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2,6,6-trimethyl-3-[2-(morpholin-4-yl)-2-oxoethyl]-1-(propan-2-yl)-4,5,6,7-tetrahydro-1H-indol-4-one
5-(3-fluoro-2-methoxybenzoyl)-1-(2-hydroxyethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
6-(3-fluoro-4-methoxyphenyl)-N-methyl-N-(1H-pyrazol-5-ylmethyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
(1-{5-[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperidin-4-yl)methanol
2-(2-chlorophenyl)-2-[(2,3-dimethylquinoxalin-6-yl)formamido]acetic acid
5-{1-[2-(3-methoxyphenyl)acetyl]piperidin-4-yl}-3-(oxolan-2-ylmethyl)-5-(pyridin-3-yl)imidazolidine-2,4-dione
(4aR,8aS)-1-[2-(4-methoxyphenyl)ethyl]-6-(4-methylbenzoyl)-decahydro-1,6-naphthyridin-2-one
9-[1-(2-methoxyethyl)-5-oxopyrrolidine-3-carbonyl]-6-(4-methoxyphenyl)-6,9-diazaspiro[4.5]decan-7-one
4-(1-ethyl-1H-imidazol-2-yl)-1-{[2-(trifluoromethyl)phenyl]methyl}piperidine
2-[(2-chloro-4,5-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
(1S,5R)-6-(2-ethylpyrimidine-5-carbonyl)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
1-(2-{2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-2-oxoethyl)-1,2-dihydropyrimidin-2-one
N-(6-methylpyridazin-3-yl)-2-phenyl-5,6,7,8-tetrahydroquinazolin-5-amine
(3S,4R)-1-(2-chloro-4-fluorobenzoyl)-4-methylpiperidine-3,4-diol
2-ethyl-8-[4-(1H-1,2,4-triazol-1-yl)butanoyl]-2,8-diazaspiro[5.5]undecan-3-one
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[7-methyl-2-(3-methylphenyl)quinolin-3-yl]methyl}propanamide
1,3-dimethyl-N-[2-methyl-1-(1-methyl-1H-imidazol-2-yl)propyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
1-[(2R,3R,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]cyclopropane-1-carboxamide
N'-(3-fluorophenyl)-N-[2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]ethanediamide
(1R,5R)-6-[(4-fluoro-3-methoxyphenyl)methyl]-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-[2-(naphthalen-1-ylmethyl)morpholin-4-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
1-(cyclohex-3-en-1-ylmethyl)-4-(pyrrolidin-1-yl)piperidine
1-{[(1-benzothiophen-2-ylmethyl)(methyl)carbamoyl]methyl}piperidine-4-carboxamide
5-{3-[(4-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}-N-[2-(pyrazin-2-yl)ethyl]pyridin-2-amine
4-[(2,5-dimethylthiophen-3-yl)sulfonyl]-3-methyl-1-(2-methylpropyl)piperazin-2-one
3-benzyl-5-[3-(3-methoxyphenyl)-1H-pyrazol-4-yl]-1H-1,2,4-triazole
2-methoxy-N-(3-methyl-1-{7-[(3-methylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)acetamide
1-{[3-(2-methylphenyl)phenyl]methyl}-4-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidine
2-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-2-oxo-S-(thiophen-2-yl)ethane-1-sulfonamido
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-4-(methylsulfanyl)benzamide
(3S,9aR)-8-(4-methylbenzenesulfonyl)-3-(2-methylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-ethyl-4-[2-(3-methoxypropyl)piperidine-1-carbonyl]pyridine
4-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonane-9-carbonyl]-2,6,8-trimethylquinoline
N-cyclopropyl-1-{1-[(4-methoxy-2,5-dimethylphenyl)methyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carboxamide
1-(2-fluorobenzenesulfonyl)-4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine
4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(pyrrolidine-1-carbonyl)piperidine
N-[3-(4-hydroxyphenyl)propyl]-4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzamide
4-{[4-(1-benzofuran-2-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-2-ethylpyrimidine
4-{3-cyclobutyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-6-ethyl-2-(pyrrolidin-1-yl)pyrimidine
4-methyl-5-(3-phenylpiperazine-1-carbonyl)-2-(pyridin-3-yl)pyrimidine
2-methoxy-N-[1-(1-{[4-(propan-2-yloxy)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]benzamide
methyl[(2-methyl-1,3-thiazol-4-yl)methyl][(2-phenyl-1,3-oxazol-4-yl)methyl]amine
2-acetamido-N-{1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}acetamide
3-[(1R,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N-cyclopropylpropanamide
1-[(4-{[1-(3-methylthiophene-2-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl]-4-phenylpiperidine
1-methyl-2-phenyl-4-{[2-(pyrrolidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}piperazine
N-(2-oxo-2-{3-[2-(pyridin-4-yl)pyridin-4-yl]pyrrolidin-1-yl}ethyl)acetamide
4-({2-[1-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
N-[2-(dimethylamino)ethyl]-N-methyl-3-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
5-[(5-phenylthiophen-2-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid