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8-(1,3-benzoxazol-2-yl)-2-[2-(1H-imidazol-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
N-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-N,5-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
1-(4-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}piperidin-1-yl)ethan-1-one
1-(6-oxo-1,6-dihydropyridine-3-carbonyl)-3-[(2E)-3-phenylprop-2-en-1-yl]piperidine-3-carboxylic acid
(5S,9aS,9bS)-5-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-yl}-2-(pyridin-3-ylmethyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
7-cyclohexyl-2-[2-(2-methoxyethoxy)acetyl]-2,7-diazaspiro[4.5]decan-6-one
methyl 3-[4-(2-fluorobenzoyl)-2-oxo-6-(pyridin-4-ylmethoxy)-1,4-diazepan-1-yl]propanoate
2-[4-(dimethylamino)phenyl]-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]acetamide
2-({[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}amino)-N-(4-methylphenyl)propanamide
3-ethyl-8-[4-(2-methylpropyl)benzoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[3-({5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)propyl]piperidin-3-ol
N'-({1-[(2-fluorophenyl)methyl]pyrrolidin-3-yl}methyl)ethanediamide
3-{5-[2-(methylsulfanyl)benzoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
methyl 1-(2-methoxyethyl)-5-[(naphthalen-1-ylmethyl)amino]-3-(3-phenylpropanamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-[(2R,3R)-2-methoxy-1'-(quinolin-8-ylmethyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(thiophen-2-yl)acetamide
2-amino-N-[(3R,4S)-4-cyclopropyl-1-(2-hydroxyethyl)pyrrolidin-3-yl]-4-methyl-1,3-thiazole-5-carboxamide
N-cyclopentyl-4-oxo-4-[4-(pyrimidin-2-yl)-1,4-diazepan-1-yl]butanamide
4-(hydroxymethyl)-1-(pyridine-3-sulfonyl)azepan-4-ol
methyl 5-[(dimethyl-1,2-oxazol-4-yl)carbamoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
N-methyl-N-[1-(pyridin-2-yl)propan-2-yl]-2-(2,3,4-trifluorophenyl)acetamide
3-[2-(6-hydroxy-1,4-oxazepan-4-yl)-2-oxoethyl]-5-methyl-2,3-dihydro-1,3-benzoxazol-2-one
1-(2-chlorophenyl)-5-methyl-4-[3-(5-methyl-1H-pyrazol-1-yl)propanoyl]piperazin-2-one
6-(2,5-dimethylfuran-3-yl)-N-(1H-imidazol-2-ylmethyl)-7-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
(2S,4S,5R)-5-(2-fluorophenyl)-1-methyl-4-[(oxan-4-ylmethyl)carbamoyl]pyrrolidine-2-carboxylic acid
3-[(7-chloro-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)methyl]-6-methyl-4H-chromen-4-one
7-fluoro-4-[1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole-5-carbonyl]-1,2,3,4-tetrahydroquinolin-2-one
1-{[3-(4-benzylpiperidine-1-carbonyl)-1,2-oxazol-5-yl]methyl}piperidin-4-ol
N-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-8-fluoroquinoline-2-carboxamide
N-[2-(diethylamino)ethyl]-N-ethyl-2-[3-(2-methylphenyl)-2,5-dioxo-1-(pyridin-4-ylmethyl)pyrrolidin-3-yl]acetamide
{5-[3-cyclopropyl-1-(2,4-difluorophenyl)-1H-1,2,4-triazol-5-yl]furan-2-yl}methanol
1-[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]propane-1,2-dione
[(3R,4R)-1-(2,6-difluoro-3-methoxybenzoyl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
{1-[3-(3-fluoropyridin-2-yl)phenyl]ethyl}dimethylamine
1-[2-(methylamino)pyridine-3-carbonyl]-4-(3-methylbut-2-en-1-yl)-1,4-diazepan-6-ol
3-chloro-N-(1H-imidazol-2-ylmethyl)-4-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-methylbenzamide
4-[4-(2-methoxypyridin-3-yl)phenyl]-4-oxobutanoic acid
methyl 6-[(3S,4R)-3-methanesulfonamido-4-(propan-2-yl)pyrrolidin-1-yl]pyrazine-2-carboxylate
3-[5-(6-aminopyridine-3-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
N,N-dimethyl-2-[6-methyl-2-oxo-4-(trifluoromethyl)-1,2-dihydropyridin-1-yl]acetamide
2-{1-[1-(2,6-difluorobenzoyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}propan-2-ol
5-[benzyl(methyl)amino]-2-(2-hydroxyethyl)-2,3-dihydropyridazin-3-one
N-[(1R,3R)-3-aminocyclopentyl]-1-ethyl-3-methyl-1H-pyrazole-4-sulfonamide
1-{2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]acetyl}-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-{8-benzyl-2,8-diazaspiro[5.5]undecan-2-yl}-2-[(2-methoxyethyl)(methyl)amino]ethan-1-one
N-{[7-(2H-1,3-benzodioxole-5-carbonyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}-3-fluorobenzamide
N-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
7-methyl-2-(1,3-thiazol-2-yl)-1H-1,3-benzodiazole
N-[3-(aminomethyl)-5-({5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}carbamoyl)phenyl]pyridine-2-carboxamide
(4aR,7aS)-4-(2-methoxypyridine-3-carbonyl)-N,N-dimethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
N3-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]-N5-cyclooctyl-1-(2-methoxyethyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide