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4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]-1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]piperidine
4-hydroxy-N,2-dimethyl-N-{3-[(4-methylphenyl)sulfanyl]propyl}pyrimidine-5-carboxamide
5-methyl-N-[1-(6-methylpyridin-2-yl)propan-2-yl]-1-[4-(pyridin-3-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
2-(3-{[(butan-2-yl)(pyridin-3-ylmethyl)amino]methyl}-1H-indol-1-yl)acetamide
[(3R,4R)-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}-1-(4-methoxy-3-methylbenzoyl)pyrrolidin-3-yl]methanol
2-(2-chloro-4-{[cyclopropyl(pyridin-2-ylmethyl)amino]methyl}phenoxy)acetamide
(3S,4S)-1-{[4-(4-hydroxybut-1-yn-1-yl)phenyl]methyl}-4-(morpholin-4-yl)pyrrolidin-3-ol
1-(4-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-methyl-2-phenylpropan-1-one
1-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]-4-(2-methyl-1H-imidazol-1-yl)piperidine-4-carboxylic acid
4-[4-(dimethylamino)-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-6-(2-methylpropyl)-1,2-dihydropyrimidin-2-one
1,1,1-trifluoro-3-{3-[3-(pyrimidin-5-yl)phenyl]-1H-pyrazol-1-yl}propan-2-ol
6-(3-fluoro-4-methoxyphenyl)-N-[1-(hydroxymethyl)cyclopentyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
3-(3,4-difluorophenyl)-N-[2-(pyridin-3-yl)ethyl]propanamide
N-(2-fluorophenyl)-2-{3-[3-(pyrimidin-5-yl)phenyl]-1H-pyrazol-1-yl}acetamide
3-{imidazo[1,2-a]pyridin-2-yl}-1-{2-[5-(propan-2-yl)-1,2-oxazol-3-yl]pyrrolidin-1-yl}propan-1-one
N-[(2-methyl-1,3-thiazol-4-yl)methyl]-2-oxo-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
2-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]-1,2-oxazolidin-4-ol
1-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
{8-methyl-2-[4-(piperidine-1-carbonyl)piperidin-1-yl]quinolin-3-yl}methanol
1-[(3S,5S)-5-[1-cyclohexyl-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylic acid
2-[(4aR,7aS)-6,6-dioxo-4-(1,3-thiazol-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}(oxolan-2-ylmethyl)(pyridin-4-ylmethyl)amine
ethyl 4-[4-(3-hydroxy-3-methylbutyl)benzamido]piperidine-1-carboxylate
(1R,5R)-6-(cyclobutylmethyl)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-(1-{dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}azetidin-3-yl)-3,5-dimethyl-1H-pyrazole
8-(2,2-dimethylpropanoyl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
4-[1-(3,4-difluorobenzoyl)piperidin-4-yl]-5-(3-methylphenyl)-2-(pyridin-4-yl)pyrimidine
2-amino-N-(2-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)-6-(propan-2-yl)pyrimidine-4-carboxamide
1-[(2,5-dimethylphenyl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-[4-({[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]carbamoyl}methoxy)phenyl]propanamide
2-[(1-ethyl-1H-pyrazol-4-yl)sulfonyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
3-(2-oxo-2-{3-[5-phenyl-2-(pyridin-4-yl)pyrimidin-4-yl]piperidin-1-yl}ethyl)-2,3-dihydro-1H-isoindol-1-one
N-[(4-methoxyphenyl)methyl]-2-methyl-N-(oxolan-2-ylmethyl)imidazo[1,2-a]pyridine-6-carboxamide
[4-(2-phenoxyethyl)-1-[3-(1H-pyrazol-1-yl)propyl]piperidin-4-yl]methanol
4-[3-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]pyridin-2-amine
2-(1-{1-[1-(3-methylphenyl)piperidin-4-yl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)propan-2-ol
(2S,4R)-4-amino-N,N-diethyl-1-[2-(2-methyl-1H-1,3-benzodiazol-5-yl)acetyl]pyrrolidine-2-carboxamide
1-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]-3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidine
3-(2-ethyl-1H-imidazol-1-yl)-1-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]propan-1-one
N-(1-methanesulfonylpiperidin-4-yl)-2-(1H-pyrrol-1-yl)pentanamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[5,8-dimethoxy-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}-4-methoxybenzamide
4-(piperidin-3-ylmethyl)-N-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}benzamide
methyl 2-(7-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)benzoate
(4aR,7aS)-1-[2-(dimethylamino)acetyl]-4-[2-oxo-2-(piperidin-1-yl)ethyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-(3-methylphenyl)ethan-1-one
3-chloro-N-methyl-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]thiophene-2-carboxamide
ethyl 2-[4-({[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]carbamoyl}amino)phenyl]acetate
N-[1-(hydroxymethyl)cycloheptyl]quinoxaline-5-carboxamide
2-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
(4S)-3-[2-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)-2-oxoethyl]-4-(propan-2-yl)-1,3-oxazolidin-2-one