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(1S,5R)-3-(5-methyl-1,2-oxazole-3-carbonyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
5-{[4-(5-chloropyridin-2-yl)piperazin-1-yl]methyl}-2-ethylpyrimidine
4-ethyl-1-methyl-3-({1-[5-(2-methylpropyl)-1,2-oxazole-3-carbonyl]piperidin-4-yl}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
9-methoxy-4-[(1-methyl-1H-pyrazol-4-yl)methyl]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-(3-methoxypropyl)-9-(2-methyl-1H-1,3-benzodiazole-5-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[2-(dimethylamino)ethyl]-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-6-oxopiperidine-3-carboxamide
3-(2-{1-[(3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamido)propanamide
ethyl 4-({[5-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-3-yl]methyl}amino)piperidine-1-carboxylate
N-[1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-4-oxo-4H-chromene-2-carboxamide
N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
{1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-3-(2-phenoxyethyl)piperidin-3-yl}methanol
1-(1H-1,2,3-benzotriazol-5-yl)-3-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]urea
4-chloro-N,N-dimethyl-5-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1H-imidazol-2-yl}-1,3-thiazol-2-amine
4-[(2-aminopyrimidin-5-yl)methyl]-7-(1-benzothiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
methyl 6-(2-{[2-(2-oxo-4-phenylpyrrolidin-1-yl)acetamido]methyl}-2,3-dihydro-1-benzofuran-7-yl)pyridine-3-carboxylate
N-[(1R,3S)-3-(thiomorpholine-4-carbonyl)cyclopentyl]-1H-indazole-3-carboxamide
4-[(1H-imidazol-2-ylmethyl)sulfamoyl]-N-(oxolan-2-ylmethyl)benzamide
N-(3-methylphenyl)-3-{1-[2-(pyridin-3-yl)acetyl]piperidin-4-yl}propanamide
1-(2-{3-methyl-2-oxo-1-oxa-3,7-diazaspiro[4.4]nonan-7-yl}-2-oxoethyl)-1H-indole-3-carboxamide
(1R,5R)-6-{2,7-dimethylimidazo[1,2-a]pyridine-3-carbonyl}-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-2,8-diazaspiro[4.5]decane-3-carboxamide
2-oxo-8-[(1-propyl-1H-pyrazol-4-yl)sulfonyl]-1,8-diazaspiro[4.5]decane-4-carboxylic acid
4-(piperidin-1-yl)-N-{[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}butanamide
2-benzyl-4-(2-phenylethyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
methyl 2-(5-chloro-2-methoxyphenyl)-1H-1,3-benzodiazole-6-carboxylate
5-acetyl-N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methylthiophene-2-carboxamide
1-methyl-3-{[2-(pyridin-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]amino}pyrrolidin-2-one
1-(propan-2-yl)-N-{[4-(pyrrolidine-1-carbonyl)phenyl]methyl}-1H-pyrazole-4-carboxamide
(2S,4S)-N,N-diethyl-4-{4-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-1H-1,2,3-triazol-1-yl}pyrrolidine-2-carboxamide
2-{2-[(pentan-3-yl)amino]pyrimidin-4-yl}pyridine-4-carboxylic acid
1-[(2-ethylpyrimidin-4-yl)methyl]-4-(2-fluorophenoxy)piperidine-4-carboxylic acid
8-(cyclopropanesulfonyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
1-(4-chloro-2-fluorophenyl)-3-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}urea
2-[1-(1-methylpiperidin-4-yl)-5-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-3-yl]pyridine
5-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)-1-(cyclohexylmethyl)piperidin-2-one
1-{4-[3-(hydroxymethyl)-3-(2-phenylethyl)piperidine-1-carbonyl]thiophen-2-yl}ethan-1-one
3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)piperidine
3-[(4-methyl-1,2,3,6-tetrahydropyridin-1-yl)sulfonyl]-N-(oxolan-3-yl)benzamide
4-(5-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridin-2-yl)thiomorpholine
1-[1-(3-cyclopentylpropanoyl)piperidin-4-yl]-N-(2-methoxyethyl)-1H-1,2,3-triazole-4-carboxamide
(3R,4S)-1-{2-[(4-methylphenyl)methyl]benzoyl}-4-propylpyrrolidin-3-amine
N,N-diethyl-2-{[2-oxo-1-(2-phenylethyl)-4-(4,4,4-trifluorobutanoyl)-1,4-diazepan-6-yl]oxy}acetamide
3-(4-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)-N,N-dimethylaniline
methyl 6-(2,3-dihydro-1-benzofuran-5-ylmethyl)-2-[(4-methylphenyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
(2S,4S)-1-[(4-chlorophenyl)methyl]-4-{[(2,6-difluorophenyl)methyl]amino}-N-ethylpyrrolidine-2-carboxamide
[1-(1-phenoxypropan-2-yl)-4-(2-phenylethyl)piperidin-4-yl]methanol
N-(pyridin-2-ylmethyl)-1-[1-(1,3-thiazole-4-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
(3S,5R)-1-[(3-hydroxyphenyl)methyl]-5-[(pyridin-4-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
4-{1-[(5-methyl-1,2-oxazol-3-yl)methyl]-1H-imidazol-2-yl}benzoic acid
5-(5-methyl-2-phenyl-1H-imidazole-4-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid