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N-{2-[(4-chlorophenyl)methoxy]ethyl}-3-(1-methylpiperidin-4-yl)propanamide
(2S,4R)-4-amino-1-(3,5-difluoro-4-methoxybenzoyl)-N-methylpyrrolidine-2-carboxamide
4-(2-methoxyphenyl)-2-methyl-1-[3-(thiophen-2-yl)-1H-pyrazole-4-carbonyl]piperazine
(2S,4R)-4-amino-1-[(2-aminopyridin-3-yl)methyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-[3-(furan-2-yl)propyl]-2-(1H-pyrazol-1-yl)butanamide
N-cyclopropyl-3-(4-fluorophenyl)-N-({4-[(3-methyloxetan-3-yl)methoxy]phenyl}methyl)benzamide
ethyl 1-[4-(dimethylamino)benzoyl]-4-[(4-methoxyphenyl)methyl]piperidine-4-carboxylate
1-{1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}-4-[3-(trifluoromethyl)phenyl]piperazine
methyl 2-({1-[(3-methoxyphenyl)methyl]piperidin-3-yl}amino)-6-methylpyrimidine-4-carboxylate
4-[5-(1-cyclohexylpiperidin-4-yl)-1,2,4-oxadiazol-3-yl]pyridine
4-[7-(5-propylthiophene-3-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]morpholine
1-[(1-methylpiperidin-4-yl)methyl]-4-(5-phenyl-1,2-oxazole-4-carbonyl)piperazine
N-[1-(3-ethyl-1,2-oxazol-5-yl)ethyl]-4-[(2-methylprop-2-en-1-yl)oxy]benzamide
2-{[2-(3-fluorophenyl)acetamido]methyl}-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
6-(2-aminoethyl)-N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]pyrimidin-4-amine
2-(methylsulfanyl)-4-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine
N-[(2S)-1-hydroxy-3-phenylpropan-2-yl]-2-methyl-3-[(pyridin-3-ylmethyl)amino]benzamide
8-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
2-(ethoxymethyl)-7-(furan-3-ylmethyl)-N-methyl-N-(prop-2-en-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
5-[1-(2H-1,3-benzodioxol-5-ylmethyl)-1H-1,2,4-triazol-5-yl]-4-methyl-1,3-thiazol-2-amine
11-(5-methyl-4-{[(5-methylfuran-2-yl)methyl]amino}thieno[2,3-d]pyrimidine-6-carbonyl)-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
4-(methylsulfanyl)-N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}benzamide
2-[1-(3-methylbutyl)-1H-pyrazol-4-yl]-2-(morpholin-4-yl)acetic acid
3-(dimethyl-1,2-oxazol-4-yl)-N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}propanamide
(2S,4S)-N-ethyl-4-(2-hydroxy-5-methylbenzamido)-1-(oxan-4-yl)pyrrolidine-2-carboxamide
(1R,5R)-N,N-dimethyl-6-{7-oxo-7H-[1,3]thiazolo[3,2-a]pyrimidine-5-carbonyl}-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
5-{1-[5-(1H-imidazol-4-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}-1H-1,2,4-triazole
2-methoxy-5-{2-[2-(propan-2-yl)pyrimidin-5-yl]-1H-imidazol-1-yl}benzoic acid
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-[6-(propan-2-yl)pyridin-2-yl]pyrrolidin-3-yl]methanol
3-methanesulfonyl-N-methyl-N-[1-(pyridin-2-yl)ethyl]benzamide
{1-[2-amino-6-(pyrrolidin-1-yl)pyrimidin-4-yl]-3-(prop-2-en-1-yl)piperidin-3-yl}methanol
N-{2-[3-cyclopentyl-1-(2-methylphenyl)-1H-1,2,4-triazol-5-yl]ethyl}methanesulfonamide
4-[3-(4-cyclohexyl-1,4-diazepane-1-carbonyl)phenyl]-2-methylbutan-2-ol
8-(3,5,7-trimethyl-1H-indole-2-carbonyl)-1,3-dioxa-8-azaspiro[4.5]decan-2-one
4-(2-methylpropyl)-3-[2-(1,2-oxazinan-2-yl)-2-oxoethyl]piperazin-2-one
N-[(1,2-dimethyl-1H-1,3-benzodiazol-5-yl)methyl]-4-(3-hydroxy-3-methylbutyl)benzamide
N-[3-(4-methylpiperazin-1-yl)propyl]imidazo[1,2-a]pyridine-6-carboxamide
1-tert-butyl-N-{1-[(2-chlorophenyl)methyl]-5-oxopyrrolidin-3-yl}-1H-pyrrole-3-carboxamide
N-[(2-methylphenyl)methyl]-2-[3-(2-oxopyrrolidin-1-yl)piperidin-1-yl]acetamide
1-(2-methylpropyl)-4-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]-1,4-diazepane
2-[3-(oxolan-3-yl)-5-[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]-1H-1,2,4-triazol-1-yl]acetic acid
[(3R,4R)-4-{[ethyl(methyl)amino]methyl}-1-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}pyrrolidin-3-yl]methanol
7-{[3-(2-methylpiperidin-1-yl)azetidin-1-yl]methyl}-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
4-(3-fluorophenoxy)-1-(2-oxo-2,3-dihydro-1H-imidazole-4-carbonyl)piperidine-4-carboxylic acid
7-[(6-methylquinolin-8-yl)sulfonyl]-2,7-diazaspiro[4.4]nonane-1,3-dione
2-[1-(2,2-diphenylethyl)-3-oxopiperazin-2-yl]-N-[2-(4-methyl-1H-imidazol-2-yl)ethyl]acetamide
3-({[(3-chlorophenyl)methyl](methyl)amino}methyl)-1,2-dihydroquinolin-2-one
(1S,4S)-2-{[3-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-4-yl]methyl}-2-azabicyclo[2.2.1]heptane
4-methyl-2-[1-(6-methylpyridine-3-carbonyl)piperidin-4-yl]-1H-1,3-benzodiazole
N-[3-(1,3-thiazol-4-yl)phenyl]-1-(thiophen-3-ylmethyl)piperidine-4-carboxamide