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methyl 1-[5-methyl-4-(4-methylpiperazin-1-yl)thieno[2,3-d]pyrimidine-6-carbonyl]piperidine-2-carboxylate
5-{2-[4-(3-methoxyphenyl)-3-oxopiperazin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
2-(3-fluorophenyl)-2-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]formamido}acetic acid
methyl[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]{[3-(1H-pyrazol-1-yl)phenyl]methyl}amine
dimethyl({3-[2-(1-{4H-thieno[3,2-b]pyrrole-5-carbonyl}piperidin-3-yl)-1H-imidazol-1-yl]propyl})amine
N-cyclooctyl-1-(prop-2-en-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-{3-[2-(3-fluorophenyl)ethyl]piperidin-1-yl}propanoic acid
N-[4-(1H-pyrazol-1-yl)phenyl]-6-[2-(pyridin-4-ylsulfanyl)acetyl]-6-azaspiro[2.5]octane-1-carboxamide
3-({[2-(3-chlorophenyl)-7-methylquinolin-3-yl]methyl}amino)-1λ6-thiolane-1,1-dione
1-[4-({4-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperazin-1-yl]ethan-1-one
5-[2-(ethanesulfinyl)ethyl]-1-(2-methoxyphenyl)-3-(propan-2-yl)-1H-1,2,4-triazole
3-[(3S,4R)-1-benzyl-4-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-3-yl]-N-(3-methoxyphenyl)propanamide
4-[5-chloro-2-(piperidine-1-carbonyl)phenoxy]-1-(cyclohex-3-en-1-ylmethyl)piperidine
N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-2-(thiophen-3-yl)acetamide
methyl (2S,4R)-1-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-4-(4-fluorobenzamido)pyrrolidine-2-carboxylate
{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}(methyl)[(4-methyl-1H-imidazol-2-yl)methyl]amine
5-ethoxy-N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]furan-2-carboxamide
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-2-methyl-2-(thiophen-2-ylformamido)propanamide
3-{[benzyl(methyl)amino]methyl}-7-methyl-1-(pyridin-2-ylmethyl)-1,2-dihydroquinolin-2-one
(5S,9aS,9bS)-2-methyl-5-(3,4,5-trimethoxyphenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-[1-(4-chloro-1,5-dimethyl-1H-pyrazole-3-carbonyl)piperidin-4-yl]-2-phenylethan-1-ol
N-[2-(1-hydroxycyclopentyl)ethyl]-N,3,5,7-tetramethyl-1H-indole-2-carboxamide
1-[3-(1-oxo-2,3-dihydro-1H-isoindol-2-yl)propanoyl]-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
2-{3-[3-methyl-1-(quinolin-8-yl)-1H-1,2,4-triazol-5-yl]phenoxy}acetamide
2,3-dimethyl-7-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
N-benzyl-4-oxo-5-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
N-[(1R,3R)-3-aminocyclopentyl]-4-(3,5-dimethyl-1H-pyrazol-1-yl)butanamide
1-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]-4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-5-one
7-cyclopropanecarbonyl-N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-[(2-butyl-1H-imidazol-4-yl)methyl]-4-(pyridin-3-yl)piperazine
methyl 4-{[2-(dimethylamino)ethyl]({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)carbamoyl}butanoate
5-[1-(2-oxo-2-phenylacetyl)piperidin-4-yl]-5-(pyridin-3-yl)-3-(thiophen-3-ylmethyl)imidazolidine-2,4-dione
7,7-dimethyl-2-(2-methylphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-7-(2-phenylethyl)-2,7-diazaspiro[4.5]decane
4-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-[(4-methoxyphenyl)methyl]-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
2-(benzyloxy)-N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}acetamide
N-[1-(3-fluorophenyl)-4-(propan-2-yloxy)-1H-indazol-3-yl]-2-(2-oxopyrrolidin-1-yl)acetamide
1-{[3-(3-fluorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidine-3-carboxamide
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-1,3-oxazole-4-carboxamide
1-{3-[({[5-(methoxymethyl)furan-2-yl]methyl}amino)methyl]pyridin-2-yl}piperidin-3-ol
2-(2-oxo-2-{4-[2-(oxolan-2-yl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}ethyl)-4-phenyl-1,2-dihydrophthalazin-1-one
4-{3-cyclopentyl-1-[(4-fluorophenyl)methyl]-1H-1,2,4-triazol-5-yl}-1λ6-thiane-1,1-dione
1-[3-(morpholin-4-yl)propyl]-5-{4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carbonyl}piperidin-2-one
2-cyclooctyl-4-{3-[(2S)-2-(hydroxymethyl)pyrrolidine-1-carbonyl]piperidin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
3-{[3-(N-methylacetamido)pyrrolidin-1-yl]methyl}-N-(5-methylpyridin-3-yl)benzamide
1-{1-[(2-methylphenyl)methyl]piperidin-4-yl}-N-(oxan-4-yl)piperidine-4-carboxamide
2-cyclopentyl-N-cyclopropyl-N-{[2-(4-hydroxypiperidin-1-yl)-8-methylquinolin-3-yl]methyl}-2-phenylacetamide
N-[4-(4-{methyl[1-(4-methyl-1,3-thiazol-2-yl)ethyl]amino}piperidin-1-yl)phenyl]-2-phenoxyacetamide
N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-2,5-dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
1-[2-(furan-2-yl)azepan-1-yl]-4-(2-methyl-1H-imidazol-1-yl)butan-1-one