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3-[5-(thiophen-2-yl)-1H-pyrazole-4-carbonyl]-3,9-diazaspiro[5.6]dodecan-10-one
4-(2,3-dimethoxyphenyl)-6-(4-methylpiperazin-1-yl)pyrimidin-2-amine
N-[(1,5-dimethyl-1H-pyrazol-3-yl)methyl]-2-[1-(3-methylbutyl)-3-oxopiperazin-2-yl]acetamide
1-[(4-chlorophenyl)methyl]-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
4-[(1S,4S)-2-azabicyclo[2.2.1]heptane-2-carbonyl]-7-methyl-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]quinoline
2-(4-{[3-(3,4-dimethoxybenzoyl)piperidin-1-yl]methyl}phenoxy)ethan-1-ol
5-(1,2-oxazinane-2-carbonyl)-1,3-benzothiazol-2-amine
2-[4-(4-methoxyphenyl)piperazin-1-yl]-4-(pyridin-2-yl)pyrimidine
N-[(1R,3R)-3-aminocyclopentyl]-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
3-[(3R,4S)-1-{[5-(hydroxymethyl)furan-2-yl]methyl}-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
3-(3-methoxyphenyl)-N-[(3R,4R)-4-(morpholin-4-yl)oxolan-3-yl]-1H-pyrazole-5-carboxamide
6-chloro-N,2-dimethyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}imidazo[1,2-a]pyridine-3-carboxamide
N-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-(cyclohexylmethyl)piperidin-3-amine
1-(2-{[methyl(pyridin-3-ylmethyl)amino]methyl}phenoxy)-3-(piperidin-1-yl)propan-2-ol
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-[1-(naphthalen-1-ylmethyl)-3-oxopiperazin-2-yl]acetamide
2-(4-{[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]methyl}phenoxy)propanoic acid
6-({2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}amino)-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
4-{3-[2-(2-methylphenyl)ethyl]piperidine-1-carbonyl}-2-(4H-1,2,4-triazol-4-yl)pyridine
(3R,4R)-4-(2-methoxyethyl)-3-methyl-1-[(6-methylquinolin-5-yl)methyl]piperidin-4-ol
8-[(4-methoxyphenyl)methyl]-1-(3-methoxypropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[1-(2-methoxyphenyl)ethyl]-N-methyl-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
N-[(5-fluoro-1H-indol-2-yl)methyl]-3-(2-phenylethyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
8-(5-acetyl-2,4-dimethyl-1H-pyrrole-3-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[4-(1H-indol-2-yl)phenyl]-1-[3-(1H-pyrazol-1-yl)propyl]piperidine-4-carboxamide
dimethyl[(5-{[3-(pyridin-2-yl)phenyl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)methyl]amine
N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-{1-[(4-ethoxyphenyl)methyl]-4-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl}ethan-1-ol
1-methyl-4-phenyl-3-{[1-(1,3-thiazol-2-yl)piperidin-4-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
1-methyl-N-[3-(morpholin-4-yl)propyl]-2-oxo-1,2-dihydroquinoline-4-carboxamide
2-(5-acetylthiophen-3-yl)-1-(6-hydroxy-1,4-oxazepan-4-yl)ethan-1-one
3-(benzyloxy)-1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}piperidine
N5-benzyl-N3-methyl-4-oxo-N3-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
(3S,4S)-1-(2-chloro-6-fluoro-3-methylbenzoyl)-4-propylpyrrolidine-3-carboxylic acid
1-{1-[(3-methoxyphenyl)methyl]-5-[1-(propan-2-yl)piperidin-4-yl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}piperidin-3-ol
5-[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]-N-methyl-N-(1-methylpiperidin-4-yl)pyridin-2-amine
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[1-(pyridin-2-yl)propan-2-yl]benzamide
1-[3-({[(2-methyl-1,3-thiazol-4-yl)methyl]amino}methyl)phenoxy]-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
(1S,3R)-3-amino-N-[4-(4-methyl-4H-1,2,4-triazol-3-yl)phenyl]cyclopentane-1-carboxamide
N-{2-[benzyl(methyl)amino]-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl}-3-methyl-1H-pyrazole-5-carboxamide
2-[4-(6-chloroquinolin-2-yl)-1H-pyrazol-1-yl]-N-(2-methyl-2H-1,2,3-triazol-4-yl)acetamide
3-(2-{4-[(4-methylphenyl)methyl]-3-oxopiperazin-1-yl}-2-oxoethyl)-2,3-dihydro-1H-isoindol-1-one
1-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-1-methyl-3-[1-(propan-2-yl)-1H-1,2,3-triazol-4-yl]urea
8-(4-methyl-1H-imidazole-5-carbonyl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2,5-dimethyl-3-(4-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}piperazin-1-yl)pyrazine
1-{[2-(3,5-dimethoxyphenoxy)phenyl]methyl}-4-methylpiperazine
1-methyl-4-{5-[1-(2-methyl-1H-imidazol-1-yl)ethyl]-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-1-yl}piperidine
N-[(3S,4R)-1-(3-phenylpropyl)-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
2-amino-6-(4-hydroxyphenyl)-4-[1-(2-methoxyethyl)piperidin-4-yl]-5-methylpyridine-3-carbonitrile
2-[1-(1-methyl-1H-indole-2-carbonyl)piperidin-4-yl]-1,2,3,4-tetrahydroisoquinoline
N-[(2R)-1-(3,3-diphenylpiperidin-1-yl)-1-oxopropan-2-yl]acetamide