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4-(1-{4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]benzoyl}piperidin-4-yl)pyridine
5-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepane-1-carbonyl]-1,2-dihydropyridin-2-one
N-[(3S,4R)-1-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
4-{1-[3-(2-oxoazepan-1-yl)propanoyl]piperidin-3-yl}benzoic acid
N-{4-[1-(furan-2-ylmethyl)-4-phenyl-1H-imidazol-5-yl]phenyl}acetamide
N-benzyl-N-ethyl-2-[(quinolin-6-yloxy)methyl]-1,3-oxazole-4-carboxamide
methyl 4-{[7-(1-hydroxy-2-phenylethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}benzoate
5-[3-(4-fluorophenyl)-1H-pyrazol-5-yl]-1-methyl-1H-1,2,4-triazole
2,2-dimethyl-N-[1-(1-{6-methylimidazo[2,1-b][1,3]thiazole-5-carbonyl}piperidin-4-yl)-1H-pyrazol-5-yl]propanamide
N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-4-(piperidin-1-ylmethyl)benzamide
2-[3-({dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}amino)propyl]phenol
6-ethyl-N,1,5-trimethyl-2-oxo-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-1,2-dihydropyridine-3-carboxamide
1-{3-fluoroimidazo[1,2-a]pyridine-2-carbonyl}-3-(3-methylphenoxymethyl)piperidine
5-chloro-4-{1-[(4,6-dimethylpyridin-3-yl)methyl]-1H-imidazol-2-yl}-2-methoxyphenol
N-{[1-(furan-2-ylmethyl)pyrrolidin-3-yl]methyl}-4-hydroxy-3-methoxybenzamide
1-cyclohexyl-N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
2-chloro-4-({[6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}methyl)-6-methoxyphenol
3-{[(3-hydroxypyrrolidin-3-yl)methyl]amino}-N-phenylpropanamide
2-cyclopropyl-8-(2-hydroxy-3-methylbenzoyl)-2,8-diazaspiro[5.5]undecan-3-one
1-methyl-3-{2-[3-(pyridin-2-ylmethoxy)phenyl]-1H-imidazol-1-yl}pyrrolidin-2-one
methyl 4-{5-chloro-2-[(2-acetamidoacetamido)methyl]-2,3-dihydro-1-benzofuran-7-yl}benzoate
(2S,4R)-1-[(2,5-difluorophenyl)methyl]-N,N-dimethyl-4-[(1-methyl-1H-imidazol-2-yl)sulfanyl]pyrrolidine-2-carboxamide
N-[3-(1,3-benzoxazol-2-yl)propyl]-2-(4-oxo-3,4-dihydroquinazolin-3-yl)acetamide
5-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]isoquinoline
1-[4-(piperidin-1-ylmethyl)benzoyl]azetidin-3-ol
N-[3-(3-acetamidobutanamido)phenyl]-3-methylbenzamide
6-methyl-2-{[1-oxo-1-(3-oxo-4-phenylpiperazin-1-yl)propan-2-yl]sulfanyl}-3,4-dihydropyrimidin-4-one
8-methyl-3-({methyl[3-(1-methyl-1H-pyrazol-4-yl)propyl]amino}methyl)-1,2-dihydroquinolin-2-one
3-methyl-4-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}pyridine
5-[(2-methoxyethyl)(pyridin-2-ylmethyl)carbamoyl]-1H-imidazole-4-carboxylic acid
N-cyclopropyl-N-({3-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)-4-(trifluoromethyl)benzamide
6-methoxy-1-methyl-N-[2-(pyrrolidine-1-sulfonyl)ethyl]-1H-indole-2-carboxamide
3-{8-chloro-5-methyl-[1,2,4]triazolo[4,3-a]quinolin-1-yl}-1-ethylpiperidine
2-ethyl-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}benzamide
N-[(3R,4S)-1-(carbamoylmethyl)-4-(propan-2-yl)pyrrolidin-3-yl]-2-methoxy-5-methylbenzamide
3-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-1-(2-methoxyethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylic acid
2-(3,4-dichlorophenyl)-4-(1H-imidazol-4-ylmethyl)morpholine
2-{4-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-1-[(5-methylfuran-2-yl)methyl]piperazin-2-yl}ethan-1-ol
2-(2-hydroxyethyl)-9-[4-(4-methylphenyl)-4-oxobutyl]-2,9-diazaspiro[5.5]undecan-3-one
3-[2-(dimethylamino)ethyl]-5-[1-(3,5-dimethylbenzoyl)piperidin-4-yl]-5-(2-phenylethyl)imidazolidine-2,4-dione
2-(pentan-2-yl)-1H-1,3-benzodiazole-6-carboxylic acid
N-[2-(dimethylamino)ethyl]-7-(1,3-thiazole-4-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-({3-[3-(pyrazin-2-yl)phenyl]-1H-pyrazol-1-yl}methyl)-1,3-benzothiazole
4-{[(1-ethyl-1H-pyrazol-4-yl)methyl]amino}-1-[2-(4-fluorophenyl)ethyl]pyrrolidin-2-one
8-[2-(1H-imidazol-2-yl)benzoyl]-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
1-benzyl-N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]pyrrolidin-3-amine
2-(2-{4-[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]-1H-1,2,3-triazol-1-yl}propyl)-3-methylpyridine
7-(3,4-dimethoxyphenyl)-4-[(3-fluorophenyl)methyl]-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-phenyl-N-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}-1H-1,2,3-triazole-5-carboxamide
N-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide