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2-cyclopropyl-6-[4-(2,6-dimethylpyridin-4-yl)piperazine-1-carbonyl]-1,3-benzoxazole
5-(2,6-dimethylphenoxymethyl)-N-(1H-indol-2-ylmethyl)-1,2-oxazole-3-carboxamide
2-amino-6-(3,5-dimethyl-1H-pyrazol-4-yl)-4-[4-methoxy-3-(methoxymethyl)phenyl]pyridine-3-carbonitrile
1-(5-tert-butyl-2-methoxyphenyl)-3-methyl-3-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]urea
(1R,5R)-6-[2-(1H-imidazol-2-yl)benzoyl]-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane
(1-{[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)methanol
(1R,5S,6R)-3-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-N-(pyridin-3-ylmethyl)-3-azabicyclo[3.1.0]hexane-6-carboxamide
3-methyl-1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]-3-{[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}urea
[(4-chloro-3-fluorophenyl)methyl]({1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
4-(1-methyl-1H-pyrazol-4-yl)-2-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}pyrimidine
3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-1-[(4-methoxy-3-methylphenyl)methyl]piperidine
1-[1-(furan-3-ylmethyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
1-(3-{2-[(4-fluorophenyl)methyl]morpholine-4-carbonyl}phenyl)imidazolidin-2-one
4-(2,4-dioxoimidazolidin-1-yl)-N-(1,2,3,4-tetrahydronaphthalen-2-yl)benzamide
3-[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]-N-(4-methoxy-2-methylphenyl)propanamide
3-[({1-[4-(1H-imidazol-1-yl)benzoyl]piperidin-3-yl}oxy)methyl]pyridine
2-[7-(hydroxymethyl)-3,9-diazaspiro[5.5]undecan-3-yl]-N-(2-phenylethyl)acetamide
N3-tert-butyl-1-cyclohexyl-4-oxo-N5-[2-(propan-2-yloxy)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
2-[1-cyclopropyl-2,5-dioxo-3-(4-phenylphenyl)pyrrolidin-3-yl]-N-methyl-N-[(5-propyl-1H-pyrazol-3-yl)methyl]acetamide
(2R,3R,6R)-5-(1H-imidazol-2-ylmethyl)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-(3-methylbut-2-en-1-yl)-8-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-2,8-diazaspiro[4.5]decan-3-one
1'-[2-(methylsulfanyl)pyrimidine-5-carbonyl]-5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-ethoxy-6-{[4-(5-propylpyrimidin-2-yl)piperazin-1-yl]methyl}phenol
2-(2,6-dimethoxy-4-methylphenyl)-2-[4-(pyrazin-2-yl)piperazin-1-yl]acetic acid
(3aR,6aS)-5-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
8-[1-(4-chlorophenyl)cyclobutanecarbonyl]-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
8-fluoro-N-(2-methoxyethyl)-N-(thiophen-3-ylmethyl)quinoline-2-carboxamide
N-{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-N-methylcyclohexanamine
{1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}({[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl})amine
N-[(2R,4S,6S)-2-(4-chlorophenyl)-6-(4-acetamidophenyl)oxan-4-yl]acetamide
7-[3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)propanoyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
8-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-1,3-dioxa-8-azaspiro[4.5]decan-2-one
N-[(1R,2R)-2-(benzyloxy)cyclohexyl]-1-(pyrimidin-2-yl)piperidin-4-amine
1-phenyl-4-[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)propanoyl]piperazin-2-one
4-{4-[3-(4-fluorophenoxy)propyl]piperazine-1-carbonyl}pyrrolidin-2-one
3-{1-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]piperidin-4-yl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[4-({3-[2-(1,3-thiazol-2-yl)pyrrolidine-1-carbonyl]-1,2-oxazol-5-yl}methoxy)phenyl]-1H-1,2,4-triazole
4,6-dimethyl-3-[2-(4-methyl-1,2,5-oxadiazol-3-yl)pyrrolidine-1-carbonyl]-1,2-dihydropyridin-2-one
4-methyl-N-[1-(pyrimidin-2-yl)piperidin-3-yl]-1,2,3-thiadiazole-5-carboxamide
N-[(6-methoxy-1H-1,3-benzodiazol-2-yl)methyl]-6-(morpholin-4-yl)pyrimidin-4-amine
5-oxo-1-phenyl-N-[1-(pyridin-2-ylmethyl)piperidin-3-yl]-2,5-dihydro-1H-pyrazole-3-carboxamide
1-(2-{1-[2-(methylamino)acetyl]piperidin-2-yl}ethyl)pyrrolidin-2-one
2-(4-chloro-1H-pyrazol-1-yl)-1-(3-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)ethan-1-one
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-6-(4-fluorophenyl)-N-methylimidazo[2,1-b][1,3]thiazole-3-carboxamide
5-methoxy-9-{2-methylpyrido[2,3-d]pyrimidin-4-yl}-1-oxa-9-azaspiro[5.5]undecane
6-[(2E)-3-(2,5-difluorophenyl)prop-2-enoyl]-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
N,N-dimethyl-5-{[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}furan-2-carboxamide
ethyl 3-[(3-methoxyphenyl)methyl]-1-methylpiperidine-3-carboxylate
2-methyl-6-{2-[4-(pentan-2-yl)-1H-1,2,3-triazol-1-yl]ethyl}pyrimidin-4-ol
3-hydroxy-3-({[1-(hydroxymethyl)cyclopentyl]amino}methyl)-1-(3-phenylpropyl)piperidin-2-one