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3-(5-amino-1H-1,2,4-triazol-3-yl)-1-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-N-(propan-2-yl)-2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]acetamide
2-cyclopropyl-9-{[2-(2-hydroxyethoxy)phenyl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
2-(2-{1-[3-(5-methyl-1H-1,2,4-triazol-3-yl)propanoyl]piperidin-4-yl}-1H-imidazol-1-yl)acetamide
1-{3-[4-(2-methoxyphenoxy)piperidine-1-carbonyl]piperidin-1-yl}ethan-1-one
N-[(2-ethoxypyridin-3-yl)methyl]-3-phenyl-1H-pyrazole-4-carboxamide
N-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-2-[(1-methyl-1H-indol-3-yl)sulfanyl]acetamide
2-[4-(7-fluoro-2-methylquinoline-4-carbonyl)piperazin-1-yl]pyridine-3-carbonitrile
3-(furan-2-yl)-5-(5-methyl-2H-1,2,3-triazol-4-yl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazole
3-(5-fluoro-1H-1,3-benzodiazol-2-yl)-1-{1-oxa-7-azaspiro[3.5]nonan-7-yl}propan-1-one
4-ethyl-1-methyl-3-[(1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-5-carbonyl}piperidin-4-yl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-2-oxo-1,2-dihydroquinoline-4-carboxamide
{3-[(3-methoxyphenyl)methyl]-1-(quinolin-8-ylmethyl)piperidin-3-yl}methanol
2-(2-methoxyethoxy)-1-{2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}ethan-1-one
4-[(1-cyclopentylpiperidin-4-yl)oxy]-3-methoxy-N-[(1-methyl-1H-pyrazol-4-yl)methyl]benzamide
(3R,4S)-1-[(1-benzyl-1H-imidazol-2-yl)methyl]-3,4-dimethylpiperidin-4-ol
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-N,2,3-trimethylquinoxaline-6-carboxamide
N-methyl-3-{1-[3-(1,2-oxazinan-2-yl)propanoyl]piperidin-3-yl}-N-[2-(pyridin-2-yl)ethyl]propanamide
(2R,3R,6R)-3-(4-fluorophenyl)-5-[(2-propylpyrimidin-5-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
1-{7-[(4-acetylpiperazin-1-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}-2-(3-methylphenyl)ethan-1-one
1,9-dimethyl-4-[2-(2-methyl-1H-1,3-benzodiazol-5-yl)acetyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
4-[(6-methoxypyrimidin-4-yl)amino]-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-2-one
N-[(2-amino-1,3-thiazol-4-yl)methyl]-2-(2,3-difluorophenoxymethyl)-1,3-oxazole-4-carboxamide
N-(3,3-diphenylpropyl)-6-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)-6-azaspiro[2.5]octane-1-carboxamide
N-[(1-ethyl-1H-imidazol-5-yl)methyl]-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
(1R,7S)-N-(1H-imidazol-2-ylmethyl)-N-methyl-3-[(3-methylphenyl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
4-[(8-methoxy-2H-chromen-3-yl)methyl]-1,8-dioxa-4,11-diazaspiro[5.6]dodecane
(4aS,7aR)-1-{2-[cyclopentyl(methyl)amino]acetyl}-4-(2-methoxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N,2-dimethyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]-1,3-thiazole-4-carboxamide
1-[(3aR,5R,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindol-2-yl]-2-(2-chloro-4-fluorophenyl)ethan-1-one
3-[1-(3,6-dimethyl-1-benzofuran-2-carbonyl)piperidin-4-yl]-1-(morpholin-4-yl)propan-1-one
N-{2H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-N-methyl-N'-[2-(propan-2-yl)phenyl]butanediamide
4-{4-[4-(4-methylphenyl)piperazine-1-carbonyl]piperidin-1-yl}-2-[1-(1,3-thiazol-2-yl)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
4-(5-{[2-(pyridin-2-yl)pyrrolidin-1-yl]methyl}-1,3-thiazol-2-yl)morpholine
3-ethyl-3-[2-(1H-pyrazol-1-yl)ethyl]-1-[2-(trifluoromethoxy)phenyl]urea
5-(1-phenoxyethyl)-3-phenyl-1H-1,2,4-triazole
methyl (1S,3S,3aR,6aS)-1-(hydroxymethyl)-5-methyl-4,6-dioxo-3-(1,3-thiazol-2-yl)-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-1-(2-methylpropyl)piperidin-4-amine
1-cyclohexyl-N-(isoquinolin-5-ylmethyl)-N-methyl-1H-1,2,3-triazole-4-carboxamide
{4-[(4-methoxyphenyl)methyl]-1-(thiolan-3-yl)piperidin-4-yl}methanol
3-(4-fluorophenyl)-2-{[1-methyl-3-(2-methylpropyl)-1H-pyrazol-5-yl]formamido}propanoic acid
5-[({1-[3-(4-fluorophenyl)phenyl]piperidin-4-yl}amino)methyl]pyrrolidin-2-one
4-[(2-fluoro-4-methoxyphenyl)methyl]-1-(3-methoxyphenyl)piperazin-2-one
1-(1,3-benzothiazol-2-yl)-3-(piperidin-1-ylmethyl)pyrrolidin-3-ol
1-cyclobutanecarbonyl-3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
6-methyl-2-(2-{2-[4-(methylsulfanyl)phenyl]-1H-imidazol-1-yl}ethyl)-3,4-dihydropyrimidin-4-one
2-{5-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-methyl-1H-1,2,4-triazol-5-yl]-1H-pyrazol-3-yl}pyridine
(1R,2R,6S,7S)-4-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}-10-oxa-4-azatricyclo[5.2.1.02,6]decane
N-(2-oxo-2-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}ethyl)acetamide
1-(2,2-dimethylpropyl)-3-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine