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N-ethyl-N-methyl-3-oxo-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecane-9-sulfonamide
3-(4-chlorobenzoyl)-9-methoxy-N-[(3-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-(3-{imidazo[1,2-a]pyridin-2-yl}propanoyl)-3-propylpiperidine-3-carboxylic acid
3-(5-{2-[5-(butan-2-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}-1,2,4-oxadiazol-3-yl)pyridine
4-(oxolan-2-ylmethyl)-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N-[(3R,4S)-4-cyclopropyl-1-(3-methoxypropyl)pyrrolidin-3-yl]-3-fluoro-4-methoxybenzamide
3-(1H-imidazol-2-ylmethyl)-7-methyl-3H,4H-thieno[3,2-d]pyrimidin-4-one
3,5-difluoro-2-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]pyridine
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-3-methyl-4-oxo-3,4-dihydroquinazoline-7-carboxamide
2-[3-(3-ethylphenoxy)azetidine-1-carbonyl]-5-methylpyrazine
1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-4-(2-methoxyethoxy)piperidine
N-methyl-3-(2-oxoazepan-1-yl)-N-[1-(pyridin-3-yl)ethyl]propanamide
3-{4-[(1S,5R)-6-methyl-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]-4-oxobutyl}-3,4-dihydroquinazolin-4-one
4-[2-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]phenol
N-[(2,4-dichlorophenyl)methyl]-N,4,6-trimethyl-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
1-{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(furan-2-carbonyl)piperazine
N-cyclopropyl-7-{pyrazolo[1,5-a]pyrimidine-2-carbonyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methylnaphthalene-2-carboxamide
2-{1'-[(5-methylthiophen-2-yl)methyl]-2-oxo-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-1-yl}acetamide
2-{2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxybenzoyl}-1,2-oxazinane
(3S,4R)-4-(hydroxymethyl)-1-(1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)piperidin-3-ol
N-[(3-fluorophenyl)methyl]-2-(2-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-4-(thiophen-2-yl)phenoxy)acetamide
1-(2-aminoethyl)-N-{[(2R,3R,5S)-2-(2-fluorophenyl)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]methyl}-1H-1,2,3-triazole-4-carboxamide
3-[2-oxo-2-(4-phenylpiperazin-1-yl)ethyl]-4-(pyridin-2-ylmethyl)piperazin-2-one
3-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-4-methoxyphenyl]pyridin-4-amine
1-(4-{imidazo[1,2-b]pyridazin-6-yl}piperazin-1-yl)-3-(3-methoxyphenyl)propan-1-one
N-{5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}-1-cyclopropanecarbonylpiperidine-4-carboxamide
methyl 3-{[(2-chlorophenyl)methyl](propan-2-yl)carbamoyl}propanoate
1-[(4-chlorophenyl)methyl]-6-oxo-N-(2,2,2-trifluoroethyl)piperidine-3-carboxamide
N-{[5,8-dimethoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-2-(3-methyl-1H-pyrazol-1-yl)acetamide
3,5-dimethoxy-N-[(5-{[(3-methylphenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)methyl]benzamide
3-({cyclopropyl[(1-methyl-1H-imidazol-2-yl)methyl]amino}methyl)-N-phenylbenzamide
methyl 4-{4-[2-chloro-4-(cyclopentylcarbamoyl)phenoxy]piperidin-1-yl}-4-oxobutanoate
6-{[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
5-(5-chloro-2-methylphenyl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
N-tert-butyl-6-(morpholine-4-sulfonyl)-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
2-methyl-1-{1-[4-(pyrrolidin-1-ylmethyl)benzoyl]azetidin-3-yl}piperidine
4-(2-{4-[(benzyloxy)methyl]-1H-1,2,3-triazol-1-yl}ethyl)morpholine
2-acetyl-8-(4,6-dimethoxypyrimidin-2-yl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
7-(4-chlorophenyl)-2-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-{5-[2-(1H-pyrrol-1-yl)pentanoyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
N-[(2R,3R)-1'-(1-benzothiophen-2-ylmethyl)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]furan-2-carboxamide
8-(4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl)-5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine
1-methyl-4-(4-oxo-4H-chromen-3-yl)-3-(pyridin-3-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
(1-{2-[5-(5-ethylfuran-2-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}piperidin-3-yl)methanol
1-(4-ethylpiperazin-1-yl)-3-{4-[(4-ethylpiperazin-1-yl)methyl]-2-methoxyphenoxy}propan-2-ol
2-[(3-chlorophenyl)methyl]-N-[(5-methyl-4H-1,2,4-triazol-3-yl)methyl]-1,3-benzoxazole-6-carboxamide
8-{dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-2-methyl-2,8-diazaspiro[4.5]decan-3-one
[(3R,4R)-4-[(4-methylpiperazin-1-yl)methyl]-1-[3-(trifluoromethyl)benzoyl]pyrrolidin-3-yl]methanol
N-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]-2-methoxybenzene-1-sulfonamide