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1-(morpholin-4-yl)-3-(3-{[(3-phenylpropyl)amino]methyl}phenoxy)propan-2-ol
N-[3-(3-chlorophenyl)phenyl]-1-[(6-methylpyridin-2-yl)methyl]piperidine-4-carboxamide
(3S,4R)-4-(2-methoxyphenyl)-1-[2-(pyridin-4-ylsulfanyl)acetyl]pyrrolidine-3-carboxylic acid
4'-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-[(3-methylphenyl)methyl]-4-[6-(piperidin-1-yl)pyrimidin-4-yl]piperazin-2-one
5-[(2-fluoro-5-methoxyphenyl)methyl]-5-{3-oxo-3-[4-(pyrimidin-2-yl)-1,4-diazepan-1-yl]propyl}pyrrolidin-2-one
4-({2-[5-(ethanesulfonyl)thiophen-2-yl]phenyl}methyl)morpholine
3-(7,8-dimethyl-4-oxo-3,4-dihydroquinazolin-3-yl)-1λ6-thiolane-1,1-dione
methyl 1-{[4-(4-acetyl-1,4-diazepan-1-yl)quinazolin-2-yl]methyl}piperidine-2-carboxylate
N-[2-(1-oxo-1,2-dihydrophthalazin-2-yl)ethyl]-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
[(3R,4R)-1-[(2-fluoro-4-methylphenyl)methyl]-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
(2S,4R)-4-amino-1-[2-(2-hydroxyphenyl)-6-methylpyrimidin-4-yl]-N-methylpyrrolidine-2-carboxamide
2-{[1-(4,6-dimethylpyrimidin-2-yl)piperidin-4-yl]amino}-1-(3-fluorophenyl)ethan-1-ol
(2S,4R)-N-methyl-1-(propan-2-yl)-4-{[2-(2,6,6-trimethylcyclohex-1-en-1-yl)ethyl]amino}pyrrolidine-2-carboxamide
N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-1-(prop-2-en-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-{[3-cyclopropyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-2-fluorophenol
2-(methylsulfanyl)-3-{3-[4-(methylsulfanyl)benzoyl]piperidine-1-carbonyl}pyridine
1-[(3,5-dimethylphenyl)methyl]-4-[4-(2-methyl-1H-imidazol-1-yl)butanoyl]piperazin-2-one
2-[4-(difluoromethoxy)phenyl]-1-(propan-2-yl)-1H-imidazole
4-chloro-N-{2-[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]ethyl}-1H-pyrrolo[2,3-b]pyridin-6-amine
1-(2-fluorophenyl)-5-[2-(1H-imidazol-1-yl)ethyl]-3-(2-phenylethyl)-1H-1,2,4-triazole
N-{1-[1-(3,4-dimethylbenzoyl)piperidin-4-yl]-2-phenylethyl}-N-methylthiophene-2-carboxamide
(3aR,6aR)-2-acetyl-5-[(5-hydroxy-2-methoxyphenyl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(1S,6R)-9-{[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-3,9-diazabicyclo[4.2.1]nonan-4-one
[(5-cyclopropyl-1,2-oxazol-3-yl)methyl](methyl)[(1-methyl-1H-imidazol-5-yl)methyl]amine
1-benzyl-N3-cyclopropyl-N5-[(2,5-difluorophenyl)methyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2-({4-[(1,5-dimethyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazol-4-yl)methyl]-2-oxo-1-(2-phenylethyl)-1,4-diazepan-6-yl}oxy)-N,N-diethylacetamide
1-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-3-(5-methyl-1,2,4-oxadiazol-3-yl)piperidine
N,N,4-trimethyl-3-({[2-(1H-1,2,4-triazol-1-yl)ethyl]carbamoyl}methyl)-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-(1,3-thiazole-5-carbonyl)piperidine-4-carboxamide
1-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]-3-(pyridin-4-yl)propan-1-one
3-[(5-cyclopropyl-1,2-oxazol-3-yl)methyl]-3-methyl-1-[2-(propan-2-yl)phenyl]urea
N-[(2,5-dimethylphenyl)(pyridin-3-yl)methyl]-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
1-[4-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(4-fluorophenyl)-2-hydroxyethan-1-one
methyl 8-[3-(1H-1,3-benzodiazol-1-yl)propanoyl]-1-ethoxy-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indole-3-carboxamide
{4-[3-(2,6-dimethylphenoxy)azetidine-1-carbonyl]phenyl}methanol
(1-{[methyl(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)amino]methyl}cyclopentyl)methanol
(4aR,7aS)-1-methanesulfonyl-4-[3-(pyridin-3-yl)propanoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-{3,5-dimethyl-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl}-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethan-1-one
N-[(3S,4R)-4-ethoxyoxolan-3-yl]-3-azaspiro[5.5]undecan-9-amine
(3R,4R)-1-{[5-(4-chlorophenyl)furan-2-yl]methyl}-4-(4-methylpiperazin-1-yl)piperidin-3-ol
4-(4-{[3-(methoxymethyl)pyrrolidin-1-yl]methyl}phenyl)-2-methylbutan-2-ol
N-[2-(2-oxoimidazolidin-1-yl)ethyl]-3-(propan-2-yl)-1,2-oxazole-5-carboxamide
N-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]-3-(propan-2-yl)-1,2-oxazole-5-carboxamide
1-(2-methoxyphenyl)-5-[(methylsulfanyl)methyl]-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazole
2-(3-methoxypropyl)-9-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}-2,9-diazaspiro[5.5]undecan-3-one
1-[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-methoxyethan-1-one
methyl 3-(cyclobutylmethoxy)-5-{[(3R)-piperidin-3-yl]carbamoyl}benzoate
9-[(3,4-difluorophenyl)methyl]-2-(2-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one