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2-(5-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}-1H-pyrazol-3-yl)phenol
methyl 1-[(3R,5S)-1-benzyl-5-{[2-(3-chlorophenyl)ethyl]carbamoyl}pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
methyl({[8-methyl-2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})[2-methyl-3-(pyrrolidin-1-yl)propyl]amine
N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-N,3-dimethyl-4-oxo-3,4-dihydrophthalazine-1-carboxamide
2-ethyl-N-[6-(propan-2-yloxy)-1-(2,2,2-trifluoroethyl)-1H-indazol-3-yl]pyrimidine-5-carboxamide
5-{[(2,4-difluorophenyl)methyl]amino}-N-(furan-2-ylmethyl)-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-[2-methyl-3-(1H-1,2,4-triazol-1-yl)propanoyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
3-{1-[(1-hexylpiperidin-4-yl)methyl]-1H-1,2,3-triazol-4-yl}propan-1-ol
{3-[(4-fluorophenyl)methyl]-1-methylpiperidin-3-yl}methanol
({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)(methyl)(pyridin-3-ylmethyl)amine
(3S)-3-benzyl-4-(cyclopentylmethyl)piperazin-2-one
(4aR,7aS)-N,N-dimethyl-4-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
N-(2-chloro-4,6-dimethylphenyl)-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
N-[1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
N,N-dimethyl-3-{3-[({2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}carbamoyl)amino]phenyl}propanamide
2-(3-cyclopropyl-1H-1,2,4-triazol-5-yl)-5,7-dimethylquinolin-8-ol
1-{5-[3-(phenylamino)piperidine-1-carbonyl]thiophen-2-yl}ethan-1-one
3-(2H-1,3-benzodioxol-5-yl)-N-ethyl-N-[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]propanamide
(3R,4S)-4-[4-(3,5,7-trimethyl-1H-indole-2-carbonyl)-1,4-diazepan-1-yl]oxolan-3-ol
1-methyl-9-(prop-2-en-1-yl)-4-{[1,2,4]triazolo[1,5-a]pyrimidin-2-ylmethyl}-1,4,9-triazaspiro[5.6]dodecan-10-one
3-(1-hydroxy-3-methylbutan-2-yl)-7,8-dimethyl-3,4-dihydroquinazolin-4-one
N-[1-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-3,6-dimethyl-1-benzofuran-2-carboxamide
3-({[2-(2,4-dimethylphenoxy)ethyl](methyl)amino}methyl)-5-methyl-1H-indole-2-carboxylic acid
N-(2-fluorophenyl)-4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carboxamide
4-phenyl-3-(piperidin-3-yl)-1-[2-(1H-pyrrol-1-yl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
3-[5-(furan-2-yl)-1,3,4-thiadiazol-2-yl]-1-[2-(5-methylthiophen-2-yl)ethyl]urea
3-(propan-2-yl)-5-(1-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}pyrrolidin-2-yl)-1,2,4-oxadiazole
7-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-4-(furan-3-ylmethyl)-9-(oxolan-2-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-{[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazol-4-yl]methyl}-1-(oxolan-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
1-{2-[3-cyclopropyl-1-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-1,2,4-triazol-5-yl]ethyl}-6-methyl-1,2-dihydropyridin-2-one
5-chloro-N-(oxolan-2-ylmethyl)-N-({4-[2-(pyridin-2-yl)ethoxy]phenyl}methyl)thiophene-2-sulfonamide
(2S,4S)-4-amino-1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
(3R,4R)-4-(2-ethyl-4-methyl-1H-imidazol-5-yl)-1-methyl-N-(oxan-4-yl)pyrrolidine-3-carboxamide
2-(2,6-dioxo-1,3-diazinan-1-yl)-N-ethyl-N-[(2E)-3-phenylprop-2-en-1-yl]acetamide
1-[5-(4-methoxyphenyl)furan-2-carbonyl]-3-(pyrrolidine-1-carbonyl)piperidine
3-(3-fluorophenyl)-4-{[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}piperazin-2-one
(1S,5R)-6-(1H-indol-5-ylmethyl)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
2-amino-3-ethyl-N-{imidazo[1,2-a]pyrimidin-2-ylmethyl}-3H-imidazo[4,5-b]pyridine-6-carboxamide
3-ethoxy-N-ethyl-N-(2-methoxyethyl)-4-(prop-2-en-1-yloxy)benzamide
N,N-diethyl-4-{[2-(2-fluorophenyl)ethyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
5-{[1-(2,3-dihydro-1H-inden-5-yl)-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]methyl}imidazolidine-2,4-dione
4-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]-N-methyl-N-(2-methylpropyl)morpholine-2-carboxamide
2-amino-6-cyclobutyl-4-[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]pyridine-3-carbonitrile
5-(3-benzyl-1,2,4-oxadiazol-5-yl)-N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]pyridin-2-amine
3-(2,2-difluoroethyl)-1-(2-fluoro-4-methylphenyl)urea
1-(2-{[5-(methoxymethyl)thiophen-2-yl]formamido}ethyl)piperidine-3-carboxamide
7-acetamido-N-methyl-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]-1-[2-(pyridin-2-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
6-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)-3-(propan-2-yl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-N-methyl-2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
1-(4-{1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperazin-1-yl)ethan-1-one