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N-[(2,4-dimethoxyphenyl)methyl]-3-[1-(pyrrolidine-1-carbonyl)piperidin-3-yl]propanamide
{[2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)(1,2-oxazol-5-ylmethyl)amine
6-[4-(1-ethoxyethyl)phenyl]-3H-imidazo[4,5-b]pyridine
2-(1-{5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carbonyl}piperidin-2-yl)pyridine
1-(1,3-benzothiazol-2-yl)-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)piperidin-4-amine
(3S,4R)-1-(4-carboxybutanoyl)-4-(4-fluorophenyl)pyrrolidine-3-carboxylic acid
1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-N-methyl-N-(2-methylpropyl)piperidine-4-carboxamide
3-{[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1-(propan-2-yl)pyrrolidine
3-chloro-N-ethyl-4-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-propylbenzamide
methyl 3-(cyclobutylmethoxy)-5-[(1S,4S)-2,5-diazabicyclo[2.2.1]heptane-2-carbonyl]benzoate
6-oxo-N-[3-(pyridin-4-yl)propyl]-1,6-dihydropyridine-2-carboxamide
(2S,4R)-4-amino-N-ethyl-1-[3-(2-methyl-1H-imidazol-1-yl)propanoyl]pyrrolidine-2-carboxamide
4-{4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}morpholine
3,3-dimethyl-1-[(3S,4R)-1-[2-(2-methyl-1H-indol-3-yl)acetyl]-4-(propan-2-yl)pyrrolidin-3-yl]urea
3-[5-(5-methyl-1,2-oxazol-3-yl)-1,3,4-oxadiazol-2-yl]-N-(2-phenylpropyl)propanamide
4-fluoro-N-{[1-(pyridin-4-ylmethyl)piperidin-3-yl]methyl}benzamide
1-[5-chloro-2-(1H-1,2,4-triazol-1-yl)phenyl]-3-(1-methoxypropan-2-yl)urea
7-ethyl-3-[2-(1H-pyrazol-1-yl)ethyl]-2,4,5,7-tetraazatricyclo[6.4.0.02,6]dodeca-1(12),3,5,8,10-pentaene
1-(cyclopropylmethyl)-5-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]-N-methyl-N-(1,3-thiazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-(5-fluoro-2-methoxyphenyl)-5-[(2-methoxyethyl)sulfamoyl]benzoic acid
4-methyl-N-{[3-(oxolan-3-yloxy)phenyl]methyl}-N-(pyridin-4-ylmethyl)benzamide
2-amino-N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
3-(2,3-dimethoxy-5-methylphenyl)-5-(morpholine-4-sulfonyl)benzoic acid
5-[(1S,6R)-4-oxo-3,9-diazabicyclo[4.2.1]nonane-9-carbonyl]-2,3-dihydro-1H-1,3-benzodiazol-2-one
2-(3-chlorophenyl)-N-(4-{4-[4-(pyridin-4-yl)piperidin-1-yl]piperidin-1-yl}phenyl)acetamide
N-[(5-ethylpyridin-2-yl)methyl]-N,1,3-trimethyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-{[1-(methoxymethyl)cyclopropyl]methyl}-5-(1-methyl-1H-imidazol-2-yl)-4-phenyl-1H-imidazole
N-[(2-chlorophenyl)methyl]-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]-N-(prop-2-yn-1-yl)acetamide
{2-[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]-1,3-thiazol-4-yl}methanol
N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-[3-(phenylamino)piperidin-1-yl]but-3-en-1-one
4-(1-{[2-(2,3-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine-4-carbonyl)morpholine
4-{furo[3,2-c]pyridin-4-yl}-2-(6-methoxynaphthalen-2-yl)morpholine
ethyl 4-[(4-chlorophenyl)methyl]-1-(2,3-dihydro-1-benzofuran-2-carbonyl)piperidine-4-carboxylate
(2S,4S)-4-amino-N-ethyl-1-[1-(4-methoxyphenyl)cyclopentanecarbonyl]pyrrolidine-2-carboxamide
N-({5-[3-(methylsulfanyl)propyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)methanesulfonamide
3-fluoro-N-{[7-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)benzamide
1-{4-[(1R,5R)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]phenyl}pyrrolidin-2-one
N-[(4,6-dimethylpyrimidin-2-yl)methyl]-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
3-(4-benzoylpiperazine-1-carbonyl)-1H-pyrazol-5-amine
2-(dimethyl-1,2-oxazol-4-yl)-1-{3-[(2-methyl-1H-imidazol-1-yl)methyl]piperidin-1-yl}ethan-1-one
5-chloro-3-methyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1H-indole-2-carboxamide
[(3R,4R)-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}-1-[2-(1H-pyrazol-1-yl)benzoyl]pyrrolidin-3-yl]methanol
N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-2-methyl-2-(thiophen-2-ylformamido)propanamide
N-(furan-3-ylmethyl)-4-hydroxy-N,2-dimethylpyrimidine-5-carboxamide
2-(1-ethyl-1H-pyrazol-4-yl)-6-fluoro-N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]quinoline-4-carboxamide
2-{1-[(3,5-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(3-methylpyridin-2-yl)ethyl]acetamide
2-(2-chlorophenyl)-2-hydroxy-1-{5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}ethan-1-one
1-[3-(morpholine-4-carbonyl)-1-(2-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-(pyridin-2-ylsulfanyl)ethan-1-one
3-methyl-7-[2-(1-oxo-1,2-dihydroisoquinolin-2-yl)acetyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one