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N-[(1-propyl-1H-imidazol-2-yl)methyl]-N-(1,3-thiazol-2-ylmethyl)cyclopropanamine
2,5-dioxo-6-[(3-propyl-1,2-oxazol-5-yl)methyl]-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
N-(1-{7-[(3,4-difluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)furan-3-carboxamide
(3R,4R)-1-[2-(dimethylamino)-6-ethylpyrimidin-4-yl]-4-(4-methylpiperazin-1-yl)piperidin-3-ol
2-[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]acetamide
1-cyclohexyl-3-[2-(3-hydroxyazetidin-1-yl)-2-oxoethyl]-2,6,6-trimethyl-4,5,6,7-tetrahydro-1H-indol-4-one
N-ethyl-2-phenyl-N-propylimidazo[1,2-a]pyridine-6-carboxamide
2-(2-methoxyethoxy)-1-[(1S,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
[1-(1H-1,3-benzodiazol-2-yl)-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]methanol
9-[(2R)-2-hydroxy-3-methylbutanoyl]-2-[3-(1H-imidazol-1-yl)propyl]-2,9-diazaspiro[5.5]undecan-3-one
ethyl 5-[(4-methyl-1H-imidazol-2-yl)methyl]-1-(2-methylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-[(2S)-1-hydroxy-4-(methylsulfanyl)butan-2-yl]-2-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
1-[1-(propane-1-sulfonyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
1-[5-(pyrrolidin-1-ylmethyl)imidazo[2,1-b][1,3]thiazole-6-carbonyl]piperidine
1-(3,5-dimethyl-1-benzofuran-2-carbonyl)-N,N-diethylpiperidine-3-carboxamide
N-(2-chlorophenyl)-3-{1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperidin-4-yl}propanamide
4-(4-fluorophenoxy)-1-{spiro[2.3]hexane-1-carbonyl}piperidine-4-carboxylic acid
5-{[benzyl(methyl)amino]methyl}-N-[2-(3-methylpyridin-2-yl)ethyl]-1,2-oxazole-3-carboxamide
1-(adamantan-2-yl)-4-(cyclohex-3-en-1-yl)-1H-1,2,3-triazole
N-[4-(3-fluorophenyl)phenyl]-1-(5-methylthiophene-2-carbonyl)piperidine-3-carboxamide
N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-2-(4-methoxyphenoxymethyl)-1,3-oxazole-4-carboxamide
ethyl 4-[({5-[(3-fluorophenyl)methyl]-6-oxo-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-7-yl}methyl)amino]piperidine-1-carboxylate
1-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-4-phenylpiperidine-4-carbonitrile
1-[(1-methyl-1H-imidazol-5-yl)methyl]-4-(3-methylpyridin-2-yl)piperazine
N-methyl-N-[(5-{[4-(pyridin-3-yl)piperazin-1-yl]methyl}furan-2-yl)methyl]methanesulfonamide
N-[(2-chlorophenyl)methyl]-3-cyclopropyl-N-(prop-2-en-1-yl)-1H-pyrazole-5-carboxamide
4-{5-[(4-methyl-1H-imidazol-2-yl)methyl]-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}morpholine
4-(2-chloro-6-methoxyphenyl)-5,6-dimethylthieno[2,3-d]pyrimidine
1-{4-[(2-methylphenyl)methyl]piperazin-1-yl}-2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethan-1-one
(4aS,7aR)-1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-4-(2-methylpropanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(dimethyl-1,2-oxazol-4-yl)-1-(4-{2-[2-(3-methoxyphenyl)ethyl]-3H-imidazo[4,5-b]pyridin-3-yl}piperidin-1-yl)ethan-1-one
(2,1,3-benzoxadiazol-4-ylmethyl)[1-(dimethyl-1,3-thiazol-4-yl)ethyl]methylamine
2-(3-{3-[2-(methylsulfanyl)pyrimidin-4-yl]phenyl}-1H-pyrazol-1-yl)ethan-1-ol
N-[(3,4-difluorophenyl)methyl]-1-methyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-cyclopentyl-4-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-4-oxobutanamide
[(1-ethyl-1H-imidazol-2-yl)methyl](methyl)[(5-phenyl-1,2-oxazol-3-yl)methyl]amine
[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]({[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl})amine
(3S,4R)-1-[4-(4-fluorophenyl)oxane-4-carbonyl]-3-methoxypiperidin-4-amine
N-{[2-(4-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-2-methyl-3-(morpholin-4-yl)propanamide
N-[2-(2,5-dimethylphenoxy)ethyl]oxolane-3-carboxamide
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-2-ethylpyrimidine-5-carboxamide
7-(1-benzofuran-5-ylmethyl)-2,7-diazaspiro[4.4]nonane-1,3-dione
1-[benzyl(methyl)amino]-3-[4-({[3-(methylsulfanyl)propyl]amino}methyl)phenoxy]propan-2-ol
8-methoxy-N-[2-(5-phenyl-1,2,4-oxadiazol-3-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-methyl-4-{3-[(1R,5R)-6-methyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-3-oxopropyl}benzene-1-sulfonamide
3-{2-[methyl(2-methylpropyl)amino]ethyl}-8-[(2-methyl-1,3-oxazol-4-yl)methyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-{4-[1-(cyclohexylmethyl)-1H-1,2,3-triazole-4-carbonyl]piperazin-1-yl}-1,3-benzoxazole
1-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-4-(3-methoxyphenyl)piperazine
4-(6,7-dimethoxy-1-methyl-1,2,3,4-tetrahydroisoquinolin-2-yl)-N-(propan-2-yl)pyridine-2-carboxamide
1-{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}-4-[(3-methylphenyl)methyl]piperazine