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2-{2-[4-(1H-pyrazol-5-yl)phenyl]phenyl}ethan-1-amine
3-[(1R,5S)-3,8-diazabicyclo[3.2.1]octan-3-ylmethyl]-N-(1H-indazol-6-yl)benzamide
2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)-N-(2,2,2-trifluoroethyl)acetamide
[(3R,4R)-1-[(5-methylthiophen-2-yl)methyl]-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
3-[5-chloro-2-(propan-2-yloxy)phenyl]-6-methoxypyridazine
1-[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]cyclobutan-1-amine
2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-{1-methyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}ethan-1-one
1-{[2-(2-aminoethyl)quinazolin-4-yl]amino}-3-(2,4-dimethylphenoxy)propan-2-ol
N-[(3S,4R)-1-(dimethyl-1,3-thiazole-5-carbonyl)-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
{1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}({[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl})amine
N-cyclopropyl-1-[(1s,4s)-4-({[5-(2-chlorophenyl)furan-2-yl]methyl}amino)cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
(2R,3R,6R)-3-(3-methoxyphenyl)-5-(4-methylpyrimidine-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-({8-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
3-(3-hydroxy-3-methylbutyl)-N-methyl-N-[2-(morpholin-4-yl)propyl]benzamide
N-[(3R,4R)-1-[2-(3,5-difluorophenyl)acetyl]-3-hydroxypiperidin-4-yl]pyridine-4-carboxamide
(1S,5R)-3-[(2-chloro-4-fluorophenyl)methyl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane
N-(4-fluorophenyl)-1-(propan-2-yl)piperidin-3-amine
N-[2-(2-fluorophenyl)-1-{1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}ethyl]-N-methylthiophene-2-carboxamide
4-{4-[3-(dimethylamino)pyrrolidine-1-carbonyl]phenyl}-2-methylbutan-2-ol
3-methyl-7-[4-(1H-1,2,4-triazol-1-yl)butanoyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
2-hydroxy-N-[1-(3-methylphenyl)piperidin-4-yl]-4-(methylsulfanyl)butanamide
N-benzyl-2-(3-methoxypiperidine-1-carbonyl)-N-methyl-2,3-dihydro-1H-inden-2-amine
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}thieno[3,2-d]pyrimidin-4-amine
1-ethyl-8-[3-(1H-pyrazol-1-yl)benzoyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
1-(1-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-4-yl)piperidin-3-ol
1-ethyl-5-{methyl[(1-methyl-1H-imidazol-2-yl)methyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
1-({3-methanesulfonylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)-4-(5-methylpyridin-2-yl)piperidin-4-ol
(3S,4S)-1-[(2,3-dimethoxyphenyl)methyl]-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
5-(2-methylpropyl)-1'-[1-(propan-2-yl)-1H-pyrrole-2-carbonyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-(2-methoxy-5-{[methyl(1,2-oxazol-3-ylmethyl)amino]methyl}phenoxy)-3-(4-methyl-1,4-diazepan-1-yl)propan-2-ol
1-[(5-methylfuran-2-yl)methyl]-3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine
1-(2,3-dihydro-1H-inden-4-yl)-2-(4-methanesulfonylphenyl)-1H-imidazole
N-cyclopropyl-1-[1-(1-methyl-6-oxo-1,6-dihydropyridine-3-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
4-{1-[(2-chlorophenyl)methyl]-1H-imidazol-2-yl}-1,5-dimethyl-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
N-[(3S,4R)-1-(2-ethylpyridine-4-carbonyl)-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
N-benzyl-N,1-diethyl-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-[benzyl(quinoxalin-2-ylmethyl)amino]-2-methylpropan-1-ol
4-(5-acetylthiophen-3-yl)-1-benzyl-3-methyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
1-(oxan-2-ylmethyl)-2-oxo-3-(pentan-3-yl)-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
1-[2-({[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}methyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol
2-[3-oxo-1-(pyridin-3-ylmethyl)piperazin-2-yl]-N-{[2-(trifluoromethoxy)phenyl]methyl}acetamide
ethyl 2-{[(3aS,6aR)-3-[(2-methoxyphenyl)methyl]-2-oxo-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazole-5-carbonyl]amino}acetate
3,5-dimethyl-N-[2-(methylsulfamoyl)ethyl]-1H-indole-2-carboxamide
[(2S,6S)-4-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
(3R,5S)-N3-[2-(4-methylphenyl)ethyl]-N5-(6-methylpyridin-3-yl)piperidine-3,5-dicarboxamide
2-(2,3-dihydro-1H-inden-1-yl)-N-[3-(1H-imidazol-1-yl)propyl]acetamide
1-{1-[5-(4-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]azetidin-3-yl}-3,5-dimethyl-1H-pyrazole
2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(3-methylpyridin-2-yl)methyl]acetamide
1-(2,4-dimethoxybenzoyl)-N-(4-fluorophenyl)piperidin-3-amine