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(2S)-2-amino-1-(4-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-3-(1H-imidazol-4-yl)propan-1-one
6-(4-fluorophenyl)-7-(prop-2-en-1-yl)-2-(pyrrolidine-1-carbonyl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
2-[2-(4-cyclopentyl-3-oxopiperazin-1-yl)-2-oxoethyl]-5-(pyrrolidin-1-yl)-2,3-dihydropyridazin-3-one
N-methyl-2-[4-(4-methyl-1H-pyrazol-1-yl)phenoxy]acetamide
N-[(8-methoxyquinolin-5-yl)methyl]-N-methyl-5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-carboxamide
(1S,5R)-3-[(2-ethoxyphenyl)methyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-N-methylpyridazine-4-carboxamide
[1-({1-[(4-methylphenyl)methyl]-1H-1,3-benzodiazol-2-yl}methyl)pyrrolidin-3-yl]methanamine
N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-4,5,6,7-tetrahydro-1,3-benzothiazole-2-carboxamide
3-(furan-2-ylmethyl)-1-{2-[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)morpholin-2-yl]ethyl}urea
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-4-(3-methylpyridin-4-yl)-1,4-diazepane
N-{2-[5-(1-ethyl-1H-pyrazol-4-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}-N-methylmethanesulfonamide
2-(4-chlorophenyl)-N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
7-(cyclohex-3-en-1-ylmethyl)-N-[2-(1H-1,2,3-triazol-1-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
4,6-dimethyl-5-{4-[(3-methylphenyl)methyl]piperazine-1-carbonyl}-2H-pyran-2-one
6-(morpholin-4-yl)-N-(quinolin-6-ylmethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
2-[2-methoxy-5-(pyrrolidin-1-ylmethyl)phenoxy]-5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridine
1-{[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-[(2E)-3-phenylprop-2-en-1-yl]piperazine
3-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]-2,3-dihydro-1H-inden-1-one
1-(5-fluoropyrimidin-2-yl)-N,N-dimethylazepan-4-amine
4-(4-chlorophenyl)-1-[1-(2-methoxyethyl)pyrrolidine-3-carbonyl]piperidin-4-ol
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-1-(oxan-4-yl)piperidine-4-carboxamide
2-(5-acetylthiophen-3-yl)-1-[3-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]ethan-1-one
2-[4-(4-methoxyphenoxy)piperidin-1-yl]pyrazine
1-(2,3-dihydro-1H-indene-1-carbonyl)-4-(pyridin-4-ylmethyl)-1,4-diazepane
({2-methoxy-5-[(E)-2-phenylethenyl]phenyl}methyl)(methyl)amine
[(3aS,6aS)-2-{[2-(pyrrolidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}-octahydrocyclopenta[c]pyrrol-3a-yl]methanol
1-[3-(thiomorpholine-4-carbonyl)benzenesulfonyl]piperidine-3-carbonitrile
N-cyclopropyl-2-ethyl-4-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-1,3-thiazole-5-carboxamide
2-(2,4-difluorophenoxy)-1-[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonan-7-yl]ethan-1-one
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(2-methoxyethyl)-2-(2-oxopyrrolidin-1-yl)propanamide
2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)-N-[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]acetamide
N-methyl-2-{4-[2-(5-oxo-2-phenylcyclopent-1-en-1-yl)acetyl]morpholin-3-yl}acetamide
2-(1-phenylpiperazine-2-carbonyl)-1,2-oxazinane
(3S)-1-[5-(3,3-diethylpyrrolidine-1-carbonyl)-1-methyl-1H-1,3-benzodiazol-2-yl]pyrrolidin-3-ol
3-(3-methoxyphenyl)-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-1H-pyrazole-4-carboxamide
[(3R,4R)-1-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
2-(4-fluorophenyl)-1-[7-(2-methylphenyl)-9-(oxolan-3-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
(1R,4S)-2-[2-(4-methanesulfonylphenyl)pyridine-3-carbonyl]-2-azabicyclo[2.2.1]heptane
N-{1-[(5-cyano-1-ethyl-1H-pyrrol-3-yl)methyl]piperidin-4-yl}methanesulfonamide
7-(3,4-dihydronaphthalen-2-yl)-4-[(2E)-2-methylbut-2-en-1-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[2-(4-chlorobenzenesulfonamido)ethyl]-2-(methylamino)pyrimidine-5-carboxamide
1-(4-acetyl-1,4-diazepan-1-yl)-2-[(6-methyl-1H-1,3-benzodiazol-2-yl)methoxy]ethan-1-one
2-[4-(1H-1,3-benzodiazol-2-ylmethyl)-1-(cyclohexylmethyl)piperazin-2-yl]ethan-1-ol
N-[1-(cyclohexylmethyl)piperidin-3-yl]-6-(2-hydroxyethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
3-(6-methoxy-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)-1-methyl-1-[3-(1-methyl-1H-pyrazol-4-yl)propyl]urea
N-[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
(1S)-1-[1-(3-methylphenyl)-3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]ethan-1-ol
1-[2-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-3-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-3-methylurea
1-{3-[(4aS,7aR)-4-methyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-3-oxopropyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione