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4-[4-(2-hydroxyethyl)piperazin-1-yl]-N-(3-methyl-1-propyl-1H-pyrazol-5-yl)piperidine-1-carboxamide
3-chloro-4-fluoro-N-{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}-1-benzothiophene-2-carboxamide
(2E)-3-(3,4-dimethoxyphenyl)-N-{[7-(5-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}prop-2-enamide
1-ethyl-5-{1-[5-(2-methyl-1,3-thiazol-5-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}-1H-1,2,4-triazole
N-ethyl-5-[1-(3-methylpyridin-4-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]pyrimidin-2-amine
2-ethyl-1-[3-(3-{[methyl(1-methylpiperidin-4-yl)amino]methyl}phenoxymethyl)piperidin-1-yl]butan-1-one
3-methyl-4-(3-phenyl-5-{[1,2,4]triazolo[1,5-a]pyrimidin-6-ylmethyl}-1H-1,2,4-triazol-1-yl)pyridine
2-methoxy-N-[2-(pyridin-3-yloxy)propyl]pyridine-3-carboxamide
4-methyl-6-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}pyrimidin-2-amine
4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-[(2-methylphenyl)methyl]piperidine
2-[1-({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)-1H-pyrazol-4-yl]ethan-1-ol
1-[2-(3-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-3-(4-hydroxyphenyl)propan-1-one
6-methyl-N4-{1-[4-(1H-1,2,4-triazol-1-yl)phenyl]ethyl}pyrimidine-2,4-diamine
2-chloro-6-fluoro-N,3-dimethyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]benzamide
2-[2-(oxolan-3-yl)ethyl]-5-(1,2,3,4-tetrahydroisoquinolin-2-yl)-2,3-dihydropyridazin-3-one
(3aS,6aS)-1-oxo-2-(prop-2-en-1-yl)-5-[3-(pyridin-2-yl)propanoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-[4-(pyrrolidin-1-ylmethyl)-1H-1,2,3-triazol-1-yl]-1-(pyrrolidine-1-sulfonyl)piperidine
1-(4-acetylphenyl)-3-[1-(thian-4-yl)piperidin-4-yl]urea
methyl 3-(5-acetylthiophene-2-carbonyl)-9-(cyclopentyloxy)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
(3S,4S)-1-(1-cyclobutanecarbonylpiperidin-4-yl)-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
1-[(1-{6-[(2,3-dihydroxypropyl)amino]pyridine-3-carbonyl}piperidin-4-yl)methyl]pyrrolidin-2-one
N-(1-{7-[(4-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-3-phenylpropanamide
2-(2-hydroxyethyl)-3-oxo-N-[4-(trifluoromethoxy)phenyl]piperazine-1-carboxamide
1-(2-{2,7-diazaspiro[4.5]decan-2-yl}-2-oxoethyl)pyrrolidin-2-one
1-(2-{3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidine-1-carbonyl}phenyl)ethan-1-one
N-(3-hydroxy-3-phenylpropyl)-N-methyl-2-(propan-2-yl)-1,3-benzoxazole-5-carboxamide
2-methyl-6-({[1-(9H-purin-6-yl)piperidin-4-yl]amino}methyl)pyrimidin-4-ol
methyl 5-{[(4aS,8aS)-4a-hydroxy-decahydroisoquinoline-2-carbonyl]amino}-2-chlorobenzoate
7-(3,6-dimethylpyrazin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-(4-methyl-3-phenylpiperazine-1-carbonyl)-2,3-dihydro-1H-imidazol-2-one
4-fluoro-N-[(1-{[2-(furan-2-yl)phenyl]methyl}piperidin-3-yl)methyl]benzamide
1-methyl-N-{3-[(5-methylpyridin-2-yl)amino]propyl}-1H-indole-6-carboxamide
3-({4-[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]-1H-1,2,3-triazol-1-yl}methyl)-1λ6-thiolane-1,1-dione
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(2-ethylpyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-methyl-7-[4-methyl-2-(propan-2-yl)pyrimidine-5-carbonyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
2-acetyl-8-[2-(2-methoxyphenoxy)ethyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-butyl-2,3-dioxo-N-(3-phenylprop-2-yn-1-yl)-1,2,3,4-tetrahydroquinoxaline-6-carboxamide
4-[6-(morpholine-4-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-2-yl]-4-oxobutanamide
3-methyl-8-[2-(2-oxo-1,2-dihydroquinoxalin-1-yl)acetyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
2-{[5-(oxan-4-yl)-4-(1-phenylethyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
2-{[(3R,4R)-4-cyclobutyl-4-hydroxy-3-methylpiperidin-1-yl]methyl}benzoic acid
3-benzyl-4-({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperazin-2-one
9-[3-(dimethylamino)benzoyl]-2-[2-(dimethylamino)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
2-[2-(3-methoxypyrrolidin-1-yl)-2-oxoethyl]-5-(piperidin-1-yl)-2,3-dihydropyridazin-3-one
N-{[6-chloro-4-(cyclopentylamino)quinazolin-2-yl]methyl}-2-phenoxyacetamide
N-[2-(2,4-dimethoxyphenyl)ethyl]-2-{1-[(4-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
N-[1-(1-phenylethyl)-1H-pyrazol-5-yl]-2-[3-(pyridin-3-yl)-1H-pyrazol-1-yl]acetamide
ethyl 3-benzyl-1-(1,2-oxazol-3-ylmethyl)piperidine-3-carboxylate
(4aS,8aR)-6-[3-(1H-pyrazol-1-yl)benzoyl]-decahydro-1,6-naphthyridine-4a-carboxylic acid
4-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]-1-methyl-2-phenylpiperazine