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3-[2-(4-hydroxypiperidin-1-yl)-2-oxoethyl]-4-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperazin-2-one
4-({ethyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amino}methyl)-N-(1,3-thiazol-2-yl)benzamide
(2S,4S)-4-amino-N,N-diethyl-1-(5-phenyl-1,3,4-thiadiazol-2-yl)pyrrolidine-2-carboxamide
2-(4-{[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenyl]methyl}-1-(3-methylbutyl)piperazin-2-yl)ethan-1-ol
2-(1-butyl-1H-pyrazol-4-yl)-6,8-dimethyl-4-(pyrrolidine-1-carbonyl)quinoline
2-[methyl(piperidin-4-yl)amino]-1-[2-methyl-4-(4-methylphenyl)piperazin-1-yl]ethan-1-one
3,5-dimethyl-N-[3-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide
1-{4-[4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]phenyl}imidazolidine-2,4-dione
5-chloro-2-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]phenol
2-[(2S,4R)-2-(diethylcarbamoyl)-4-(dimethyl-1,3-oxazole-5-amido)pyrrolidin-1-yl]acetic acid
2-{methyl[2-(morpholin-4-yl)ethyl]amino}-2-[4-(1H-pyrazol-5-yl)phenyl]acetic acid
4-({[3,3-dimethyl-1-(pyrrolidin-1-yl)butan-2-yl]amino}methyl)-4-ethylhexanenitrile
1-{[1-(2,3-dihydro-1H-inden-4-yl)-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl]methyl}pyrrolidin-2-one
4-[1-(6-ethoxy-4-methylquinazolin-2-yl)piperidine-4-carbonyl]-3-(4-fluorophenyl)piperazin-2-one
1-{2-[5-(morpholine-4-carbonyl)thiophen-2-yl]pyrrolidin-1-yl}ethan-1-one
2-(3-chlorophenoxy)-1-{4-[2-(methoxymethyl)-3H-imidazo[4,5-b]pyridin-3-yl]piperidin-1-yl}propan-1-one
1-[1-(2,2-dimethylpropyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
N,1,6-trimethyl-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-(1-cyclopropanecarbonylpiperidin-4-yl)-2-(oxolan-2-yl)-5-(trifluoromethyl)-1H-1,3-benzodiazole
5-(1-benzofuran-2-yl)-N-{[1-(morpholin-4-yl)cyclohexyl]methyl}-1,2,4-triazin-3-amine
5-(3-fluorophenoxymethyl)-N-(oxolan-2-ylmethyl)-1H-pyrazole-3-carboxamide
4-cyclopentyl-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]pyrimidin-2-amine
[3-({1-[5-(morpholin-4-ylmethyl)furan-3-carbonyl]pyrrolidin-3-yl}methyl)phenyl]methanol
2-[ethyl({[(3R,4R)-1-(7-fluoro-3-methyl-1H-indole-2-carbonyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl})amino]ethan-1-ol
N-benzyl-N,1-dimethyl-5-[methyl(1,3-thiazol-4-ylmethyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
[(6-chloropyridin-3-yl)methyl](methyl){[5-(oxan-2-yl)furan-2-yl]methyl}amine
N-(furan-2-ylmethyl)-4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-(prop-2-yn-1-yl)benzamide
2-[4-(cyclopropylmethyl)-5-oxo-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]-1,4-dihydroquinolin-4-one
1-[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propan-1-one
1-({1-[(2-methoxyphenyl)carbamoyl]piperidin-3-yl}methyl)-1H-1,2,3-triazole-4-carboxylic acid
diethyl({3-[2-(3-methyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]pyrazolo[1,5-a]pyrimidin-6-yl}methyl)amine
N-propyl-N-(pyridin-3-ylmethyl)-2-(pyridin-4-yl)quinoline-4-carboxamide
4-{[5-(1-methyl-1H-1,3-benzodiazol-2-yl)furan-2-yl]methyl}-1,4-oxazepan-6-ol
ethyl 4-{1-[(2-chlorophenyl)methyl]piperidin-3-yl}piperazine-1-carboxylate
N-[(2S,4R,6R)-2-(2,1,3-benzothiadiazol-4-yl)-6-cyclohexyloxan-4-yl]acetamide
(2S,4R)-1-[3-ethoxy-4-(prop-2-en-1-yloxy)benzoyl]-4-hydroxypyrrolidine-2-carboxylic acid
1-(4-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}phenyl)pyrrolidin-2-one
N,2,3-trimethyl-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]quinoxaline-6-carboxamide
3-methyl-7-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
4-(2-methoxyphenoxy)-1-[(trimethyl-1H-pyrazol-4-yl)methyl]piperidine
(2S,4S)-4-amino-1-{2-[cyclopentyl(methyl)amino]acetyl}-N-ethylpyrrolidine-2-carboxamide
N-[(2R,3R)-1'-(5-methylthiophene-2-carbonyl)-2-(pyridin-3-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
N,N-diethyl-2-({4-[3-(furan-2-yl)benzoyl]-1-[(4-methoxyphenyl)methyl]-2-oxo-1,4-diazepan-6-yl}oxy)acetamide
9-(butane-2-sulfonyl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-(1-benzothiophen-5-ylmethyl)-2-(ethylamino)pyrimidine-5-carboxamide
4-methyl-N-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]-3-(2-oxoimidazolidin-1-yl)benzamide
[(3R,4R)-1-(2,3-dimethoxybenzoyl)-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
N-[2-(pyridin-2-ylsulfanyl)ethyl]-1-(pyrimidin-2-yl)piperidin-4-amine
5-[(2-methyl-1,3-oxazol-4-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
(2R,3R,6R)-3-(4-fluorophenyl)-N,N-dimethyl-1,5-diazatricyclo[5.2.2.02,6]undecane-5-sulfonamide