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(pentan-2-yl)({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)amine
2-[4-(1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carbonyl)morpholin-3-yl]acetic acid
7-(cyclopropylmethyl)-6-oxo-N-(2-phenylethyl)-2,7-diazaspiro[4.5]decane-2-carboxamide
4-{2-[3-(2-methylpropyl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]ethyl}-3,4-dihydro-2H-1,4-benzoxazin-3-one
ethyl 5-{[(7-oxo-2-propanamido-4,5,6,7-tetrahydro-1,3-benzothiazol-5-yl)formamido]methyl}furan-2-carboxylate
3-(2-amino-1,3-thiazol-4-yl)-1-(7-methoxy-2,3,4,5-tetrahydro-1H-3-benzazepin-3-yl)propan-1-one
2-ethyl-4-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}pyridine
3-(1-methyl-1H-imidazol-2-yl)-1-[1-(oxan-4-yl)piperidine-4-carbonyl]piperidine
2-[1-(2-benzyl-1,3-thiazol-4-yl)-N-methylformamido]-2-(thiophen-2-yl)acetic acid
1-cycloheptyl-4-[4-(piperidine-1-carbonyl)phenoxy]piperidine
4-[(1,5-dimethyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazol-4-yl)methyl]-1-methylpiperazine-2-carboxylic acid
1-(2-aminoethyl)-N-[2-(4,5,6,7-tetrahydro-1-benzothiophen-3-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
3-(1-{[5-methyl-2-(naphthalen-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-2-yl)pyridine
1-[(1-ethylpyrrolidin-2-yl)methyl]-1,2-dihydroquinolin-2-one
5-(1,5-dimethyl-1H-pyrazol-4-yl)-N-[3-(1H-imidazol-1-yl)propyl]-1,2-oxazole-3-carboxamide
4-{[3-(3,4-dimethoxyphenyl)-1H-pyrazol-4-yl]methyl}-1,3-dimethylpiperazin-2-one
(3S,4R)-1-[1-(2-methoxyacetyl)piperidine-4-carbonyl]-4-phenylpyrrolidine-3-carboxylic acid
1-(3-{4-[(3-methylphenyl)methyl]piperazine-1-carbonyl}phenyl)imidazolidin-2-one
2-[2-(1-methyl-1H-imidazol-2-yl)ethyl]-1-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}piperidine
(2R,3R)-1'-(1H-imidazol-4-ylmethyl)-3-(morpholin-4-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
1-(2-oxo-2-{5-propanoyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}ethyl)pyrrolidin-2-one
[(8-methoxyquinolin-5-yl)methyl](methyl)({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)amine
N,N-dimethyl-5-{1-[4-(5-methyl-4H-1,2,4-triazol-3-yl)phenyl]-1H-imidazol-2-yl}-1,3-thiazol-2-amine
2-[9-methoxy-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]pyridine-3-carboxamide
2-{[5-(5-fluoro-2-methylphenyl)-4-(4-methylphenyl)pyrimidin-2-yl]amino}propane-1,3-diol
2-{[3-(3-chlorobenzoyl)piperidin-1-yl]methyl}-6-fluoro-1H-1,3-benzodiazole
2-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}-N-tert-butylbutanamide
[(2-methyl-1,3-thiazol-4-yl)methyl][4-(2-methyl-1H-imidazol-1-yl)butan-2-yl]amine
(4aR,7aS)-1-(2-methoxyethyl)-4-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-{[2-chloro-5-(1H-pyrazol-1-yl)phenyl]formamido}-N,4-dimethylpentanamide
2-methyl-5-{3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyrazine
benzyl N-{1-[(2,3-dihydro-1H-inden-4-yl)carbamoyl]pyrrolidin-3-yl}carbamate
3-(4-chloro-2-methoxy-5-methylphenyl)-1-[(4,6-dimethylpyridin-2-yl)methyl]-1-methylurea
2,3,5-trimethyl-N-[1-(3-methyl-1,2,4-oxadiazol-5-yl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
2-{2-benzyl-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}-6-methylpyridine-3-carbonitrile
N-[(2,3-dichlorophenyl)methyl]-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
(3aS,6aS)-2-[3-(1H-imidazol-2-yl)benzoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-{[6-(4-methoxy-3-methylphenyl)pyridazin-3-yl](methyl)amino}ethan-1-ol
N-cyclohexyl-2-(dimethyl-1,3-thiazol-5-yl)-N-(pyridin-4-ylmethyl)acetamide
N-[(2-chloro-6-fluorophenyl)methyl]-N-cyclopropyl-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
2-(5-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1H-1,2,3,4-tetrazol-1-yl)-N-[2-(6-methylpyridin-2-yl)ethyl]acetamide
2,6-dimethyl-N-(2-methylpropyl)-N-(pyridin-4-ylmethyl)pyridine-4-carboxamide
(1R,2R,6S,7S)-4-(4-cyclopentylpyrimidin-2-yl)-10-oxa-4-azatricyclo[5.2.1.02,6]decane
N-{3-[3-(2-ethylphenoxy)azetidin-1-yl]-3-oxopropyl}-N-methylmethanesulfonamide
N-(1,4-dimethyl-3-phenyl-1H-pyrazol-5-yl)-6-hydroxy-1,4-oxazepane-4-carboxamide
1'-(3-chloro-5-fluorobenzoyl)-5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
(4aS,7aR)-1-[(1-ethyl-1H-imidazol-2-yl)methyl]-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
6-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)-3-(2-fluorophenyl)-1-(pyridin-4-ylmethyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
1-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]-4-(2-methyl-1H-imidazol-1-yl)butan-1-one
N-{[3-(2-fluorophenyl)-1,2-oxazol-5-yl]methyl}-2-[1-(propan-2-yl)piperidin-4-yl]acetamide