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6-[(1R,3S)-1-hydroxy-3-methoxy-7-azaspiro[3.5]nonan-7-yl]pyridine-2-carbonitrile
2-(7-fluoro-2-methyl-1H-indol-3-yl)-N-{3-[(pyridin-3-yl)amino]propyl}acetamide
4-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}-N-ethyl-N-(pyridin-4-ylmethyl)benzamide
4-[2-(benzyloxy)ethyl]-9-(furan-2-carbonyl)-1-methyl-1,4,9-triazaspiro[5.5]undecane
N-[(3R,4R)-3-hydroxy-1-[3-(methylsulfanyl)propyl]piperidin-4-yl]pyridine-4-carboxamide
2-[(5-ethyl-1,3,4-oxadiazol-2-yl)sulfanyl]-1-(3-{[4-(propan-2-yl)phenyl]amino}piperidin-1-yl)ethan-1-one
(5S,9aS,9bS)-5-[4-(dimethylamino)phenyl]-2-[(4-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-(3-methylpyridin-4-yl)-4-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]-1,4-diazepane
N-cyclohexyl-1-[(3-fluorophenyl)methyl]-N-methyl-6-oxopiperidine-3-carboxamide
N-[2-(1H-imidazol-4-yl)ethyl]-4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzamide
1-{5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl}-4-(3-phenyl-1H-pyrazole-4-carbonyl)piperazine
2-(3-phenylpropyl)-N-[1-(pyrazin-2-yl)propan-2-yl]-1,3-benzoxazole-5-carboxamide
5-[2-(2,3-dihydro-1H-inden-1-yl)acetyl]-1-(2-hydroxyethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
(3aR,7aS)-2-(2,6-dimethylpyrimidine-4-carbonyl)-2,3,3a,4,7,7a-hexahydro-1H-isoindole
1-[3-ethoxy-4-(prop-2-en-1-yloxy)benzoyl]-4-(1H-1,2,3,4-tetrazol-5-yl)piperidine
2-[(isoquinolin-5-yloxy)methyl]-N-[(1S)-1-(3-methylpyridin-2-yl)ethyl]-1,3-oxazole-4-carboxamide
2-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-2,8-diazaspiro[4.5]decane
1-(2-aminoethyl)-N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
N-[3-(cyclohexyloxy)propyl]-6-methoxy-1-methyl-1H-indole-2-carboxamide
1-{2-[methyl({[3-(1H-pyrazol-1-yl)phenyl]methyl})amino]pyrimidin-4-yl}piperidin-3-ol
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(1H-indol-4-ylmethyl)piperidin-3-ol
methyl 2-[methyl(2-methylpropyl)sulfamoyl]-6-(1,2,3-thiadiazole-4-carbonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
(3S,9aR)-3-[(4-chlorophenyl)methyl]-8-(4-methoxybenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(3S,4R)-1-(1-oxo-1,2-dihydroisoquinoline-4-carbonyl)-4-phenylpyrrolidine-3-carboxylic acid
2-(3,5-dimethyl-1H-pyrazol-4-yl)-2-[(3-phenoxyphenyl)formamido]acetic acid
N,2-dimethyl-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxamide
2-{1-[2-(1H-imidazol-4-yl)ethyl]-4-phenyl-1H-imidazol-5-yl}-1-(prop-2-en-1-yl)-1H-1,3-benzodiazole
4-[(1-acetylpiperidin-4-yl)oxy]-N-cyclohexyl-3-methoxy-N-methylbenzamide
3-[methyl(pyrazin-2-ylmethyl)sulfamoyl]-N-(2-methylbutyl)benzamide
1-(2-methyl-4-{methyl[(2E)-3-phenylprop-2-en-1-yl]amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
N-[(4,6-dimethylpyrimidin-2-yl)methyl]-1-{2-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-4-amine
5-[1-(2-cyclohexylacetyl)piperidin-4-yl]-5-[(4-fluorophenyl)methyl]-3-(oxolan-3-yl)imidazolidine-2,4-dione
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-methyl-N-(oxan-2-ylmethyl)-1,3-oxazole-4-carboxamide
N-{2-[(2-methylprop-2-en-1-yl)oxy]phenyl}-4-(4H-1,2,4-triazol-4-yl)piperidine-1-carboxamide
6-[4-(2-phenylpyrimidin-4-yl)piperidine-1-carbonyl]quinoline
1-[2-(2-phenylethyl)morpholin-4-yl]-2-(pyridin-4-yl)ethan-1-one
1-cyclohexyl-4-(isoquinoline-3-carbonyl)-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
5-methoxy-1-methyl-N-[1-(3-methylphenyl)-5-oxopyrrolidin-3-yl]-1H-indole-2-carboxamide
(1R,5R)-3-(5-methyl-1,2-oxazole-4-carbonyl)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonane
1-(1-cycloheptylpiperidin-3-yl)-3-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)urea
1-cyclobutanecarbonyl-N-methyl-N-(1,2-oxazol-3-ylmethyl)piperidine-4-carboxamide
4-(1-{5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-4-yl)morpholine
N-(1H-1,3-benzodiazol-2-ylmethyl)-2-{[(2-chlorophenyl)methyl]sulfanyl}acetamide
[(3aS,6aS)-2-{trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-octahydrocyclopenta[c]pyrrol-3a-yl]methanol
(3S,4S)-4-(piperidin-1-yl)-1-{[2-(propan-2-yl)pyrimidin-5-yl]methyl}pyrrolidin-3-ol
3-[(3S,7S,8aS)-3-(4-aminobutyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-phenylurea
4-{4-[(2,5-dimethylphenyl)methyl]piperazin-1-yl}-2-(thiophen-3-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
4-{1-[2-(dimethylamino)ethyl]-6-oxopiperidine-3-carbonyl}-1-[(4-fluorophenyl)methyl]piperazin-2-one
1-(6-methylpyrimidin-4-yl)-N-[2-(pyridin-3-yloxy)phenyl]piperidine-3-carboxamide
(2S)-1-acetyl-N-({4-[(3-phenylpropyl)amino]quinazolin-2-yl}methyl)pyrrolidine-2-carboxamide