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2-{[6-(5-fluoro-2-methoxyphenyl)pyridazin-3-yl](methyl)amino}ethan-1-ol
2-{4-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]piperazin-1-yl}pyrimidin-4-amine
N-benzyl-N,1-dimethyl-5-(4-propylpiperazin-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-({1-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]pyrrolidin-3-yl}methyl)benzoic acid
N-(3,4-difluorophenyl)-4-(1-methyl-1H-imidazol-2-yl)piperidine-1-carboxamide
methyl 3-benzamido-5-(cycloheptylamino)-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-[({2-[(dimethylamino)methyl]phenyl}methyl)(methyl)amino]-2-(4-methoxy-3,5-dimethylphenyl)acetic acid
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-N-methyl-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
4-(2-oxopyrrolidin-1-yl)-N-[1-(2-phenylethyl)piperidin-3-yl]butanamide
2-[2-(methylsulfanyl)phenyl]-2-(thiomorpholin-4-yl)acetic acid
4-[(2-ethyl-1H-imidazol-1-yl)methyl]-2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazole
2-({4-[(2-ethoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)quinolin-4-ol
methyl 6-[(4-methoxy-3-methylphenyl)methyl]-2-(piperidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-(3-{octahydropyrrolo[1,2-a]piperazin-2-ylmethyl}phenyl)-1H-pyrazole
(3E)-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}pent-3-enamide
3-[1-(3-methylthiophene-2-carbonyl)piperidin-4-yl]-N-{[3-(trifluoromethyl)phenyl]methyl}propanamide
1-[2-(pyridin-2-yl)-4-[(pyridin-3-ylmethyl)amino]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
N-[(2-methoxyphenyl)methyl]-5-methyl-4-[(oxolan-2-ylmethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
(4aS,8aR)-1-(2-aminoethyl)-6-(3-chlorothiophene-2-carbonyl)-decahydro-1,6-naphthyridin-2-one
3-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]-N-[(2S)-2-hydroxy-2-phenylethyl]propanamide
2-{1-cyclopentyl-4-[(2-fluoro-5-methoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
N-[1-(1-cyclohexanecarbonylpiperidin-4-yl)-2-(2-methylphenyl)ethyl]-N-methylcyclobutanecarboxamide
1,4,6-trimethyl-N-{[2-(4-methyl-1,4-diazepan-1-yl)pyridin-3-yl]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
2-[(4-chlorophenyl)methyl]-N-[2-(1H-imidazol-4-yl)ethyl]benzamide
N-[(2-ethoxyphenyl)methyl]-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
3-[({1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}amino)methyl]-1-[(2,3-difluorophenyl)methyl]-3-hydroxypiperidin-2-one
N-[1-(6-methylpyridazin-3-yl)piperidin-4-yl]methanesulfonamide
4-chloro-2-({4-[2-(hydroxymethyl)pyridin-4-yl]piperazin-1-yl}methyl)phenol
N-{[5-(5-acetylthiophen-2-yl)-7-chloro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(2-methoxyphenoxy)acetamide
1-methyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-(2-methoxyphenyl)-N-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)-1H-pyrazole-4-carboxamide
2-methyl-N-(4-{[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]carbamoyl}phenyl)furan-3-carboxamide
3-chloro-N-(3-chloro-4-propanamidophenyl)-4-methylbenzamide
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-7-(3-methoxypropanamido)-N,1-dimethyl-2-phenyl-1H-1,3-benzodiazole-5-carboxamide
N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
4-(3-{1-[(1-ethyl-1H-imidazol-2-yl)methyl]-1H-pyrazol-3-yl}phenyl)-3-methylpyridine
N-(3-methoxyphenyl)-3-[1-(1,3-thiazole-4-carbonyl)piperidin-4-yl]propanamide
8-(2-phenoxybenzoyl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
N-[(3S,5S)-5-(ethylcarbamoyl)-1-[2-(morpholin-4-yl)ethyl]pyrrolidin-3-yl]-4-methyl-1H-imidazole-2-carboxamide
3-chloro-4-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}-N-methyl-N-[2-(1H-pyrazol-4-yl)ethyl]benzamide
(2S,4R)-1-(2,3-dihydro-1H-inden-2-yl)-N-methyl-4-({[4-(methylsulfanyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
4-(3-fluorophenoxy)-1-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}piperidine
N-[3-(4-methylpiperazin-1-yl)propyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
2-(5-{[3-(2-chlorophenyl)pyrrolidin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)pyrazine
(3S,4R)-3-benzyl-4-methyl-1-(9H-purin-6-yl)piperidin-4-ol
8-(1H-imidazol-2-ylmethyl)-3-{2-[methyl(2-methylpropyl)amino]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-({4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyridine
3-(1-ethyl-1H-imidazol-2-yl)-1-(5-phenyl-1,2-oxazole-4-carbonyl)piperidine
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-2-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-yl}acetamide
3-(2-methyl-1,4-oxazepane-4-carbonyl)naphthalen-2-ol