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2-(1-{1-[(4-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-4-yl)-1,3-benzoxazole
methyl 4-[(3-{[4-(diethylcarbamoyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)methyl]benzoate
7-(2-methoxyacetamido)-1-methyl-2-phenyl-N-[3-(pyridin-3-yl)propyl]-1H-1,3-benzodiazole-5-carboxamide
4-(4-{3-[(4-fluorophenyl)methoxy]azetidine-1-carbonyl}phenyl)-2-methylbutan-2-ol
2-amino-4-(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)-5H,7H,8H-pyrano[4,3-b]pyridine-3-carbonitrile
5-benzyl-1-(3-methoxyphenyl)-4-(1H-pyrrole-2-carbonyl)piperazin-2-one
4-[4-(4-benzyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-2-methoxypyridine
3-methyl-1-(1-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)butan-1-ol
[3-(cyclopropylmethyl)-1-{[2-(difluoromethoxy)phenyl]methyl}piperidin-3-yl]methanol
N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-{[7-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}butanamide
2-[5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]pyrimidin-4-amine
1-(1-methyl-1H-pyrrole-2-carbonyl)-3-(4-methylphenoxymethyl)piperidine
6-(4-chloro-2-methoxybenzoyl)-2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
3-benzyl-6-(3-methylfuran-2-yl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
(3S,4S)-1-[(2-hydroxy-5-methoxyphenyl)methyl]-4-(morpholin-4-yl)pyrrolidin-3-ol
1-cyclohexyl-4-[(4-fluoro-3-methoxyphenyl)methyl]-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
4-methyl-2-(1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidin-3-yl)-1H-1,3-benzodiazole
4-(2-chloro-4-fluorobenzoyl)-6-methoxy-1-(pyridin-3-ylmethyl)-1,4-diazepan-2-one
4-[(diethylamino)methyl]-5-ethyl-N-methyl-N-(pyridin-4-ylmethyl)furan-2-carboxamide
(2S,4R)-4-amino-N-methyl-1-[4-methyl-2-(piperidin-1-yl)pyrimidine-5-carbonyl]pyrrolidine-2-carboxamide
1-[2-(4-methoxyphenyl)ethyl]-8-[(3-methoxyphenyl)methyl]-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[(4-chlorophenyl)methyl]-8-[(1-ethyl-1H-pyrazol-4-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
4-[3-(2,6-dimethylphenoxy)azetidine-1-carbonyl]-N,N-dimethylaniline
2-(3-chlorophenyl)-N-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]-2-hydroxyacetamide
(4aS,8aR)-1-(2-aminoethyl)-6-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]-decahydro-1,6-naphthyridin-2-one
1-{3-[3-(2-oxopyrrolidin-1-yl)piperidin-1-yl]propyl}-2,3-dihydro-1H-imidazol-2-one
(4aS,8aR)-1-(4-hydroxybutyl)-6-(thiophen-2-ylmethyl)-decahydro-1,6-naphthyridin-2-one
N-[(3-chlorophenyl)methyl]-3-[1-(pyrimidin-2-ylmethyl)piperidin-4-yl]propanamide
2-{[3-(2-hydroxyethyl)-4-[(4-methoxy-3-methylphenyl)methyl]piperazin-1-yl]methyl}-4-methoxyphenol
2-{4-[2-(pyridin-4-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]morpholin-2-yl}ethan-1-ol
2-({1-[(4-fluorophenyl)methyl]-1H-1,2,4-triazol-5-yl}methyl)-2,3-dihydro-1H-isoindole
N-[2-hydroxy-3-(3-methoxyphenoxy)propyl]-1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
4-{4-[5-(pyrrolidin-2-yl)thiophene-2-carbonyl]piperazine-1-carbonyl}morpholine
1-ethyl-N-{[3-(trifluoromethoxy)phenyl]methyl}piperidine-2-carboxamide
(1S,5R)-6-benzyl-3-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N4-[1-(2,5-dimethoxyphenyl)ethyl]-5,6-dimethylpyrimidine-2,4-diamine
N-tert-butyl-5-(2-fluoro-6-methoxyphenyl)furan-2-carboxamide
3-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-5-ethyl-5-{1-[(4-fluoro-3-methoxyphenyl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
5-amino-N-[2-(6-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-1H-pyrazole-3-carboxamide
5-{6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-2-amine
(2R,6R)-4-[(5-methylfuran-2-yl)methyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
1-{[1-(furan-2-ylmethyl)piperidin-3-yl]methyl}-3-[2-(1H-pyrazol-1-yl)phenyl]urea
3-(1-methylpiperidin-3-yl)-1-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}propan-1-one
3-(2H-1,3-benzodioxol-5-ylmethyl)-5-ethyl-5-{1-[(4-methoxy-3-methylphenyl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
N-(1H-indazol-6-yl)-4-(thiophen-2-ylmethyl)-1,4-diazepane-1-carboxamide
{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}[(5-methylpyrazin-2-yl)methyl]amine
2-{2-[9-methoxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-oxoethyl}-4-phenyl-1,2-dihydrophthalazin-1-one
2-[(4-methoxyphenyl)methyl]-N-[2-(2-oxopyrrolidin-1-yl)ethyl]-1,3-benzoxazole-6-carboxamide
1-{1'-[2-(methylamino)-1,3-thiazole-4-carbonyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one