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methyl[(3-methyl-1H-pyrazol-5-yl)methyl]({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)amine
{4-[4-(3-phenylpropyl)piperazin-1-yl]pyridin-2-yl}methanol
2-{2-methyl-6-[3-(2-methylpropyl)pyrrolidin-1-yl]pyrimidin-4-yl}ethan-1-amine
N-butyl-1-(7-methanesulfonyl-4-methylquinazolin-2-yl)piperidine-4-carboxamide
N-cyclopentyl-N'-[(2-fluorophenyl)methyl]-N'-(1-methoxypropan-2-yl)butanediamide
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)acetamide
N-[1-(cyclohexylmethyl)-5-oxopyrrolidin-3-yl]-4-methyl-2-oxopentanamide
N-(1H-indol-4-ylmethyl)-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
1-[(1S,5R)-6-(2-methyl-1H-1,3-benzodiazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
2-{methyl[1-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)piperidin-4-yl]amino}ethan-1-ol
2-[2-(2-methoxyethyl)-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl]-6-(propan-2-yl)pyridine-3-carbonitrile
4-phenyl-N-[1-(1-propanoylpiperidin-4-yl)-1H-pyrazol-5-yl]butanamide
N-[(1-{[2-(furan-2-yl)phenyl]methyl}piperidin-3-yl)methyl]-1-phenylmethanesulfonamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-(pyridin-3-yl)piperazine
3-(1H-indol-3-yl)-1-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]propan-1-one
5-[2-(1-butyl-1H-1,2,4-triazol-5-yl)ethyl]-3-(2-fluorophenyl)-1,2,4-oxadiazole
2-({[(dimethyl-1,2-oxazol-4-yl)methyl](methyl)amino}methyl)-6-methoxyphenol
4-(4-methoxyphenyl)-4-oxo-N-{1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}butanamide
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-[(6-methylpyridin-2-yl)methyl]piperidine-3-carboxamide
N-({1-[3-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]piperidin-3-yl}methyl)naphthalene-1-carboxamide
(1S,5R)-3-[2-(1H-1,3-benzodiazol-2-yl)acetyl]-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}pyridazine
N-(pyridin-3-ylmethyl)-N-(thiophen-3-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-3-(5-{[3-(trifluoromethyl)phenyl]methyl}-1,3,4-oxadiazol-2-yl)propanamide
2-[({2-[2-hydroxy-3-(morpholin-4-yl)propoxy]-3-methoxyphenyl}methyl)(methyl)amino]-N-methylacetamide
4-[2-(2-ethyl-1H-1,3-benzodiazol-1-yl)butanoyl]-1λ6-thiomorpholine-1,1-dione
6-fluoro-N-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
6-(2,5-dimethylfuran-3-yl)-7-methyl-8-oxo-N-(oxolan-3-ylmethyl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
1-methyl-4-(2-methyl-5-propylpyrimidin-4-yl)piperazine-2-carboxylic acid
N,N,8-trimethyl-2-[1-(3-methylpyridin-4-yl)-1H-pyrazol-4-yl]quinoline-4-carboxamide
1-{[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-1,4-diazepan-5-one
4-(1H-imidazol-2-yl)-1-{[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidine
2-(pyridin-3-yl)-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}acetamide
2-(7-fluoro-2-methyl-1H-indol-3-yl)-1-[4-(1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
1-{4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-(1H-1,2,4-triazol-1-yl)propan-1-one
1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-5-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-1H-pyrazole-4-carboxamide
N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-5-methylpyrazolo[1,5-a]pyrimidin-7-amine
1-(2,3-dimethylphenyl)-4-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperazine
1-{4-[(cyclopentylamino)methyl]-2-methoxyphenoxy}-3-(pyrrolidin-1-yl)propan-2-ol
(2S)-2-[3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]pyrrolidine-1-carboxamide
N-(1-benzylpiperidin-4-yl)-2-ethyl-6-methyl-1-[(5-methylfuran-2-yl)methyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
{2-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]-1,3-thiazol-4-yl}methanol
2-{[(dimethyl-1,2-oxazol-4-yl)methyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
2-{1-[(4-methoxy-3-methylphenyl)methyl]-4-[(5-methylfuran-2-yl)methyl]piperazin-2-yl}ethan-1-ol
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N-ethyl-5-phenyl-1,2-oxazole-3-carboxamide
2-{[(2-chlorophenyl)methyl]sulfanyl}-1-[(3S,4S)-3-hydroxy-4-(morpholin-4-yl)pyrrolidin-1-yl]ethan-1-one
[(2-ethylpyrimidin-4-yl)methyl](methyl)[2-(pyridin-4-yl)ethyl]amine
N-cyclopropyl-2-[(1R,2R,6S,7S)-10-oxa-4-azatricyclo[5.2.1.02,6]decan-4-yl]pyridine-4-carboxamide
5-(methanesulfonylmethyl)-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)pyridin-2-amine
3-(5-methylfuran-2-yl)-N-[2-(4,5,6,7-tetrahydro-1-benzothiophen-3-yl)ethyl]-1H-pyrazole-5-carboxamide