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N-(1-{[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl}pyrrolidin-3-yl)acetamide
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}acetamide
propan-2-yl 4-chloro-3-(6-oxo-1,6-dihydropyrimidine-5-amido)benzoate
methyl 2-[3-(2-chlorophenyl)-N-methyl-3-phenylpropanamido]acetate
N-(1-butyl-1H-pyrazol-5-yl)-2-(4-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidine-1-carboxamide
5-(1,2-oxazol-3-yl)-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}thiophene-2-sulfonamide
methyl 3-(2,1,3-benzothiadiazol-5-ylmethyl)-7-oxo-9-(pyridin-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
5-[({1-azabicyclo[2.2.2]octan-3-yl}(pyridin-3-ylmethyl)amino)methyl]-N,N-dimethylfuran-2-carboxamide
N-[1-(2-chlorophenyl)ethyl]-3-(4,5-dimethyl-1H-pyrazol-3-yl)propanamide
8-[(2-fluoro-5-methoxyphenyl)methyl]-2-(3-hydroxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
4-(2,5-dimethoxyphenyl)-2-[(4-phenylpiperazin-1-yl)methyl]phenol
{[3-(2,5-dimethylthiophen-3-yl)-1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amine
3-(furan-2-yl)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]benzamide
8-(oxolan-3-yl)-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-(2-fluoro-6-methoxyphenyl)pyridine-4-carbonitrile
1-{spiro[2.3]hexane-1-carbonyl}-4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
5-ethyl-N4-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]pyrimidine-2,4-diamine
3-[(2-fluorophenyl)formamido]-N-[(5-methylpyrazin-2-yl)methyl]propanamide
3-(4-{1-[2-(piperidin-1-yl)ethyl]-1,2,3,6-tetrahydropyridin-4-yl}-1H-pyrazol-1-yl)-1λ6-thiolane-1,1-dione
1-[3-(methylsulfanyl)butyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-methyl-N-[2-(4-methyl-1H-pyrazol-1-yl)ethyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
3-{[ethyl(pyridin-4-ylmethyl)amino]methyl}-1-{[3-(trifluoromethyl)phenyl]methyl}-1H,2H,6H,7H,8H-cyclopenta[g]quinolin-2-one
4-[(2-fluoro-5-methoxyphenyl)methyl]morpholine-2-carboxamide
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)-1H-pyrazole-4-carboxamide
2,3-dimethyl-5-{4-[(methylsulfanyl)methyl]piperidine-1-carbonyl}pyridine
N-{[7-methoxy-2-(3-methylphenyl)quinolin-3-yl]methyl}-N-(2-methoxyethyl)-2-methyl-1,3-thiazole-4-carboxamide
3-(2,3-dihydro-1,4-benzodioxin-6-ylsulfanyl)-N-(quinolin-3-ylmethyl)propanamide
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-[(1-ethyl-1H-pyrazol-4-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
N-ethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-3-(2-oxoazepan-1-yl)propanamide
N-methyl-2-[1-(2-methylpropyl)-3-oxopiperazin-2-yl]-N-(quinolin-8-ylmethyl)acetamide
N-[3,3-dimethyl-1-(pyridin-3-yl)butyl]pyrimidin-4-amine
2-fluoro-N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-5-sulfamoylbenzamide
N-{[7-(4-chlorophenyl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-methoxypropanamide
2-(quinolin-6-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
1-[(1-methylpiperidin-3-yl)methyl]-4-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}piperazine
[5-(2,6-dimethoxypyrimidin-4-yl)-2-fluorophenyl]methanol
methyl 2-oxo-8-(3-phenylpropyl)-1-(prop-2-en-1-yloxy)-1,8-diazaspiro[4.5]decane-4-carboxylate
(3-{[(1H-indol-4-ylmethyl)amino]methyl}-2,4,6-trimethylphenyl)methyl acetate
2-(6-methoxynaphthalen-2-yl)-N-(1-methyl-1H-1,2,3-triazol-4-yl)morpholine-4-carboxamide
3-[(4-cyclopentanecarbonyl-6-hydroxy-1,4-diazepan-1-yl)methyl]benzonitrile
ethyl 2-[1-cyclobutyl-4-(4-fluorobenzenesulfonyl)piperidin-4-yl]acetate
N-cyclopentyl-4-{4-[(thiophen-3-ylmethyl)amino]piperidin-1-yl}benzamide
3-(azepan-1-ylmethyl)-N,8-dimethyl-N-(2-phenylethyl)imidazo[1,2-a]pyridine-2-carboxamide
9-[2-amino-6-(dimethylamino)pyrimidin-4-yl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-[(2-carbamoylethyl)sulfamoyl]-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]benzamide
4-(2-methoxyethoxy)-1-[3-(5-methylfuran-2-yl)butyl]piperidine
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-3-(1H-pyrazol-4-yl)propanamide
methyl 6-{3-[(2,3-dihydro-1,4-benzodioxin-6-yl)amino]piperidine-1-carbonyl}pyridine-3-carboxylate
1-(azepan-1-yl)-2-[3-(2H-1,3-benzodioxole-5-carbonyl)piperidin-1-yl]ethan-1-one
1-(pent-2-yn-1-yl)-4-phenyl-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one