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ethyl 4-(2-phenylethyl)-1-[3-(pyrazin-2-yl)propanoyl]piperidine-4-carboxylate
1-[6-ethyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-N-[(5-methylpyrazin-2-yl)methyl]piperidin-4-amine
2-(ethylsulfanyl)-5-{[3-(4-methylpiperazin-1-yl)pyrrolidin-1-yl]methyl}pyrimidine
3,5-dichloro-N,4-dimethyl-N-[1-(1,3-thiazol-5-yl)ethyl]benzamide
N-benzyl-2-(2-oxopiperidin-1-yl)-N-(2,2,2-trifluoroethyl)acetamide
(3R,5S)-N-(4-fluorophenyl)-1-(pyridin-4-ylmethyl)-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxamide
(5-methyl-7-{8-methyl-2H-[1,3]dioxolo[4,5-g]quinolin-6-yl}-2,3-dihydro-1-benzofuran-2-yl)methanamine
(3aS,6aR)-3-[2-(4-methoxyphenyl)ethyl]-5-(3-methylbut-2-en-1-yl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
(1R,5R)-6-(cyclopropylmethyl)-3-{imidazo[1,2-a]pyrimidine-2-carbonyl}-3,6-diazabicyclo[3.2.2]nonane
N-[(3,4-dimethoxyphenyl)methyl]-1-ethyl-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-(4-butyl-2,3-dioxopiperazin-1-yl)-N-methyl-N-(1-methylpiperidin-4-yl)-2-phenylacetamide
6-(2-aminoethyl)-N,2-dimethyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrimidin-4-amine
{[2-(2-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl){[3-(1H-pyrazol-1-yl)phenyl]methyl}amine
N-(3-cyclopentylpropyl)-1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-methylpiperidine-3-carboxamide
9-[3-(dimethylamino)pyrazin-2-yl]-2-[3-(1H-imidazol-1-yl)propyl]-2,9-diazaspiro[5.5]undecan-3-one
2-[3-({[(3,4-dimethylphenyl)methyl]amino}methyl)-2-methyl-1H-indol-1-yl]acetamide
N-methyl-2-{3-oxo-2-azaspiro[4.4]nonan-2-yl}-N-(thiophen-3-ylmethyl)acetamide
N-[2-(2-fluorophenyl)ethyl]-3-methoxy-4-[(1-methylpiperidin-4-yl)oxy]benzamide
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-2-oxo-1,2-dihydroquinoline-4-carboxamide
N-cyclopentyl-3-{[(3,5-dimethoxyphenyl)methyl]amino}-5-(phenylsulfamoyl)benzamide
1-{4-[2-(ethoxymethyl)pyrrolidine-1-carbonyl]phenyl}-3,5-dimethyl-1H-pyrazole
N-{1-[4-(3-chlorophenyl)-5-({[3-(trifluoromethyl)phenyl]methyl}sulfanyl)-4H-1,2,4-triazol-3-yl]ethyl}-2-(pyridin-2-ylsulfanyl)acetamide
ethyl 5-(furan-3-ylmethyl)-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-(5-chloro-1H-1,3-benzodiazol-2-yl)-N-{2-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}acetamide
(1S,5R)-3-cyclobutanecarbonyl-6-(2-methyl-1,3-thiazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
4-{octahydropyrrolo[1,2-a]piperazine-2-carbonyl}-1-(2-phenylethyl)-1H-1,2,3-triazole
1-(2-{[2-(cyclopropylamino)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]amino}ethyl)imidazolidin-2-one
N-(2-fluoroethyl)-5-(2-methoxyphenoxymethyl)-1H-pyrazole-3-carboxamide
(3R,5S)-1-[(3,4-dimethoxyphenyl)methyl]-N3-(4-fluorophenyl)-N5-(thiophen-2-ylmethyl)piperidine-3,5-dicarboxamide
4-(6-cyclopropylpyrimidin-4-yl)-2-(3,4-dichlorophenyl)morpholine
ethyl 4-{[3-(naphthalene-1-carbonyl)piperidin-1-yl]methyl}-1H-pyrazole-3-carboxylate
9-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]-2-[(1r,4r)-4-hydroxycyclohexyl]-2,9-diazaspiro[5.5]undecan-3-one
1-cyclopropyl-N-{[1-(2-fluorophenyl)cyclopentyl]methyl}-5-oxopyrrolidine-3-carboxamide
2,5,7-trimethyl-3-[(3-propyl-1,2,4-oxadiazol-5-yl)methyl]-1H-indole
N4-ethyl-N2-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}pyrimidine-2,4-diamine
N-(5-methyl-2-pentanamidophenyl)quinoxaline-5-carboxamide
N-cyclopropyl-6-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyridazin-3-amine
4-[4-(2-chlorophenyl)piperidin-4-yl]-N-[2-(1H-imidazol-1-yl)ethyl]pyrimidin-2-amine
2-[(3-methoxyphenyl)methyl]-8-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-2,8-diazaspiro[4.5]decan-3-one
6-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecan-4-yl]pyrimidine-2,4-diamine
N-benzyl-N,1-dimethyl-5-(morpholin-4-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
4-{3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidine
methyl 5-[4-(2-methylphenoxy)piperidin-1-yl]-5-oxopentanoate
1-ethyl-8-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-7-methylpyrazolo[1,5-a]pyrimidine-6-carboxamide
N-[(2S,4R,6S)-2-(2,1,3-benzoxadiazol-5-yl)-6-ethyloxan-4-yl]benzamide
4-{[3-(3-fluoro-4-phenylbenzoyl)piperidin-1-yl]methyl}-1H-pyrazole-3-carboxylic acid
8-chloro-2-{[4-hydroxy-4-(1H-imidazol-1-ylmethyl)piperidin-1-yl]methyl}quinolin-4-ol
4-(8-hydroxyquinolin-2-yl)-N-methyl-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxamide
1,5,6-trimethyl-N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)-2-oxo-1,2-dihydropyridine-3-carboxamide