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2-[(2-{[(2-ethoxypyridin-3-yl)methyl]carbamoyl}phenyl)amino]acetic acid
6-fluoro-N,N-dimethyl-2-[2-(2-methyl-1,3-thiazol-4-yl)pyrimidin-5-yl]quinoline-4-carboxamide
4-chloro-2-({4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)phenol
5-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepane-1-carbonyl}-2-methylphenol
2-(4-fluorophenyl)-1-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]piperidine
3-{[(3aR,6aR)-2-methyl-octahydropyrrolo[3,4-c]pyrrol-3a-yl]formamido}-N-cyclohexylpropanamide
N-(3-fluoro-4-methylphenyl)-2-[3-(2-oxopyrrolidin-1-yl)piperidin-1-yl]acetamide
5,7-dimethyl-N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-[1,2,4]triazolo[4,3-a]pyrimidine-3-carboxamide
3-(3-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-yl}-3-oxopropyl)-5-methyl-2,3-dihydro-1,3-benzoxazol-2-one
4-(4-{[(3-methoxyphenyl)methyl](methyl)amino}piperidin-1-yl)-N-[2-(morpholin-4-yl)ethyl]benzamide
N-{[2-(azocan-1-yl)pyridin-3-yl]methyl}-5-oxopyrrolidine-3-carboxamide
5-tert-butyl-4-[(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)methyl]furan-2-carboxamide
1-methyl-N-(pyrimidin-4-ylmethyl)-1H-indole-3-carboxamide
N,N-dimethyl-1-[2-(propan-2-yl)-1,3-benzoxazole-5-carbonyl]pyrrolidin-3-amine
2-{1-[(4-methoxy-3-methylphenyl)methyl]-4-[(5-methylthiophen-2-yl)methyl]piperazin-2-yl}ethan-1-ol
N-[5-carbamoyl-2-(2-methylpiperidin-1-yl)phenyl]-N'-(3-fluorophenyl)ethanediamide
4-ethyl-3-{1-[2-(2-phenyl-1H-imidazol-1-yl)acetyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
propyl N-{2-[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)morpholin-2-yl]ethyl}carbamate
1-methyl-4-({6-[2-(methylsulfanyl)phenyl]pyridin-3-yl}methyl)piperazine
2-(3-methoxypropyl)-9-(1-phenylcyclopropanecarbonyl)-2,9-diazaspiro[5.5]undecan-3-one
(1R,3S)-3-amino-N-(2H-1,3-benzodioxol-5-ylmethyl)-N-(pyridin-4-ylmethyl)cyclohexane-1-carboxamide
1-{2-[(3aR,7aS)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-2-oxoethyl}-4-benzyl-3-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
3-[2-({[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}amino)ethyl]-1,3-oxazolidin-2-one
4-(1-methyl-1H-pyrazol-4-yl)-N-[4-(pyridin-2-yl)butyl]pyrimidin-2-amine
N-(3-chloro-4-methoxyphenyl)-7-methyl-3,7,11-triazaspiro[5.6]dodecane-11-carboxamide
methyl({4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl})[(trimethyl-1H-pyrazol-4-yl)methyl]amine
2-[(adamantan-1-ylmethyl)({[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl})amino]ethan-1-ol
N-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]-2-(2-phenyl-1H-imidazol-1-yl)acetamide
2-cyano-N-[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]benzamide
1-ethyl-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)piperidin-4-amine
2-({6-[4-(quinolin-4-ylmethyl)piperazin-1-yl]pyrimidin-4-yl}amino)ethan-1-ol
1-{1-[(2,4,6-trimethylphenyl)methyl]piperidin-3-yl}pyrrolidin-2-one
4-{[2-(3-hydroxypiperidin-1-yl)-6-methylquinolin-3-yl]methyl}piperazin-2-one
3-[5-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanoic acid
2-(4-fluorophenyl)-1-[4-(5-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]ethan-1-one
(3aS,6aR)-5-(1H-imidazol-4-ylmethyl)-3-[3-(morpholin-4-yl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
3-(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)-1-(6-hydroxy-1,4-oxazepan-4-yl)propan-1-one
N-[(3S,4R)-1-({4-amino-6-[(3-methylphenyl)amino]-1,3,5-triazin-2-yl}methyl)-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
N-(1H-1,2,3-benzotriazol-5-yl)-2-[2-(morpholin-4-yl)ethyl]piperidine-1-carboxamide
8-[2-(dimethylamino)-2-(2-methylphenyl)acetyl]-2-methyl-2,8-diazaspiro[4.5]decan-3-one
4-methyl-6-(4-phenylazepane-1-carbonyl)pyrimidin-2-amine
1-[(2R,6R)-2,6-bis(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]-2-(4-methyl-1,4-diazepan-1-yl)ethan-1-one
N-[1-(3-cyanopyridin-2-yl)piperidin-4-yl]-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)[(2-methyl-1,3-thiazol-4-yl)methyl]amine
5-{5-[2-(benzylsulfanyl)ethyl]-1,2,4-oxadiazol-3-yl}-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridine
1-(4-methylphenyl)-4-[2-(morpholin-4-yl)benzoyl]piperazin-2-one
1-[3-(azepan-1-ylmethyl)-6-methylquinolin-2-yl]piperidin-3-ol
2-({[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}(thiophen-2-ylmethyl)amino)ethan-1-ol
N-(1,3-benzothiazol-2-ylmethyl)-5-(3,4-dimethylphenoxymethyl)-1,2-oxazole-3-carboxamide
1-{2-[(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-oxoethyl}imidazolidine-2,4-dione