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1-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]-N-[3-(4-fluorophenyl)phenyl]piperidine-3-carboxamide
1-(4-methylquinolin-2-yl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
4-methoxy-N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N,3-dimethylbenzamide
1-{5-oxo-1-[4-(propan-2-yl)phenyl]pyrrolidine-3-carbonyl}-1,4-diazepan-5-one
8-[(3,4-difluorophenyl)methyl]-1-methyl-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
N,N-dimethyl-5-[1-(2-methyl-1,8-naphthyridine-3-carbonyl)pyrrolidin-2-yl]thiophene-2-carboxamide
4-[2-(3,5-dimethyl-1H-pyrazol-4-yl)acetyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
1-(6-ethylpyrimidin-4-yl)-4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
1-[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonan-7-yl]-3-(4-methyl-1,4-diazepan-1-yl)propan-1-one
3-[(3S,4R)-3-benzyl-1-methylpiperidin-4-yl]-1-(2-chloropyridin-3-yl)urea
1,9-dimethyl-4-[(4-methylpiperidin-1-yl)sulfonyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
3-[(4S,4aS,8aS)-4-hydroxy-4-phenyl-decahydroquinolin-1-yl]-1-(pyrrolidin-1-yl)propan-1-one
2-(3-{[cyclopropyl({[4-(methylsulfanyl)phenyl]methyl})amino]methyl}phenoxy)acetamide
8-[2-(3,4-dimethylphenoxy)ethyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
(3R,4R)-3-[(dimethylamino)methyl]-N-[(3-fluorophenyl)methyl]-4-(hydroxymethyl)pyrrolidine-1-carboxamide
4-methyl-6-{8-methyl-9-oxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carbonyl}-3,4-dihydro-2H-1,4-benzoxazin-3-one
7-[(4-fluorophenyl)methyl]-2-(oxane-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
(2S,4R)-1-[(2,4-difluorophenyl)methyl]-N-[2-(dimethylamino)ethyl]-4-[(4,6-dimethylpyrimidin-2-yl)sulfanyl]pyrrolidine-2-carboxamide
(3R,4R)-1-{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}-4-(morpholin-4-yl)piperidin-3-ol
N-{[7-chloro-5-(thiophen-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}cyclobutanecarboxamide
5-(2-{4-[(3-chlorophenyl)methyl]piperazin-1-yl}-2-oxoethyl)-2,6-dimethyl-3,4-dihydropyrimidin-4-one
N-[1-methyl-6-(propan-2-yloxy)-1H-indazol-3-yl]-2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)acetamide
3-benzyl-8-(1-methoxypropan-2-yl)-1-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[(4-chlorophenyl)methanesulfonyl]-4-(1-ethyl-1H-imidazol-2-yl)piperidine
1-{3,5-dimethyl-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl}-4-[5-(4-fluorophenyl)-2H-1,2,3,4-tetrazol-2-yl]butan-1-one
3-(2-chlorophenyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-3-phenylpropanamide
2-(3-fluorophenyl)-N-({7-propyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)acetamide
1-{2-[5-(1-methylazepan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}pyrrolidin-2-one
1-(2-cyclopentyl-2-phenylacetamido)cyclopentane-1-carboxylic acid
N-[1-(4-hydroxyphenyl)propyl]-2-(1-propylpiperidin-4-yl)acetamide
3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-(2-methylpropyl)-N-(3-phenylprop-2-yn-1-yl)propanamide
3-(3-methoxyphenyl)-N-[(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]-1H-pyrazole-5-carboxamide
6-(3-oxo-3-{3-[4-(trifluoromethyl)benzoyl]piperidin-1-yl}propyl)-2,3-dihydropyridazin-3-one
(1R,5R)-6-[2-(3-hydroxyphenyl)acetyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
4-(cyclopropylmethyl)-1-{[4-(methylsulfanyl)phenyl]methyl}-1,4-diazepan-5-one
2-(4-methanesulfonylphenyl)-N,N-dimethylpyridine-3-carboxamide
2-({5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-4H-chromen-4-one
2-[2-(1H-imidazol-4-yl)ethyl]-8-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-2-(pyrrolidin-1-yl)pyrimidine-5-carboxamide
N-methyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]pyridin-4-amine
3-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-9-methyl-3,9-diazaspiro[5.6]dodecan-10-one
4-(3-benzoylpiperidine-1-carbonyl)-1-{4-methyl-6H,7H,8H-cyclopenta[g]quinazolin-2-yl}piperidine
(3S,4R)-4-(3-methylthiophen-2-yl)-1-[2-(morpholin-4-yl)pyridine-3-carbonyl]piperidin-3-ol
3-{[2-(ethoxymethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]amino}azepan-2-one
N-[4-(2-methyl-1H-imidazol-1-yl)phenyl]-1-(1-methylcyclopropanecarbonyl)pyrrolidine-2-carboxamide
1-ethyl-8-(1-methoxypropan-2-yl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3S,4S)-N-(4-butylphenyl)-3-hydroxy-4-(4-methylpiperazin-1-yl)pyrrolidine-1-carboxamide
5-amino-N-[2-(1-methylpiperidin-3-yl)ethyl]-4-phenyl-1H-pyrazole-3-carboxamide
[(3R,4R)-4-(azepan-1-ylmethyl)-1-{[4-(methylsulfanyl)phenyl]methyl}pyrrolidin-3-yl]methanol
(1-{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}piperidin-4-yl)(pyridin-3-yl)methanol