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(2S,4S)-N,1-dimethyl-4-[3-(methylsulfanyl)propanamido]-N-(naphthalen-1-ylmethyl)pyrrolidine-2-carboxamide
1-methyl-1'-[2-(2-methylphenyl)acetyl]-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
1-[2-(cyclopropylmethyl)-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl]-2-phenylethane-1,2-dione
N-benzyl-N-cyclopentyl-2-(4H-1,2,4-triazol-4-yl)benzamide
4-(cyclohex-3-en-1-yl)-1-{[2-(1H-pyrazol-1-yl)phenyl]methyl}-1H-1,2,3-triazole
N-methyl-2-[4-(pyrimidin-2-yl)piperazin-1-yl]-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)acetamide
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-2-(pyridin-3-yl)-5,6,7,8-tetrahydroquinazolin-5-amine
(3S)-N-tert-butyl-2-(3-hydroxypyridine-2-carbonyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
5-(2,4-difluorophenoxymethyl)-N-[2-(7-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-1,2-oxazole-3-carboxamide
1-cyclohexanecarbonyl-N-{[4-(2-oxopyrrolidin-1-yl)phenyl]methyl}pyrrolidine-2-carboxamide
{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}(methyl){[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}amine
N-[(3R,4S)-4-cyclopropyl-1-(diethylcarbamoyl)pyrrolidin-3-yl]-4,5,6,7-tetrahydro-1,2-benzoxazole-3-carboxamide
{1-[1-(4-chlorophenyl)piperidin-4-yl]-3-[(2-fluorophenyl)methyl]piperidin-3-yl}methanol
3-(4-chlorobenzoyl)-1-[(2,5-dimethoxyphenyl)methyl]piperidine
({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)(ethyl)[2-(phenylsulfanyl)ethyl]amine
N-{[1-(2,3-dihydro-1,4-benzodioxine-6-sulfonyl)piperidin-3-yl]methyl}thiophene-2-carboxamide
2-[1-(4-chlorophenyl)-5-oxo-3-propyl-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-(1,2-oxazol-3-ylmethyl)acetamide
ethyl 2-[methyl(5-{[methyl(1H-pyrazol-5-ylmethyl)amino]methyl}pyrimidin-2-yl)amino]acetate
N-ethyl-2-[4-methyl-6-(morpholine-4-carbonyl)-3,4-dihydro-2H-1,4-benzoxazin-3-yl]-N-propylacetamide
N-[(2R)-1-(benzyloxy)-3-hydroxypropan-2-yl]-2-[(prop-2-en-1-yl)amino]benzamide
8-fluoro-2-[4-(oxan-4-yl)piperazine-1-carbonyl]quinoline
(3R,4R)-4-(2-methoxyethyl)-3-methyl-1-(4-methyl-1,3-thiazole-5-carbonyl)piperidin-4-ol
4-(cyclopropylmethyl)-1-[6-methyl-2-(methylamino)pyrimidin-4-yl]-3-(propan-2-yl)-1,4-diazepan-5-one
N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]quinoxaline-6-carboxamide
N-methyl-3-{[(5-methylthiophen-2-yl)methyl]amino}-N-[(3-propyl-1,2,4-oxadiazol-5-yl)methyl]benzamide
(4aR,7aS)-1-benzyl-4-(pyridine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
[(1-ethyl-1H-pyrazol-4-yl)methyl](methyl)[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]amine
2-[(2-chlorophenyl)methyl]-4-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]morpholine
(1R,9aR)-1-[3-(pyrrolidin-1-ylmethyl)phenoxymethyl]-octahydro-1H-quinolizine
2-(4-methoxyphenyl)-5-{[3-(piperidin-1-yl)azetidin-1-yl]methyl}pyrimidine
3-benzyl-5-[2-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)ethyl]-1,2,4-oxadiazole
4-[4-(2-chlorophenyl)piperidin-4-yl]-N-cyclobutylpyrimidin-2-amine
3-{5H,6H,7H,8H-imidazo[1,5-a]pyrazine-7-carbonyl}-2-methyl-4,5,6,7-tetrahydro-1H-indol-4-one
2-methyl-8-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]acetyl}-2,8-diazaspiro[4.5]decan-3-one
(3S,5R)-N3-[(3,4-dimethoxyphenyl)methyl]-N5-(4-fluorophenyl)-1-(1H-indol-3-ylmethyl)piperidine-3,5-dicarboxamide
4-{5-ethyl-6-methylthieno[2,3-d]pyrimidin-4-yl}-N,N-dimethylbenzamide
N-ethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
1-benzyl-8-[(4-hydroxyphenyl)methyl]-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-{[methyl({[4-phenyl-5-(piperidin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]methyl})amino]methyl}phenol
3-(2-hydroxypyridin-3-yl)-1-(oxolan-2-ylmethyl)-1-[(2E)-3-phenylprop-2-en-1-yl]urea
5-fluoro-3-methyl-2-(4-phenyl-1,4-diazepane-1-carbonyl)-1H-indole
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(2-methoxyethyl)-1-methyl-1H-indole-2-carboxamide
(2S)-3-methyl-2-{[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}butanamide
N-[(4-fluorophenyl)methyl]-3-{1-[2-(1H-indol-3-yl)acetyl]piperidin-4-yl}propanamide
N-(2-cycloheptylethyl)-1-(2-methoxyethyl)-6-oxopiperidine-3-carboxamide
N-[1-(methoxymethyl)cyclopropyl]-N-methyl-2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,3-oxazole-4-carboxamide
2-[3-methoxy-4-(pyrrolidin-1-ylmethyl)phenoxy]pyridine-3-carbonitrile
N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
1-(2-{[6-(thiomorpholin-4-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]amino}ethyl)piperidin-2-one
4-methyl-N-{4-[2-(pyridin-2-yl)acetamido]phenyl}benzamide