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1-(3-{4-azaspiro[2.5]octan-4-ylmethyl}phenoxy)-3-(4-ethylpiperazin-1-yl)propan-2-ol
(2S,4R)-4-amino-1-[(5-butylthiophen-2-yl)methyl]-N-methylpyrrolidine-2-carboxamide
(3aR,7aS)-N-[4-chloro-3-(methylcarbamoyl)phenyl]-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carboxamide
[(1-ethyl-1H-pyrazol-4-yl)methyl]({[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl})amine
4-{4-amino-6-[(4-methylphenyl)amino]-1,3,5-triazin-2-yl}-N,N-dimethylbenzamide
(3S,4R)-1-[3-(cyclopentylcarbamoyl)propanoyl]-4-phenylpyrrolidine-3-carboxylic acid
7-[1-(2-ethoxyethyl)-3-methyl-1H-pyrazole-5-carbonyl]-2,7-diazaspiro[4.4]nonane-1,3-dione
N,3,5,7-tetramethyl-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}-1H-indole-2-carboxamide
5-{[5-(cyclohexylsulfanyl)furan-2-yl]methyl}-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
2-(2H-1,3-benzodioxol-5-yl)-1-[2-(4-fluorobenzenesulfonyl)ethyl]-1H-imidazole
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-N,2,3,6-tetramethylquinoline-4-carboxamide
4-[(4-fluorophenyl)methyl]-7-(2-methylphenyl)-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-[3-(piperidin-1-ylmethyl)piperidine-1-carbonyl]-1H,2H,5H,6H,7H-cyclopenta[b]pyridin-2-one
1-cyclohexyl-3-(cyclopropylmethyl)-2-oxo-N-(pyrimidin-4-ylmethyl)-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-[(3S)-2-oxoazepan-3-yl]-2,3-dihydro-1H-indene-2-carboxamide
4-phenyl-2-(4H-1,2,4-triazol-4-yl)phenol
(1S,5R)-3-[(5-fluoro-2-methoxyphenyl)methyl]-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonane
1-[4-(cyclopropylmethyl)piperazin-1-yl]-2-(2,4,7-trimethyl-1H-indol-3-yl)ethan-1-one
3-[1-benzyl-3-(morpholine-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1H-indole
2-[4-(2-propyl-1,3-thiazole-4-carbonyl)piperazin-1-yl]-1,3-benzothiazole
2-[4-(1-methyl-1H-pyrrole-2-carbonyl)piperazin-1-yl]-1,3-benzothiazole
(3R,4R)-4-amino-1-[4-(benzyloxy)butyl]piperidin-3-ol
5-acetamido-1-ethyl-2-(2-fluorophenyl)-N-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-1H-1,3-benzodiazole-7-carboxamide
1-(3-methoxybenzoyl)-4-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperazine
1-[2-(dimethylamino)-4-[(1H-imidazol-2-ylmethyl)(methyl)amino]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
1-[2-(3-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]azepane
1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-N-(oxan-4-yl)piperidine-4-carboxamide
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-amine
5-(7-hydroxy-6-methoxy-2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)thiophene-2-carboxylic acid
N-cyclopropyl-2-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-1H-1,3-benzodiazole-4-carboxamide
(2R,6R)-4-(1-acetylpiperidine-4-carbonyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
1-methyl-4-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperazine-2-carboxylic acid
3,3-dimethyl-1-[(3S,4R)-4-(propan-2-yl)-1-[2-(thiophen-3-yl)acetyl]pyrrolidin-3-yl]urea
1-(2-methoxypyrimidine-5-carbonyl)spiro[azepane-4,2'-chromene]
methyl 3-{[(3-ethyl-1-methyl-1H-pyrazol-5-yl)formamido]methyl}-5-(4-fluorobenzenesulfonamido)benzoate
6-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-2-[(4-methoxyphenyl)methyl]-1,3-benzoxazole
2-{1-[(3-methoxyphenyl)methyl]-4-{[4-(1H-pyrazol-1-yl)phenyl]methyl}piperazin-2-yl}ethan-1-ol
N-[1-methyl-3-(1-methyl-1,2,5,6-tetrahydropyridin-3-yl)-1H-pyrazol-5-yl]-2-phenylbutanamide
3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(pyrrolidine-1-carbonyl)piperidine
6-({3-[2-(4-fluorophenyl)pyrrolidine-1-carbonyl]-1,2-oxazol-5-yl}methoxy)quinoline
2-{4-[2-(furan-2-yl)azepane-1-carbonyl]piperidin-1-yl}acetamide
3-[(4-fluorophenyl)methyl]-5-{1-[1-(4-hydroxy-3-methoxyphenyl)propan-2-yl]piperidin-4-yl}-5-methylimidazolidine-2,4-dione
2-(4-chlorophenyl)-N-[2-(diethylamino)ethyl]-N-methyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
4-(furan-3-ylmethyl)-3-[2-(1,2-oxazinan-2-yl)-2-oxoethyl]piperazin-2-one
2-amino-4-(3-chloro-4-hydroxyphenyl)-6-(4-hydroxy-3-methoxyphenyl)pyridine-3-carbonitrile
{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]amine
2-(1H-1,3-benzodiazol-1-ylmethyl)-N-(1-phenylpiperidin-4-yl)-1,3-oxazole-4-carboxamide
N-{[2-(dimethylamino)-8-methylquinolin-3-yl]methyl}-N-[2-(dimethylamino)ethyl]-2-ethylbutanamide
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-5-methyl-1-(pyridin-2-yl)-1H-pyrazole-4-carboxamide
3-[3-cyclopentyl-5-(1H-1,2,3,4-tetrazol-1-ylmethyl)-1H-1,2,4-triazol-1-yl]-1λ6-thiolane-1,1-dione