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1-{2,4,6-trimethyl-3-[1-(oxan-2-ylmethyl)-1H-imidazol-2-yl]phenyl}ethan-1-one
9-[4-(benzyloxy)butanoyl]-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
(1-{[2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)methanol
6-{2-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]-2-oxoethyl}-3,4-dihydro-2H-1,4-benzoxazin-3-one
1-tert-butyl-4-[4-(2-phenoxyethyl)piperazine-1-carbonyl]pyrrolidin-2-one
N-[2-(dimethylsulfamoyl)ethyl]-4-(piperidin-3-yl)benzamide
N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}-2-hydroxypyridine-3-carboxamide
N-cycloheptyl-3-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]propanamide
8-chloro-2-{[(2-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-4-yl)amino]methyl}quinolin-4-ol
4-(2-hydroxyacetyl)-5-methyl-1-(2-phenylphenyl)piperazin-2-one
3-(pyrimidin-4-yl)quinoline
1-(4-chlorophenyl)-N-ethyl-N-[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]cyclopropane-1-carboxamide
(3aR,6aR)-N-[3-(1H-1,3-benzodiazol-2-yl)propyl]-2-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
1-{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}-3-(2-methoxyethyl)piperidine-3-carboxylic acid
1-(oxolane-3-carbonyl)-4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
8-(4-fluoro-2-methylbenzenesulfonyl)-5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine
N-[(3S,4R)-1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)-4-propylpyrrolidin-3-yl]methanesulfonamide
1-[4-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(2-methoxyphenyl)ethan-1-one
(2S,3R)-2-amino-1-[4-(dimethylamino)-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-3-hydroxybutan-1-one
1-{4-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]piperazin-1-yl}-3-(1H-1,2,4-triazol-1-yl)propan-1-one
2-{[(3-chlorophenyl)methyl](methyl)amino}-2-(4-methanesulfonylphenyl)acetic acid
2-cyclopentyl-1-{4-[3-(morpholine-4-carbonyl)phenoxy]piperidin-1-yl}ethan-1-one
[2-(1H-imidazol-1-yl)-1-phenylethyl](propan-2-yl)amine
3-[({3-methyl-1-[2-(piperidin-1-yl)ethyl]-1H-pyrazol-4-yl}methyl)amino]-2,3-dihydro-1λ6-thiophene-1,1-dione
1-cyclopropyl-3-[2-oxo-2-(piperidin-1-yl)ethyl]-3-[3-(trifluoromethyl)phenyl]pyrrolidine-2,5-dione
(benzylsulfamoyl)({[1-(pyrrolidin-1-yl)cyclopentyl]methyl})amine
1-[4-({[2-(cyclohex-1-en-1-yl)ethyl]amino}methyl)-2-methoxyphenoxy]-3-(morpholin-4-yl)propan-2-ol
5-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-N-[2-(dimethylamino)ethyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
(1R,5S,8R)-N,N-dimethyl-3-(1,3-thiazol-4-ylmethyl)-3-azabicyclo[3.2.1]octan-8-amine
3-({5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}methyl)-6-methoxy-1,2-dihydroquinolin-2-one
N-[(4-methylphenyl)methyl]-1-[2-(pent-4-enamido)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-(2-{3-methyl-7-oxo-7H-[1,3]thiazolo[3,2-b][1,2,4]triazin-6-yl}phenyl)-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
2-(4-ethylpiperazin-1-yl)-1-{3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}ethan-1-one
(1S,5R)-6-propyl-3-(quinoline-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-{4-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-(thiophen-3-ylmethyl)piperazin-2-yl}ethan-1-ol
1-{1,9-dioxaspiro[5.5]undecan-4-yl}-4-(2-methylphenyl)piperazine
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-1,3,6-trimethyl-1H-pyrazolo[3,4-b]pyridine-4-carboxamide
1-(4-fluorophenyl)-4-{1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperidin-3-yl}piperazine
1-[(3-fluorophenyl)methyl]-4-[2-(methylamino)pyridine-3-carbonyl]piperazin-2-one
N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1-methylazepane-2-carboxamide
1-(2-methoxyphenyl)-3-{1-[1-(3-phenylprop-2-ynoyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
2-[4-({4-[(3,4-difluorophenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)phenoxy]ethan-1-ol
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-2-(4-phenylpiperidin-1-yl)acetamide
2-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyridine-4-carboxamide
3-[3-ethyl-4-(4-fluorophenyl)-1-methyl-1H-pyrazol-5-yl]-1-methyl-1-[(4-methyl-1H-imidazol-2-yl)methyl]urea
methyl[(1-methyl-1H-pyrazol-4-yl)methyl][(4-{[1-(thiophene-2-carbonyl)piperidin-4-yl]oxy}phenyl)methyl]amine
2-{[3-(dimethylamino)propyl](methyl)sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
(3S,4R)-4-(2,3-dimethoxyphenyl)-1-[(2-fluoro-3-methylphenyl)methyl]pyrrolidine-3-carboxylic acid
5-[2-(dimethylamino)-5,6-dimethylpyrimidin-4-yl]-N-methyl-2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-(1-benzylpiperidin-4-yl)-1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-2,6-dimethyl-4-oxo-1,4-dihydropyridine-3-carboxamide