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4-methyl-6-(propan-2-yl)-2-{4-[4-(pyrazin-2-yl)piperazine-1-carbonyl]piperidin-1-yl}quinazoline
9-{3-[(dimethylamino)methyl]benzoyl}-1-oxa-9-azaspiro[5.5]undecan-5-ol
N-cyclopropyl-N-[(3-hydroxyphenyl)methyl]-2-methyl-4-phenylpyrimidine-5-carboxamide
1-(furan-3-carbonyl)-4-{[1-(2-hydroxyethyl)-3-methyl-1H-pyrazol-4-yl]methyl}-1,4-diazepan-6-ol
N-[(4-fluorophenyl)methyl]-N-(3-methoxypropyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
2-(1H-indol-3-yl)-N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}acetamide
N-[4-(morpholin-4-ylmethyl)phenyl]-1H-indazole-3-carboxamide
N-methyl-N-[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]-2-[1-(3-methylbut-2-en-1-yl)-3-oxopiperazin-2-yl]acetamide
4-ethyl-3-{1-[5-(1H-imidazol-2-yl)thiophene-2-carbonyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(2-ethylbutanoyl)-N-[3-(4-fluorophenyl)phenyl]piperidine-3-carboxamide
methyl (2S)-2-phenyl-2-({1-[4-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)phenyl]piperidin-4-yl}amino)acetate
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-3-hydroxy-4-methylbenzamide
N-(2,6-dimethylphenyl)-3-[3-(3-hydroxy-1,2-oxazol-5-yl)propanamido]benzamide
2-(4-{[3-(ethoxymethyl)-4-methoxyphenyl]methyl}-1-[(2-ethoxyphenyl)methyl]piperazin-2-yl)ethan-1-ol
N-{[4-(2,3-dihydro-1H-inden-2-yloxy)-3-methoxyphenyl]methyl}-3,5-dimethoxy-N-(oxolan-2-ylmethyl)benzamide
1-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-3-(4-ethyl-1,3-dimethyl-1H-pyrazol-5-yl)urea
6-[(2E)-3-(4-fluorophenyl)prop-2-enoyl]-N-[2-(pyridin-2-yl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
3-[4-(2-methylphenyl)-1H-pyrazol-5-yl]-1-[4-(methylsulfanyl)benzoyl]piperidine
3,5-dimethyl-N-{2-[3-(1-methyl-1,2,3,6-tetrahydropyridin-4-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1,2-oxazole-4-carboxamide
N-[(3R,7S,8aS)-3-benzyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-ethylbenzamide
2-[2-(4-methylpentyl)morpholine-4-carbonyl]-4-(1H-pyrrol-1-yl)phenol
3-(4-acetylpiperazin-1-yl)-N-(2,6-diethylphenyl)propanamide
(1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}-3-(2-phenoxyethyl)piperidin-3-yl)methanol
2-[(2R,3S,6R)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-1,3-thiazole-4-carboxamide
2-[({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}amino)methyl]-3,4-dihydroquinazolin-4-one
1-[(1-methylpyrrolidin-3-yl)methyl]-4-phenyl-5-(3-phenyl-1H-pyrazol-4-yl)-1H-imidazole
1-(6-ethoxy-4-methylquinazolin-2-yl)-N-[2-(pyrazin-2-yl)ethyl]piperidine-3-carboxamide
N-[2-(methylsulfanyl)ethyl]-2-{3-oxo-1-[(3-phenoxyphenyl)methyl]piperazin-2-yl}acetamide
diethyl[(4-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine-8-carbonyl}-5-methylfuran-2-yl)methyl]amine
N-[(1R,3S)-3-[(2-methoxyethyl)(methyl)carbamoyl]cyclopentyl]-2H,3H-thieno[3,4-b][1,4]dioxine-5-carboxamide
1-[(1-butyl-2-cyclobutylmethanesulfonyl-1H-imidazol-5-yl)methyl]-3-methoxypiperidine
(2S)-1-acetyl-N-{[5-(2-acetylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}pyrrolidine-2-carboxamide
bis(1,3-oxazol-4-ylmethyl)({[5-(oxolan-2-yl)thiophen-2-yl]methyl})amine
1-[(1-methyl-1H-imidazol-2-yl)methyl]-3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidine
{1-[5-(2,6-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]piperidin-4-yl}(pyridin-2-yl)methanol
N-({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)-2-methoxypyrimidine-5-carboxamide
2-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-2,7-diazaspiro[4.5]decane
(2R)-2-amino-3-(4-chlorophenyl)-N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]propanamide
[(3aS,6aS)-2-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]-octahydrocyclopenta[c]pyrrol-3a-yl]methanol
3-(2-hydroxy-2-phenylethyl)-3H,4H-pyrido[2,3-d]pyrimidin-4-one
2-[({[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)methyl]benzonitrile
2-[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]ethan-1-ol
1-(3,5-dimethylphenyl)-4-[2-(hydroxymethyl)-1H-1,3-benzodiazole-5-carbonyl]piperazin-2-one
(3R,5S)-N-(2,3-dihydro-1H-inden-5-yl)-1-(2-methylpropyl)-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxamide
[4-(4-methanesulfonylphenyl)phenyl]methanamine
1-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-[3-(4H-1,2,4-triazol-4-yl)benzoyl]piperazine
N-[(1-benzylpiperidin-4-yl)methyl]-N-methyl-2-(2-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetamide
(1R,4S)-1,7,7-trimethyl-4-{4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-2-oxabicyclo[2.2.1]heptan-3-one
N,N-dimethyl-1-{7-[(4-methyl-1H-imidazol-5-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}pyrrolidin-3-amine
2-chloro-6-methoxy-3-(6-methyl-1H-1,3-benzodiazol-2-yl)phenol