(oxolan-2-ylmethyl)-4-(1H-1,2,3,4-tetrazol-1-yl)benzamide
3-(3,5-dimethylphenyl)-5-[(4-methylpiperazin-1-yl)sulfonyl]benzoic acid
ethyl 1-{4-[(2-methylprop-2-en-1-yl)oxy]benzoyl}piperidine-2-carboxylate
4-{[5-(2-chlorophenyl)furan-2-yl]methyl}-9-methoxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-amino-N-[2-(dimethylamino)ethyl]-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)-2-methylpropanamide
2-methyl-3-[(4-methyl-1,2,3,6-tetrahydropyridin-1-yl)methyl]quinoxaline
propyl 2-(phenylcarbamoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxylate
3-[(3,4-dimethoxypyridin-2-yl)methyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-[1-(1H-imidazol-4-ylmethyl)piperidin-3-yl]-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-cyclopropyl-N-[3-(4-ethoxyphenyl)propyl]pyrimidine-5-carboxamide
6-ethyl-1-methyl-N-{1-[2-(1H-pyrazol-1-yl)phenyl]ethyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1'-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-[(5-phenyl-1H-pyrazol-3-yl)methyl]-3-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)propanamide
2-amino-N-({2-[4-(2-methylphenyl)piperazin-1-yl]pyridin-3-yl}methyl)acetamide
5-{1-[(2-fluorophenyl)methyl]-4-hydroxypiperidin-4-yl}-N-(oxolan-2-ylmethyl)-1-benzofuran-2-carboxamide
1-[(1-{3,3-dimethyl-2-methylidenebicyclo[2.2.1]heptane-1-carbonyl}piperidin-3-yl)methyl]pyrrolidin-2-one
methyl 3-{3-[3-oxo-3-(pyrrolidin-1-yl)propyl]piperidine-1-carbonyl}benzoate
1-[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]azetidin-3-amine
1-(2,1,3-benzoxadiazol-5-ylmethyl)-3-(1-ethyl-1H-1,2,3-triazol-4-yl)-1-methylurea
N-benzyl-5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carboxamide
4-[(4-ethoxyphenyl)methyl]-3-[2-oxo-2-(4-phenyl-1,4-diazepan-1-yl)ethyl]piperazin-2-one