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[3-(methylsulfanyl)propyl]({[2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
N-[(3R,4S)-4-cyclopropyl-1-(2-phenylethyl)pyrrolidin-3-yl]-3-hydroxypropanamide
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-3-{5-[2-(2-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propanamide
(1r,4r)-4-[(3-propoxypiperidin-1-yl)methyl]cyclohexan-1-ol
3-(dimethyl-1,2-oxazol-4-yl)-1-[4-(4-methoxyphenoxy)piperidin-1-yl]propan-1-one
N-[4-fluoro-3-(trifluoromethyl)phenyl]-3-oxo-2,8-diazaspiro[4.5]decane-8-carboxamide
1-benzyl-N3-ethyl-4-oxo-N5-[2,2,2-trifluoro-1-(furan-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
(8R,9aS)-2-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-8-hydroxy-octahydro-1H-pyrido[1,2-a]piperazine-1,4-dione
4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}benzamide
5-[4-(furan-3-carbonyl)-1,4-diazepane-1-carbonyl]-N,N,4-trimethylpyrimidin-2-amine
(3S,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-7-{[(3-methoxyphenyl)methyl]amino}-octahydropyrrolo[1,2-a]piperazine-1,4-dione
7-[(3-methoxyphenyl)methyl]-2-(5-methylpyrazine-2-carbonyl)-2,7-diazaspiro[4.5]decane
3-(2H-1,3-benzodioxol-5-yl)-5-(furan-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
1-(3,6-dimethyl-1-benzofuran-2-carbonyl)-3-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidine
methyl (2S,3S)-2-[(3-benzyl-1,2-oxazol-5-yl)formamido]-3-methylpentanoate
2-(2,4-dichlorophenoxy)-N-[2-(pyrazin-2-yl)ethyl]acetamide
4-[(2,6-difluorophenyl)methyl]-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-(5-fluoro-2-methoxyphenyl)-2-{methyl[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amino}acetic acid
N-{[7-(5-acetyl-2-fluorophenyl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}-3,4,5-trimethoxybenzamide
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
(8R,9aS)-8-hydroxy-2-[(2-propyl-1,3-thiazol-4-yl)methyl]-octahydro-1H-pyrido[1,2-a]piperazine-1,4-dione
1-{2-amino-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-1,4-diazepan-6-ol
N5-[2-(cyclohex-1-en-1-yl)ethyl]-N3-methyl-N3-(2-methylpropyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
N-methyl-4-(piperidin-3-yl)-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)benzamide
2-(4-ethylpiperazin-1-yl)-N-(pyridin-3-ylmethyl)-2,3-dihydro-1H-indene-2-carboxamide
3-(4-methyl-1,3-thiazol-5-yl)-N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]propanamide
3-{[(2-amino-5,6,7,8-tetrahydroquinazolin-4-yl)amino]methyl}-6-ethyl-2-methoxy-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
1-[(2-fluorophenyl)methyl]-N,N-bis(prop-2-en-1-yl)-1H-1,2,3-triazole-4-carboxamide
3-[({[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}amino)methyl]-3-hydroxy-1-methylpiperidin-2-one
1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}azocane
1-ethyl-4-{[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]methyl}-1H-pyrrole-2-carbonitrile
2-{1-[(4-fluorophenyl)methyl]-4-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]amine
3-methyl-4-{[3-(2-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1-propyl-1H-pyrazole
2-(2-methyl-1,3-thiazol-4-yl)-N,N-bis(pyridin-3-ylmethyl)acetamide
4-methyl-N-(2-{7-[(4-phenyl-1,3-thiazol-2-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)benzamide
1-(4,6-dimethylquinazolin-2-yl)-N-(1-phenylcyclopropyl)piperidine-4-carboxamide
5-amino-N-[(2E)-3-phenylprop-2-en-1-yl]-N-propyl-1H-pyrazole-3-carboxamide
N-[(3S,4R)-1-{2-[(2-methoxyethyl)(methyl)amino]acetyl}-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
5-(methoxymethyl)-N-[(1-methylpiperidin-4-yl)methyl]-N-(2-phenylethyl)furan-2-carboxamide
2-{[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]amino}-N-(2-fluoro-5-methylphenyl)acetamide
(1S,6R)-9-(benzenesulfonyl)-3,9-diazabicyclo[4.2.1]nonan-4-one
(4aS,8aR)-1-[2-(cyclohex-1-en-1-yl)ethyl]-6-(2-methylpyrimidin-4-yl)-decahydro-1,6-naphthyridin-2-one
2-[4-(methylsulfanyl)phenyl]-1-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
5-(3,4-difluorophenoxymethyl)-N-ethyl-N-[2-(pyrrolidin-1-yl)ethyl]-1,2-oxazole-3-carboxamide
4-[2-(2,3-dihydro-1H-indol-1-yl)-2-oxoethyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
2-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-oxopiperazin-2-yl}-N-(pyridin-4-ylmethyl)acetamide
N-{[2-(azepan-1-yl)-7-fluoroquinolin-3-yl]methyl}-3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-(2-methoxyethyl)propanamide
2-methyl-4-(2-methylphenyl)-1-(1,3-thiazole-4-carbonyl)piperazine