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1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-4-(4H-1,2,4-triazol-4-yl)piperidine
1-(2-{[2-(dimethylamino)-2-(3-methylthiophen-2-yl)ethyl]amino}-4-methylpyrimidin-5-yl)ethan-1-one
(3R,4R)-1-(5-chloropyridine-2-carbonyl)-4-ethylpiperidine-3,4-diol
9-(but-3-yn-1-yloxy)-4-(2-fluorobenzoyl)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
5-hydroxy-1,2-dimethyl-N-[3-(methylsulfanyl)propyl]-1H-indole-3-carboxamide
2-{[(1-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}piperidin-3-yl)oxy]methyl}pyridine
(1-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-3-yl)methanamine
7-(oxan-4-yl)-2-(pyridine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
2-[(1R,5S)-6-azabicyclo[3.2.1]octan-6-ylmethyl]-N,N-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-sulfonamide
3-[1-(3,6-dimethyl-1-benzofuran-2-carbonyl)piperidin-4-yl]-N-[(4-fluorophenyl)methyl]propanamide
N-{1-[(3-chlorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-2-methoxypyridine-4-carboxamide
2-[4-(trimethyl-1H-pyrazole-4-carbonyl)piperazin-1-yl]-1,3-benzothiazole
4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1-propanoyl-1,4-diazepan-5-one
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]-3-(pyridin-3-yl)propan-1-one
4-[1-cyclohexyl-5-(1H-pyrrol-2-yl)-1H-1,2,4-triazol-3-yl]pyridine
5-[4-(1-benzyl-1H-imidazol-2-yl)piperidine-1-carbonyl]pyridine-2-carbonitrile
1-propyl-N-[3-(pyridin-4-yl)propyl]-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(3S,4R)-N,N-dimethyl-4-(4-methylphenyl)-1-[4-(4H-1,2,4-triazol-4-yl)benzoyl]pyrrolidin-3-amine
3-{2-[2,2-bis(prop-2-en-1-yl)pyrrolidin-1-yl]-2-oxoethyl}-4-[(2-fluoro-4-methoxyphenyl)methyl]piperazin-2-one
6-(1-cyclobutanecarbonylpiperidine-4-carbonyl)-1-methyl-1H,4H,5H,6H,7H-pyrrolo[2,3-c]pyridine-2-carboxamide
3-[(3S,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2,4-dichlorophenyl)urea
(2S,4S)-1-{[4-(diethylamino)phenyl]methyl}-N-(2-methoxyethyl)-4-{[(4-phenylphenyl)methyl]amino}pyrrolidine-2-carboxamide
N-(furan-2-ylmethyl)-1-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}acetyl)piperidine-4-carboxamide
5-{[4-(thiophen-2-ylmethyl)-1,4-diazepan-1-yl]methyl}-2,1,3-benzothiadiazole
3-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-1-(4-methyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)urea
N-(3-methylphenyl)-3-[1-(oxolane-3-carbonyl)piperidin-4-yl]propanamide
ethyl 4-[2-(ethylamino)pyrimidine-5-amido]piperidine-1-carboxylate
N-[2-(pyridin-2-yl)ethyl]-2-[(quinolin-6-yloxy)methyl]-1,3-oxazole-4-carboxamide
7-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-{imidazo[1,2-a]pyridin-2-ylmethyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
(2,1,3-benzoxadiazol-5-ylmethyl)(methyl){[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}amine
4-methyl-N-[2-(7-{[2-(trifluoromethyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]benzamide
2,6-dimethyl-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]pyrimidine-4-carboxamide
2-{2-methoxy-4-[(2-methyl-1,4-oxazepan-4-yl)methyl]phenoxy}acetamide
(2S)-2-amino-1-[4-(4-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]-3-(1H-imidazol-4-yl)propan-1-one
3-[(5-{8-chloro-[1,2,4]triazolo[4,3-a]pyridin-3-yl}furan-2-yl)sulfanyl]-4H-1,2,4-triazole
(1H-imidazol-2-ylmethyl)(methyl)[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]amine
N-[2-(dimethylamino)ethyl]-N,1-dimethyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-{2-[(1S,3R)-1-ethoxy-3-hydroxy-7-azaspiro[3.5]nonan-7-yl]-2-oxoethyl}-1,2-dihydropyrimidin-2-one
N-cyclopropyl-1-[1-(1-methyl-1H-pyrrole-2-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
2-(3-methoxyphenyl)-5-(oxolane-3-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
6-fluoro-3-{imidazo[1,2-a]pyridin-2-ylmethyl}-3,4-dihydroquinazolin-4-one
5-[(4-benzylpiperidin-1-yl)methyl]-N-[1-(pyridin-3-yl)propan-2-yl]-1,2-oxazole-3-carboxamide
4-(5-propylthiophene-3-carbonyl)-1,4-oxazepan-6-ol
(1S,5R)-6-(3-methylbut-2-en-1-yl)-3-[1-(pyridine-3-carbonyl)piperidin-4-yl]-3,6-diazabicyclo[3.2.2]nonane
1-[2-(2,3-dihydro-1,4-benzodioxin-6-yl)pyrimidin-4-yl]pyrrolidin-3-ol
N-(2-methoxyethyl)-3-{[1-(quinolin-4-ylmethyl)piperidin-4-yl]oxy}benzamide
5-(methoxymethyl)-N-(2-methylpropyl)-N-(3-phenylprop-2-yn-1-yl)furan-2-carboxamide
N-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-3-sulfamoylthiophene-2-carboxamide
4-[2-(2-ethoxypyridin-3-yl)pyridine-4-carbonyl]morpholine