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5-methoxy-2-[3-(thiophen-2-ylmethyl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]-1,4-dihydropyridin-4-one
(4aR,8aR)-2-methanesulfonyl-7-{pyrazolo[1,5-a]pyridine-3-carbonyl}-decahydro-2,7-naphthyridin-4a-ol
(1H-1,3-benzodiazol-2-ylmethyl)({[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl})methylamine
2-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-3-carbonitrile
N-[2-(ethylsulfanyl)ethyl]-4-(piperidin-1-ylmethyl)benzamide
N-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}imidazo[1,2-a]pyridine-2-carboxamide
1-(2-chlorophenyl)-3-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]urea
(3aR,6aR)-2-methyl-N-[(3,4,5-trimethoxyphenyl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
2-[2-({[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}(methyl)amino)pyrimidin-4-yl]pyridine-4-carboxylic acid
N-cyclohexyl-3-(2,5-dioxoimidazolidin-4-yl)-N-(pyridin-4-ylmethyl)propanamide
5-benzyl-4-(2-hydroxyacetyl)-1-(4-methylphenyl)piperazin-2-one
3-ethyl-1-{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}piperidine-3-carboxylic acid
1-(azocan-1-yl)-3-(2-methoxy-4-{[methyl(pyrimidin-4-ylmethyl)amino]methyl}phenoxy)propan-2-ol
N-[3-(dimethylamino)-2,2-dimethylpropyl]-6-methyl-2-(pyridin-3-yl)pyrimidin-4-amine
1-(3-methyl-1,2,4-thiadiazol-5-yl)-3-{1-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl}urea
N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
N-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]-4-(piperidin-1-ylmethyl)benzamide
N-({1-[(1-phenyl-1H-pyrazol-5-yl)methyl]pyrrolidin-3-yl}methyl)propanamide
1-acetyl-N-(2-{2-methyl-1-azatricyclo[6.3.1.04,12]dodeca-2,4,6,8(12)-tetraen-3-yl}ethyl)piperidine-3-carboxamide
N-methyl-3-{1-[(2E)-4-methylpent-2-enoyl]piperidin-3-yl}-N-(1-methylpiperidin-4-yl)propanamide
5-{dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}thiophene-2-carboxylic acid
N,N-dimethyl-5-({4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyridin-2-amine
methyl({2-[4-(4-methylpiperazine-1-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}){[4-(propan-2-yl)phenyl]methyl}amine
(1,4-dioxan-2-ylmethyl)(methyl){[3-(pyridin-2-ylmethoxy)phenyl]methyl}amine
6-ethyl-N,N-dimethyl-2-[2-(morpholin-4-yl)pyrimidin-5-yl]quinoline-4-carboxamide
2-[3-({methyl[2-(1-methyl-1H-pyrazol-4-yl)ethyl]carbamoyl}amino)phenyl]acetamide
(3S)-3-ethyl-4-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}morpholine
2-amino-4-(3-ethyl-1,2-oxazol-5-yl)-6-(4-hydroxyphenyl)-5-methylpyridine-3-carbonitrile
1-[3-(1H-imidazol-1-yl)propyl]-2-[5-(oxan-2-yl)furan-2-yl]-1H-imidazole
(2S,4S)-4-amino-1-[(2E)-3-(5-chloro-2-hydroxyphenyl)-2-methylprop-2-en-1-yl]-N-ethylpyrrolidine-2-carboxamide
4-[2-(3-tert-butyl-1,2,4-oxadiazol-5-yl)ethyl]phenol
4-methoxy-N-(2-methoxyethyl)-2-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}oxy)benzamide
3-(4-fluorophenyl)-N-(2-methoxyethyl)-N-(pyridin-4-ylmethyl)-1H-pyrazole-5-carboxamide
1-(4-{[2-(hydroxymethyl)phenyl]methyl}piperazin-1-yl)-3-(1-methylpiperidin-2-yl)propan-1-one
4-(4-fluorophenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]butan-1-one
2-(2-methoxyethyl)-8-[3-(2-methyl-1H-imidazol-1-yl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one
1-cyclobutanecarbonyl-4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine
4-[2-(benzenesulfonyl)ethyl]-1-[(3,4-dimethylphenyl)methyl]-1,4-diazepan-5-one
1-{4-[(4,4-difluoropiperidin-1-yl)methyl]-2-methoxyphenoxy}-3-(pyrrolidin-1-yl)propan-2-ol
7-[(4-ethylpiperazin-1-yl)sulfonyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
3-{1-[2-methyl-6-(trifluoromethyl)quinolin-4-yl]piperidin-3-yl}propanamide
1-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-3-[1-(propan-2-yl)-1H-1,2,3-triazol-4-yl]urea
ethyl 1-[3-(5-methylthiophen-2-yl)-5-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]piperidine-4-carboxylate
N-[3-(1H-imidazol-1-yl)propyl]-2-[2-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]acetamide
2-[1-(2-hydroxyethyl)-1H-pyrazol-4-yl]-7-methoxy-N,N-dimethylquinoline-4-carboxamide
2-(2-hydroxypropyl)-9-(2-methyl-1H-pyrrole-3-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
3-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}-N-{1,9-dioxaspiro[5.5]undecan-4-yl}propanamide
4-cyclobutaneamido-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]benzamide
2-[1-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperidin-3-yl]-1,3-benzoxazole
(2S,4R)-4-amino-N-methyl-1-[6-methyl-2-(pyridin-3-yl)quinoline-4-carbonyl]pyrrolidine-2-carboxamide