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methyl 4-(2-carbamoylphenyl)benzoate
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-methyl-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
1-{4-[(piperidin-4-ylmethyl)amino]-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
1'-(5-fluoropyrimidin-2-yl)-1-methyl-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
1-{[2-(ethanesulfonyl)-1-(3-phenylpropyl)-1H-imidazol-5-yl]methyl}-3-methylpiperidine
(3aS,6aS)-2-(2,3-dihydro-1,4-benzodioxine-6-sulfonyl)-5-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidin-1-yl]-3-(2-methylphenyl)propan-1-one
N-[(3R,7S,8aS)-3-[(benzylsulfanyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]naphthalene-2-carboxamide
1-[benzyl(methyl)amino]-3-[4-(morpholin-4-ylmethyl)phenoxy]propan-2-ol
2-[2-(propan-2-yl)-1H-imidazol-1-yl]-1-[4-(1H-1,2,4-triazole-3-carbonyl)piperazin-1-yl]propan-1-one
(3S,4R)-1-[2-(3-oxo-2,3-dihydro-1H-indazol-2-yl)acetyl]-4-phenylpyrrolidine-3-carboxylic acid
N-cyclopropyl-1-[2-(2-methoxyphenyl)acetyl]piperazine-2-carboxamide
N-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-2-propyl-1,3-thiazole-4-carboxamide
(1s,4s)-4-({methyl[(5-propyl-1H-pyrazol-3-yl)methyl]amino}methyl)cyclohexan-1-amine
1-{[4-(2,3-dihydro-1,4-benzodioxin-6-yl)phenyl]methyl}-1H-imidazole
(4aS,8aR)-6-(1,3-dihydroxypropan-2-yl)-1-[3-(1H-imidazol-1-yl)propyl]-decahydro-1,6-naphthyridin-2-one
3-ethyl-N-[3-(4-hydroxyphenyl)propyl]-4-methyl-1H-pyrazole-5-carboxamide
ethyl 4-(4-{4-[(pyridin-4-ylmethyl)amino]piperidin-1-yl}benzoyl)piperazine-1-carboxylate
(5S,9aS,9bS)-5-(6-chloro-2H-chromen-3-yl)-2-[(2-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-cyclopropyl-4-{4-[3-(propan-2-yloxy)phenyl]-1H-imidazol-2-yl}pyrrolidin-2-one
6-ethyl-1,5-dimethyl-3-[2-(1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-1,2-dihydropyridin-2-one
2,5-dimethyl-N-[(1-methyl-1H-imidazol-2-yl)(phenyl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
methyl 5-[(4-methoxy-4-methylpentan-2-yl)amino]-3-(oxolane-3-amido)-1-(2-phenylethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-(2-fluorophenyl)-N-(2-methoxyethyl)-2,2-dimethyl-N-(pyridin-2-ylmethyl)cyclopropane-1-carboxamide
1-[3-(2H-1,3-benzodioxol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propane-1,2-dione
2-(4-{[5-(2-chlorophenyl)furan-2-yl]methyl}-1-methylpiperazin-2-yl)ethan-1-ol
1-[1-(3-methyl-5-propyl-1-benzofuran-2-carbonyl)-4-phenylpiperidin-4-yl]ethan-1-one
1-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(1H-pyrrole-2-carbonyl)piperazine
3-(3-fluoro-2,4-dimethylphenyl)-12-methyl-1,2,4,5,10,11-hexaazatricyclo[7.3.0.02,6]dodeca-3,5,7,9,11-pentaene
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)propan-2-yl]-2-(1H-pyrazol-1-yl)benzamide
2-{1-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]pyrrolidin-2-yl}pyridine
7-(2-cyclohexylethyl)-2-(6-methylpyridine-3-carbonyl)-2,7-diazaspiro[4.5]decane
5-{[2-(3-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-N,N-dimethylpyridin-2-amine
N-[3-(furan-2-yl)phenyl]-1-(oxan-4-yl)piperidine-4-carboxamide
3-[(dimethylamino)methyl]-1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxypiperidin-2-one
8-(5-hydroxypyrazine-2-carbonyl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[(3,4-dimethoxyphenyl)methyl]-N-(1-methoxypropan-2-yl)-1H-pyrazole-3-carboxamide
N-(1-{1-[(dimethylcarbamoyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2H-1,3-benzodioxole-5-carboxamide
4-[4-(dimethylamino)-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-N-methyl-4-oxobutanamide
(2H-1,3-benzodioxol-4-ylmethyl)(benzyl)(1,3-thiazol-2-ylmethyl)amine
2-(2-{2-[2-(furan-2-yl)pyrimidin-5-yl]-1H-imidazol-1-yl}ethyl)-1H-1,3-benzodiazole
3-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-9-methoxy-N-[(4-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-[(4-methoxyphenyl)methyl]-4-[2-(methylsulfanyl)pyridine-3-carbonyl]piperazin-2-one
N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]-2,3-dihydro-1,4-benzodioxine-2-carboxamide
N-methyl-N-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-3-(1H-pyrazol-1-ylmethyl)benzamide
ethyl 2-[4-(2-{4-[2-(2-methoxyphenyl)acetamido]-1H-pyrazol-1-yl}acetyl)morpholin-3-yl]acetate
N4-[(5-ethylpyridin-2-yl)methyl]-N4-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
N-{imidazo[1,2-a]pyrimidin-2-ylmethyl}-3-(trimethyl-1H-pyrazol-4-yl)propanamide
4-{5-[3-ethyl-4-(propan-2-yl)piperazine-1-carbonyl]pyridin-2-yl}morpholine
1-[(3S,4R)-3-(dimethylamino)-4-propylpyrrolidin-1-yl]-2-(3-methoxyphenyl)ethan-1-one