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N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}-2,2-dimethylpropanamide
N-(1-{1-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]piperidin-4-yl}-2-phenylethyl)-N,1-dimethyl-1H-pyrazole-3-carboxamide
(1S,5R)-6-(1-ethyl-1H-pyrazole-3-carbonyl)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane
4-(1-ethyl-1H-imidazol-2-yl)-1-[3-(3-methoxyphenyl)-1H-pyrazole-4-carbonyl]piperidine
N-(2-methoxy-5-methylphenyl)-2-[2-(pyridin-2-yl)-1H-imidazol-1-yl]acetamide
ethyl 5-(2,2-dimethylpropanoyl)-1-[3-(pyridin-3-yl)propyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-({7-[(2,3-difluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-2-methylbutanamide
1-(furan-3-ylmethyl)-N-[4-(1H-pyrazol-5-yl)phenyl]piperidine-3-carboxamide
3-[4-({3-[3-(azepan-1-yl)-2-hydroxypropoxy]phenyl}methyl)piperazin-1-yl]propanamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[(3-ethoxy-4-hydroxyphenyl)methyl]piperidin-3-ol
2-phenoxy-N-{1-[({[4-(1H-pyrazol-1-yl)phenyl]methyl}carbamoyl)methyl]-1H-pyrazol-4-yl}acetamide
2,4,6-trimethyl-5-{[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]methoxy}pyrimidine
1-(2-{[(4-fluorophenyl)methyl]carbamoyl}ethyl)-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-1,3-thiazole-5-carboxamide
1-{3-[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]-3-oxopropyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-({5-[1-(1H-imidazol-2-ylmethyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)morpholine
(5S,9aS,9bS)-5-[4-(furan-2-yl)phenyl]-2-(1-methylpiperidin-4-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-methyl-5-[1-(1-methylpiperidin-4-yl)-3-(oxolan-3-yl)-1H-1,2,4-triazol-5-yl]pyrimidin-2-amine
1-[(2-methylphenyl)methyl]-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
(1-methyl-1H-imidazol-2-yl)[1-({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-4-yl]methanol
1-[(1R,5S,8R)-8-hydroxy-3-azabicyclo[3.2.1]octan-3-yl]-3-(4-hydroxyphenyl)propan-1-one
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-2-(2-oxo-4-phenylpyrrolidin-1-yl)acetamide
4-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonane-9-carbonyl]-2,3,6-trimethylquinoline
6-[(2-chlorophenyl)methyl]-3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
3-(1H-1,3-benzodiazol-1-yl)-1-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]propan-1-one
2-(7-chloro-2,3-dihydro-1,4-benzodioxin-6-yl)-1-{3-[(dimethylamino)methyl]-3-hydroxypyrrolidin-1-yl}ethan-1-one
6-[1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl]pyridine-2-carbonitrile
3-{5-[(2,5-dimethoxyphenyl)methyl]-1,3,4-oxadiazol-2-yl}-N-[(1-ethylpyrrolidin-2-yl)methyl]propanamide
2-(3,4-dichlorophenyl)-4-(1,4-dimethylpiperidine-4-carbonyl)morpholine
(4aS,7aR)-1-(3-phenyl-1H-pyrazole-5-carbonyl)-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-methyl-2-phenyl-1-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
3-{[(2-methoxyethyl)(pyridin-4-ylmethyl)carbamoyl]amino}-N,N,2-trimethylbenzamide
1-[1-(2H-1,3-benzodioxol-5-ylmethyl)-4-phenylpiperidin-4-yl]ethan-1-one
2-methoxy-N-[2-(8-methoxy-2-methylquinolin-5-yl)phenyl]acetamide
1-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-{2-[4-(methylsulfanyl)phenyl]acetyl}-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
N-[(4-fluorophenyl)methyl]-N-(3-methoxypropyl)-2-(2-oxopiperidin-1-yl)acetamide
(4aS,8aR)-6-(2-propoxybenzoyl)-1-propyl-decahydro-1,6-naphthyridin-2-one
(1R,6S)-9-methyl-3-{2-phenylimidazo[1,2-a]pyridine-6-carbonyl}-3,9-diazabicyclo[4.2.1]nonane
4-fluoro-N-{[1-(pent-4-enoyl)piperidin-3-yl]methyl}benzamide
N-{[2-(3-methoxyphenyl)-1,3-thiazol-5-yl]methyl}-1H-1,2,3-triazole-5-carboxamide
(3aS,6aR)-3-cyclopentyl-5-{[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
4-methoxy-N-(2-methoxyethyl)-2-{[1-(thiophen-3-ylmethyl)piperidin-4-yl]oxy}benzamide
4-(oxan-2-ylmethyl)-1-(5-phenyl-1,2,4-oxadiazol-3-yl)piperidine-4-carboxylic acid
3-{[5-(4-fluorophenyl)-1,2,4-triazin-3-yl]amino}-2,2-dimethylpropan-1-ol
N-ethyl-2,2-dimethyl-N-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}oxan-4-amine
[(1,3-dimethyl-1H-pyrazol-5-yl)methyl](2-methoxyethyl)[(3-methylthiophen-2-yl)methyl]amine
1-{2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-1,3-oxazole-4-carbonyl}-3-phenylpiperidine
8-(2-amino-2-methylpropanoyl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
methyl 3-({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}amino)-3-phenylpropanoate
N,N-dimethyl-5-{[methyl(oxan-2-ylmethyl)amino]methyl}pyrimidin-2-amine