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2-[2-(piperidin-1-yl)ethyl]-5-(thiomorpholine-4-carbonyl)-2,3-dihydro-1H-isoindol-1-one
N-(pyridin-2-ylmethyl)-5-[2-(pyrrolidin-1-yl)acetyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
4-(4-ethyl-1,2,3-thiadiazole-5-carbonyl)-1-(2-methoxyphenyl)-5-methylpiperazin-2-one
N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-2-{tricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl}acetamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)acetamide
1-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
methyl (2S,4R)-4-(3-cyano-5-fluorobenzamido)-1-methylpyrrolidine-2-carboxylate
3-{1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-1,2,5,6,7,8-hexahydroquinolin-2-one
(1S,5R)-6-(2-methoxyethyl)-3-(2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-methyl-1'-[2-(methylsulfanyl)pyridine-3-carbonyl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
3-{2-[2-(4-fluorophenyl)piperidin-1-yl]-2-oxoethyl}-1,3-diazinane-2,4-dione
(4aS,8aR)-1-(3-hydroxypropyl)-6-[(2-methyl-1H-imidazol-4-yl)methyl]-decahydro-1,6-naphthyridin-2-one
6-(4-{1-azabicyclo[2.2.2]octan-3-yl}piperazine-1-carbonyl)-2-methyl-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
N-methyl-2-(1-methyl-3-oxopiperazin-2-yl)-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
(3R,4R)-1-{[4-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]methyl}-4-{methyl[2-(pyridin-2-yl)ethyl]amino}piperidin-3-ol
N-(2H-1,3-benzodioxol-5-ylmethyl)-4-(pyridin-3-yl)pyrimidin-2-amine
1-{[3-fluoro-2-(trifluoromethyl)phenyl]methyl}piperidine-2,6-dione
(3aS,6aS)-2-acetyl-5-[(1-ethyl-1H-pyrazol-5-yl)sulfonyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-({methyl[(3-methyloxetan-3-yl)methyl]amino}methyl)-N-(2,4,6-trimethylphenyl)benzamide
3-[5-(2H-1,3-benzodioxol-5-yl)-1,3,4-oxadiazol-2-yl]-N-ethyl-N-(2-methylprop-2-en-1-yl)propanamide
(2S)-2-amino-2-cyclohexyl-1-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]ethan-1-one
5-(2-chloro-4,5-dimethoxyphenyl)-1-ethyl-1H,4H-pyrazolo[3,4-d]imidazole
2-[(2-fluorophenyl)methyl]-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1,3-benzoxazole-6-carboxamide
N-[2-({4-[(2-methylpyridin-3-yl)oxy]piperidin-4-yl}formamido)ethyl]acetamide
5-methyl-N-[3-(4-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}phenoxy)propyl]thiophene-2-carboxamide
(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)[(5-ethylpyridin-2-yl)methyl]methylamine
(3R,4R)-1-(4-cyclobutyl-6-methylpyrimidin-2-yl)-3,4-dimethylpyrrolidin-3-ol
(4aS,7aR)-1-{imidazo[1,2-a]pyridine-3-carbonyl}-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(1R,2S,9R)-11-({1-methyl-4-oxo-1H,4H,5H-pyrazolo[3,4-d]pyrimidin-6-yl}methyl)-7,11-diazatricyclo[7.3.1.02,7]tridecan-6-one
N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-N-[(4-methoxyphenyl)methyl]thiophene-2-carboxamide
4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-7H-pyrrolo[2,3-d]pyrimidine
9-[(1-cyclopropyl-1H-imidazol-2-yl)methyl]-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[1-(3,5-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-1,5-dimethyl-1H-pyrazole-3-carboxamide
(2S)-1-[1-(6-ethoxy-4-methylquinazolin-2-yl)piperidine-4-carbonyl]pyrrolidine-2-carboxamide
methyl (2S,4S,5R)-1,2-dimethyl-5-(2-methylphenyl)-4-{[2-(pyridin-3-yl)ethyl]carbamoyl}pyrrolidine-2-carboxylate
8-(1-aminocyclopropanecarbonyl)-2-[2-(pyridin-2-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
2-(methoxymethyl)-1-{5-[3-(trifluoromethyl)phenoxymethyl]-1,2-oxazole-3-carbonyl}piperidine
(3aR,7aS)-5-methyl-2-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-2,3,3a,4,7,7a-hexahydro-1H-isoindole
2-methyl-N-[1-(thian-4-yl)piperidin-4-yl]-1H-1,3-benzodiazole-5-carboxamide
N-[(3R,4R)-4-(morpholin-4-yl)oxolan-3-yl]-4-sulfamoylbenzamide
3-({[1-(hydroxymethyl)cyclopropyl]methyl}sulfamoyl)-N-methyl-N-[2-(methylsulfanyl)ethyl]benzamide
1-[2-methoxy-4-({methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}methyl)phenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
1-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-3-{[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}urea
5-amino-3-(2-methoxypyrimidin-5-yl)-1,6-diazatricyclo[6.2.2.02,7]dodeca-2,4,6-triene-4-carbonitrile
(5-{[({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)(methyl)amino]methyl}-2-ethoxyphenyl)methanol
4-(1H-1,3-benzodiazol-1-yl)-1-(furan-2-ylmethyl)piperidine-4-carboxylic acid
5-[1-(3-fluorobenzoyl)piperidin-4-yl]-5-(pyridin-3-yl)-3-(thiophen-3-ylmethyl)imidazolidine-2,4-dione
N-(4-{[4-(6-ethoxy-4-methylquinazolin-2-yl)-1,4-diazepan-1-yl]methyl}phenyl)acetamide
1-{2-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-2-oxoethyl}-2-methyl-1,4-dihydroquinolin-4-one
5-(2-chloro-4-fluorophenoxymethyl)-N-[1-(pyridin-4-yl)propyl]-1,2-oxazole-3-carboxamide