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N-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-2-{2-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}acetamide
2-(4-{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}-1-cyclopentylpiperazin-2-yl)ethan-1-ol
3-{1-[2-(2H-1,2,3-benzotriazol-2-yl)acetyl]piperidin-3-yl}-N-[(3-methoxyphenyl)methyl]propanamide
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-methyl-1H-pyrrole-3-carboxamide
(1R,7S)-3-[(2,5-dimethylphenyl)methyl]-N-methyl-4-oxo-N-(1H-pyrazol-3-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
N-phenyl-5-[4-(pyridin-2-ylmethyl)piperazine-1-carbonyl]pyrimidin-2-amine
(3aS,6aR)-5-[(2-chloro-6-fluorophenyl)methyl]-3-[2-(piperidin-1-yl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
6-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}pyridine-2-carbonitrile
4-[1-(4-chlorophenyl)cyclopropanecarbonyl]-1-(2-methoxyphenyl)piperazin-2-one
2-[1-benzyl-5-(4-sulfamoylphenyl)-1H-1,2,4-triazol-3-yl]acetamide
N-[(3R,5S)-5-(methylcarbamoyl)-1-[2-(pyridin-2-yl)acetyl]pyrrolidin-3-yl]pyridine-4-carboxamide
6-(1-methyl-1H-1,2,4-triazol-5-yl)-1,2,3,4-tetrahydroquinoxaline-2,3-dione
8-[4-(dimethylamino)-5-methylpyrimidin-2-yl]-2-(3-hydroxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
9-[5-(methoxymethyl)thiophene-2-carbonyl]-2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecane
N-(2,4-dimethylphenyl)-N'-{1-[4-(1H-1,2,4-triazol-1-yl)phenyl]ethyl}propanediamide
4-benzyl-3-[2-oxo-2-(pyrrolidin-1-yl)ethyl]piperazin-2-one
4-({2-[3-(1-methyl-1H-imidazole-2-carbonyl)phenyl]phenyl}methyl)morpholine
methyl 3-[(3S,4R)-1-(adamantan-2-yl)-4-(pyrrolidin-1-yl)piperidin-3-yl]propanoate
4-(cyclohex-3-ene-1-carbonyl)-1-[(2-methyl-1,3-thiazol-4-yl)methyl]-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
methyl 3-[(2,3-difluorophenyl)methyl]-7-oxo-9-[3-(pyridin-3-yl)propoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-(5-methyl-1-propyl-1H-pyrazole-4-amido)-1,2,3,4-tetrahydronaphthalene-1-carboxylic acid
2-{[6-(hydroxymethyl)-1,4-oxazepan-4-yl]methyl}benzoic acid
N-[3-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]-6-oxo-1,6-dihydropyrimidine-5-carboxamide
{[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}[2-(1H-pyrazol-1-yl)ethyl]amine
5-{[3-(4-fluorophenyl)pyrrolidin-1-yl]methyl}-3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazole
(4aS,7aR)-4-[2-(dimethylamino)acetyl]-N,N-dimethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
(3R,5S)-1-benzyl-N-(2-methylpropyl)-5-{[(6-methylpyridin-3-yl)oxy]methyl}piperidine-3-carboxamide
1-{2-[4-(1H-imidazol-2-yl)-1H-1,2,3-triazol-1-yl]ethyl}piperidine-3-carboxamide
N-[(3R,4S)-4-cyclopropyl-1-{[2-methoxy-5-(propan-2-yl)phenyl]methyl}pyrrolidin-3-yl]-2-hydroxyacetamide
N-(1-butyl-4-methyl-1H-pyrazol-5-yl)-3-fluoro-4-methoxybenzamide
5-cyclobutanecarbonyl-1'-(pyridin-3-ylmethyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
7-(propan-2-yl)-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
1-[(1-propyl-1H-imidazol-2-yl)methyl]-3-(4H-1,2,4-triazol-3-yl)piperidine
1-phenyl-4-[4-(pyrrolidin-1-ylmethyl)benzoyl]piperazin-2-one
methyl 4-[(2-butyl-4-methyl-3-oxopiperazine-1-carbonyl)amino]benzoate
ethyl 1-{[4-(methoxycarbonyl)phenyl]carbamoyl}-4-(oxan-2-ylmethyl)piperidine-4-carboxylate
5-methyl-1-[4-(pyridin-3-yl)pyrimidin-2-yl]-N-[3-(pyridin-4-yl)propyl]-1H-pyrazole-4-carboxamide
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-[1-(2-methylpropyl)-3-oxopiperazin-2-yl]acetamide
3-[3-(3-methoxyphenoxy)azetidine-1-carbonyl]-N,N-dimethylpiperidine-1-carboxamide
(2R,3R,6R)-3-(3-methoxyphenyl)-5-(6-methoxypyrimidin-4-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-methyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
1-[2-(azepan-1-yl)-2-oxoethyl]-4-benzylpyrrolidin-2-one
ethyl 4-(3-benzyl-4,5-dihydro-1,2-oxazole-5-amido)piperidine-1-carboxylate
(4aR,7aS)-4-[(3,4-dimethylphenyl)methyl]-N,N-dimethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
1-{2-[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperazin-1-yl]-2-oxoethyl}azepan-2-one
4-[(4-{3-[benzyl(methyl)amino]-2-hydroxypropoxy}phenyl)methyl]-1-methylpiperazin-2-one
2-[5-({3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}carbamoyl)pyridin-2-yl]benzoic acid
(2S,4S)-4-{[(3-chlorophenyl)methyl]amino}-N-ethyl-1-(2-methylpropyl)pyrrolidine-2-carboxamide
methyl 3-cyclopropaneamido-6-{[3-(diethylcarbamoyl)piperidin-1-yl]methyl}thieno[2,3-b]pyridine-2-carboxylate
2-ethyl-1-(propan-2-yl)-4-[4-(1H-pyrazol-3-yl)benzoyl]piperazine