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5-methyl-5-phenyl-1-[2-(pyrazin-2-yl)ethyl]piperidin-2-one
1-cyclohexyl-6-hydroxy-4-(1-methylpiperidin-4-yl)-1,4-diazepan-2-one
3-cyano-N-[4-ethoxy-3-(trifluoromethyl)phenyl]piperidine-1-carboxamide
6-amino-N-[1-(pyridin-4-yl)propyl]pyridine-2-carboxamide
N-(1-benzothiophen-5-ylmethyl)-2-(1,4-dimethylpiperazin-2-yl)acetamide
4-{[4-(benzyloxy)-3-methoxyphenyl]methyl}-1,4-oxazepan-6-ol
3-{2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl}-3-phenyl-1-[3-(pyridin-3-yloxy)propyl]pyrrolidine-2,5-dione
1-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-3-(1-propyl-1H-1,2,3-triazol-4-yl)urea
3-(2,5-dioxoimidazolidin-4-yl)-N-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]propanamide
4-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1-methyl-3-(pyridin-3-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-{2-azatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-5-yl}-3-[(3S,4R)-1-[(2-chlorophenyl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]propanamide
1-(2,3-dimethoxyphenyl)-2-(2,5-dimethylfuran-3-carbonyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-1,9-dioxaspiro[5.5]undecan-4-amine
(2S,4S)-1-[(3-chlorophenyl)methyl]-4-[(4,6-dimethylpyrimidin-2-yl)sulfanyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-[(3R,4R)-3-hydroxy-1-[2-(3-methoxyphenyl)acetyl]piperidin-4-yl]pyrazine-2-carboxamide
N-[(3-methylphenyl)methyl]-2-[2-(2-oxopyrrolidin-1-yl)propanamido]benzamide
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
ethyl 4-{3-[2-(dimethylamino)ethyl]-1-ethyl-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-8-yl}piperidine-1-carboxylate
3-{1-[5-(methoxymethyl)thiophene-2-carbonyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)propanamide
1-[(4-fluorophenyl)methyl]-4-{2-methylimidazo[1,2-a]pyridine-6-carbonyl}-1,4-diazepane
3-(1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}piperidin-3-yl)-N-[(2-fluorophenyl)methyl]propanamide
4-({8-methyl-2,8-diazaspiro[4.5]decan-2-yl}methyl)benzoic acid
N-[(1-methyl-1H-imidazol-2-yl)(phenyl)methyl]-2-(methylamino)-1,3-thiazole-4-carboxamide
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
5-(2-methylpropyl)-N-[2-(4,5,6,7-tetrahydro-2H-indazol-3-yl)ethyl]-1,2-oxazole-3-carboxamide
5-methyl-N-[2-(pyridin-2-ylsulfanyl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
5-methyl-2-(3-methylthiophen-2-yl)-4-[2-(pyrrolidine-1-carbonyl)phenoxymethyl]-1,3-oxazole
2-methyl-N-[1-(3,4,5-trimethoxyphenyl)ethyl]thieno[2,3-d]pyrimidin-4-amine
[(2R)-1-(3-{2-azaspiro[4.4]nonane-2-carbonyl}benzenesulfonyl)pyrrolidin-2-yl]methanol
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-2-(3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetamide
N-{2-[(2-methylprop-2-en-1-yl)oxy]phenyl}-4-(pyridin-3-ylmethoxy)piperidine-1-carboxamide
(3R,9aR)-8-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-3-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-(5-{1-[2-(3-methoxyphenyl)ethyl]-1H-1,2,3-triazol-4-yl}pyrimidin-2-yl)morpholine
1-[4-(hydroxymethyl)piperidin-1-yl]-3-(2-methylphenyl)-3-phenylpropan-1-one
1-[(4-methoxyphenyl)methyl]-N-[2-(4-methoxyphenyl)phenyl]piperidine-3-carboxamide
ethyl[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]{[3-(methylsulfanyl)phenyl]methyl}amine
(4aR,7aS)-1-(2-hydroxyethyl)-4-[2-(2,6,6-trimethylcyclohex-1-en-1-yl)ethyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[(2-methoxyethyl)carbamoyl]-4-(pyrazin-2-yl)-1,4-diazepane-6-carboxylic acid
4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1-(propane-2-sulfonyl)-1,4-diazepan-5-one
1-(1-benzylpiperidin-4-yl)-N-(2-methoxyethyl)piperidine-3-carboxamide
N-ethyl-4-[(6-methoxypyrimidin-4-yl)amino]piperidine-1-carboxamide
8-[2-(cyclopent-2-en-1-yl)acetyl]-2-(3-methoxypropyl)-2,8-diazaspiro[4.5]decan-3-one
1-{3-[4-(methylsulfanyl)benzoyl]piperidin-1-yl}-3-(1,2-oxazolidin-2-yl)propan-1-one
2-[3-(1-methyl-1H-1,3-benzodiazol-2-yl)-1H-pyrazol-1-yl]-N-[1-(propan-2-yl)-1H-pyrazol-5-yl]acetamide
[3-(3-phenylpropyl)-1-[(2,4,5-trimethoxyphenyl)methyl]piperidin-3-yl]methanol
N-({1-[(3-methoxyphenyl)methyl]-1H-1,2,4-triazol-5-yl}methyl)acetamide
N-[1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]cyclopropanesulfonamide
N-{[1-(4-formylbenzoyl)piperidin-3-yl]methyl}-2,3-dimethoxybenzamide
2-{[(5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}furan-2-yl)methyl]sulfanyl}pyrimidine
1-methanesulfonyl-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]piperidin-4-amine