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(1S,5R)-6-(cyclopropylmethyl)-N-(4-ethoxyphenyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
2-{8-methylimidazo[1,2-a]pyridin-3-yl}-N-[2-(4-sulfamoylphenyl)ethyl]acetamide
4-(cyclopropylmethyl)-1-(3,5-dimethyl-1H-indole-2-carbonyl)-3-(propan-2-yl)-1,4-diazepan-5-one
1-[3-(furan-2-yl)propyl]-4-phenylpiperidin-4-ol
N-[4-({7-[1-(2-fluorophenyl)-4-hydroxypiperidin-4-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}methyl)phenyl]acetamide
N-(cyclopropylmethyl)-2-(3-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
5-[4-(morpholin-4-yl)piperidine-1-carbonyl]-N-(pentan-3-yl)pyridin-2-amine
({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)(2-methoxyethyl)[(2-methoxyphenyl)methyl]amine
5-(azocane-1-carbonyl)-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidin-2-one
N-[(2R,3R)-2-methoxy-1'-[(4-methoxy-3-methylphenyl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(methylsulfanyl)acetamide
3-{[1-(2-chloro-6-fluoro-3-methylbenzoyl)pyrrolidin-3-yl]methyl}benzamide
1-[(4aR,8aS)-1-propanoyl-decahydro-1,6-naphthyridin-6-yl]-4-phenylbutan-1-one
1-(2H-1,3-benzodioxol-5-ylmethyl)-N-[2-(diethylamino)ethyl]-N-ethyl-6-methyl-4-oxo-2-propyl-1,4-dihydropyridine-3-carboxamide
4-(4-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}piperazin-1-yl)quinazoline
N-[(1-cyclohexylpyrrolidin-3-yl)methyl]-1H-pyrazole-4-carboxamide
5-{[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1,2,4-oxadiazole-3-carboxamide
3-(2-amino-1,3-thiazol-4-yl)-1-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]propan-1-one
2-[4-(methylsulfanyl)phenyl]-1-[3-(pyrrolidin-1-ylmethyl)piperidin-1-yl]ethan-1-one
dimethyl[(4-{1-[(2-methyl-1,3-thiazol-4-yl)methyl]piperidin-2-yl}phenyl)methyl]amine
(1S,6R)-3-methyl-9-(2-propyl-1,3-thiazole-4-carbonyl)-3,9-diazabicyclo[4.2.1]nonan-4-one
N-[(2-chlorophenyl)methyl]-4-[4-(2-methoxyacetamido)-1H-pyrazol-1-yl]benzamide
1-(2,1,3-benzoxadiazol-4-ylmethyl)-N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methylpiperidin-3-amine
4-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}-2-(2-phenylethyl)morpholine
8-(oxolan-3-ylmethyl)-3-{2-[4-(propan-2-yl)piperazin-1-yl]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-{[8-(2-methoxyethyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]methyl}benzonitrile
N-{2-[7-(naphthalen-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}cyclobutanecarboxamide
N5-methyl-N5-(oxan-4-yl)-N6-(thiophen-2-ylmethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
2-{4-[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]piperidin-1-yl}pyridine-3-carbonitrile
4-[4-(7-{[4-(2-hydroxyethyl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)phenyl]-2-methylbut-3-yn-2-ol
7-cyclobutanecarbonyl-N-[2-(1,3-thiazol-2-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-[(4aR,7aS)-4-(5-fluoropentyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
1-[(3R,5S)-3-[(dimethylamino)methyl]-5-(hydroxymethyl)piperidin-1-yl]-3-(2-ethyl-1H-imidazol-1-yl)propan-1-one
4-[(2-hydroxyphenyl)methyl]-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
5-ethyl-N-[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]pyrimidin-2-amine
[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl][(1-cyclopentylpiperidin-4-yl)methyl](oxolan-2-ylmethyl)amine
(3S,4R)-4-methyl-3-(2-methylpropyl)-1-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidin-4-ol
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)cyclopentanecarboxamide
4-(4-methanesulfonylpiperazine-1-carbonyl)-1-(pyridin-3-ylmethyl)pyrrolidin-2-one
6-[(3-methoxyphenyl)methoxy]-1-(2-methylpropyl)-4-[3-(1H-pyrazol-1-yl)propanoyl]-1,4-diazepan-2-one
1-[4-({[(1-ethylpyrrolidin-2-yl)methyl]({[1-(2-methoxyethyl)piperidin-4-yl]methyl})amino}methyl)thiophen-2-yl]ethan-1-one
(3R,4R)-1-[(7-chloro-3-methyl-1H-indol-2-yl)methyl]-4-cyclobutyl-3-methylpiperidin-4-ol
5-{[(6-methylpyridin-3-yl)oxy]methyl}-N-[5-(morpholin-4-yl)pentyl]-1,2-oxazole-3-carboxamide
7-methoxy-3-[(4-propyl-1,4-diazepan-1-yl)methyl]-1,2-dihydroquinolin-2-one
3-(2-fluorophenyl)-N-[2-(2-oxopyrrolidin-1-yl)ethyl]benzamide
3-[(3-cyanopiperidin-1-yl)methyl]-N-(4-acetamidophenyl)benzamide
N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-4-methyl-1,2,5-oxadiazole-3-carboxamide
(benzylsulfamoyl)[2-(2,3-dihydro-1H-indol-1-yl)ethyl]amine
1-(6-ethyl-2-methylpyrimidin-4-yl)-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}piperidin-4-amine
methyl 4-(4-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}piperazin-1-yl)benzoate
N-(1-benzylpyrrolidin-3-yl)-3-[1-(2-hydroxyacetyl)piperidin-4-yl]propanamide