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N-{2-methyl-4-[3-(3-methylbutyl)-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl]pentan-2-yl}acetamide
N-[1-(2,5-difluorophenyl)cyclopropyl]-4-(piperidin-1-yl)butanamide
2-({4-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]phenyl}(methyl)amino)ethan-1-ol
3-({3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl}methyl)-N-methyl-1,2,4-oxadiazole-5-carboxamide
(3R,4R)-1-[2-(benzyloxy)ethyl]-3-methyl-4-(oxan-4-yl)piperidin-4-ol
1-(2-{7-[(2-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-2-oxoethyl)-1,2,3,6-tetrahydropyridazine-3,6-dione
N-(4-{[4-(3-cyanopyrazin-2-yl)piperazin-1-yl]methyl}phenyl)acetamide
N-[(3-chlorophenyl)methyl]-2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)-N-methylacetamide
4,6-dimethyl-5-{4-[1-(piperidin-1-yl)ethyl]phenyl}-1H-pyrazolo[3,4-b]pyridin-3-amine
N-benzyl-N-(1,1-dioxo-1λ6-thiolan-3-yl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
3-methyl-8-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
1-{[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-3-(3-fluorophenoxymethyl)piperidine
2-methyl-3-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidine-1-carbonyl]-4,5,6,7-tetrahydro-1-benzofuran-4-one
(1-{[2-fluoro-5-(trifluoromethyl)phenyl]methyl}-3-(2-methoxyethyl)piperidin-3-yl)methanol
2-methyl-N-{2-oxo-2-[3-oxo-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-9-yl]ethyl}propanamide
5-(2,5-dimethylphenoxymethyl)-N-methyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1,2-oxazole-3-carboxamide
2-ethyl-9-(6-oxo-1,6-dihydropyrimidine-5-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
1-{3,9-diazaspiro[5.6]dodecan-9-yl}-2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethan-1-one
7-(2,3-dimethyl-1H-indole-7-carbonyl)-N,N-dimethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
3-[1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)piperidin-4-yl]-N-(3-methoxyphenyl)propanamide
(1S,4S)-2-[4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]-2-azabicyclo[2.2.1]heptane
2-(1-{[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-2-yl)pyridine
N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}isoquinoline-1-carboxamide
1-[3-(dimethylamino)benzoyl]-N-(4-fluorophenyl)piperidin-3-amine
2-[2-(1H-imidazol-4-yl)ethyl]-8-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
4-(4-hydroxy-2-phenylpyrimidine-5-carbonyl)piperazin-2-one
N-(1-{7-[(3-ethoxy-4-hydroxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)pyridine-3-carboxamide
1-(3-chlorophenyl)-4-(2,4-dimethoxybenzoyl)piperazin-2-one
4-(2-aminopyrimidin-4-yl)-N-(pyridin-2-ylmethyl)piperazine-2-carboxamide
2-methoxy-N-{[1-(pent-2-yn-1-yl)-1,2,5,6-tetrahydropyridin-3-yl]methyl}acetamide
1-(3-methoxybenzoyl)-4-{pyrazolo[1,5-a]pyridine-3-carbonyl}piperazine
2-{[4-(trifluoromethyl)phenyl]methyl}-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-ethyl-2-{[3-(pyrrolidin-1-yl)piperidin-1-yl]methyl}-1H-1,3-benzodiazole
1-{2-[(4S)-4-hydroxy-3,3,4-trimethylpiperidin-1-yl]-2-oxoethyl}piperidin-2-one
N-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]-2-[4-(2-methylfuran-3-carbonyl)morpholin-3-yl]acetamide
4-[2-(adamantan-1-yl)acetyl]-3-(4-fluorophenyl)piperazin-2-one
3-[2-(6-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidine-1-carbonyl]-1,2,5,6,7,8-hexahydroquinolin-2-one
1-(1-{5H,6H-benzo[h]quinazolin-2-yl}-5-(methoxymethyl)-1H-pyrazole-4-carbonyl)-4-(piperidin-1-yl)piperidine
1-(4-hydroxyphenyl)-N-(2-methoxyethyl)-5-oxo-N-(thiophen-2-ylmethyl)pyrrolidine-3-carboxamide
5,6-dimethyl-2-oxo-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-1,2-dihydropyridine-3-carboxamide
1-[(1S,5R)-6-[5-(methoxymethyl)thiophene-2-carbonyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
6-{3-[(2-fluorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}pyrazine-2-carboxamide
(3-{2-[1-(5-methoxyfuran-2-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)dimethylamine
1-[(4-fluoro-3-methoxyphenyl)methyl]-N-[2-(4-methoxyphenyl)phenyl]piperidine-3-carboxamide
1-(4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-(1H-pyrazol-1-yl)ethan-1-one
4-[(5-ethylpyridin-2-yl)methyl]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-[4-({[(1-ethyl-1H-imidazol-2-yl)methyl]amino}methyl)-2-methoxyphenoxy]-3-(thiomorpholin-4-yl)propan-2-ol
[(3R,4R)-1-(3-chloro-4-fluorobenzoyl)-4-{[ethyl(methyl)amino]methyl}pyrrolidin-3-yl]methanol
N-benzyl-N-ethyl-6-(3-fluorophenyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
1-(8-methoxyquinolin-2-yl)-3-(piperidin-1-ylmethyl)pyrrolidin-3-ol