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N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2-oxo-6-[(4-phenylazepan-1-yl)methyl]-1,2-dihydropyridine-3-carboxamide
8-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-2-(3-hydroxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
3-{[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}benzonitrile
(1H-1,3-benzodiazol-2-ylmethyl)({[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl})methylamine
2-[3-(dimethylamino)propyl]-9-(naphthalen-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
8-methyl-3-{[4-(prop-2-en-1-yl)piperazin-1-yl]methyl}-1,2-dihydroquinolin-2-one
2-(pyrazin-2-yl)-1-{4-[2-(pyrrolidine-1-carbonyl)phenoxy]piperidin-1-yl}ethan-1-one
(2S,4S,5R)-4-{[2-(1H-imidazol-4-yl)ethyl]carbamoyl}-1,2-dimethyl-5-phenylpyrrolidine-2-carboxylic acid
3-methyl-7-[1-methyl-3-(thiophen-2-yl)-1H-pyrazole-5-carbonyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
4-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}-N-(2-methoxyethyl)-N-(propan-2-yl)benzamide
(2,4,6-trimethyl-3-{[(oxolan-2-ylmethyl)(pyridin-2-ylmethyl)amino]methyl}phenyl)methanol
1-(4-{[(3R,4S)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]methyl}phenyl)ethan-1-one
N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-2,3-dihydro-1-benzofuran-5-carboxamide
N-{imidazo[1,2-a]pyridin-3-ylmethyl}-5-(2-methoxyacetamido)-N-methyl-1-(2-phenylethyl)-1H-1,3-benzodiazole-7-carboxamide
3,4,7-trimethyl-N-[3-(1H-1,2,3-triazol-1-yl)propyl]-1H-indole-2-carboxamide
4-(4-{[({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)(methyl)amino]methyl}phenyl)-2-methylbut-3-yn-2-ol
N-cyclopropyl-2-[2,6,6-trimethyl-1-(2-methylpropyl)-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
1-[2-(2-chlorophenyl)-3-methyl-3H-imidazo[4,5-b]pyridine-6-carbonyl]-4-methylpiperazine
N-[2-(1-benzothiophen-2-yl)-2-hydroxyethyl]-2-(2-methyl-1,3-thiazol-4-yl)acetamide
3-(2-{1-[(4-methyl-1,3-thiazol-5-yl)methyl]piperidin-2-yl}ethyl)phenol
4-hydroxy-N-{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}-2-(4-methylphenyl)pyrimidine-5-carboxamide
2-[6-(morpholine-4-carbonyl)pyrazin-2-yl]-1,2,3,4-tetrahydroisoquinolin-4-ol
1-phenyl-3-(propan-2-yl)-4-(1,3-thiazol-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
3-[4-(adamantan-2-yl)piperazine-1-carbonyl]-2-(cyclopentylmethyl)-1-(2-methoxyethyl)-6-methyl-1,4-dihydropyridin-4-one
1-[(5-fluoro-2-methoxyphenyl)methyl]-3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
N-{2-[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]ethyl}-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
3-[1-(3-propyl-1,2,4-oxadiazol-5-yl)ethyl]-3H,4H-thieno[2,3-d]pyrimidin-4-one
1-(4-methyl-1,2,5-oxadiazol-3-yl)-4-(3-{[4-(propan-2-yl)phenyl]methyl}-1,2-oxazole-5-carbonyl)piperazine
N5-(cyclohexylmethyl)-N3-(2-hydroxy-2-phenylethyl)-N3-methyl-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
(3S,4S)-1-[(5-chloro-2,4-dimethoxyphenyl)methyl]-4-(pyrrolidin-1-yl)pyrrolidin-3-ol
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-2-(methylamino)pyridine-4-carboxamide
3-(pentan-2-yl)-8-(quinoxaline-5-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-(3-fluorophenyl)-1-[2-(piperidin-1-yl)ethyl]-6-(1,3-thiazole-5-carbonyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
4-cyclopentyl-3-(2-{4-[(3,4-dimethylphenyl)methyl]-3-oxopiperazin-1-yl}-2-oxoethyl)piperazin-2-one
1-[(3,4-difluorophenyl)methyl]-N-[4-(1,3-thiazol-4-yl)phenyl]piperidine-3-carboxamide
2-{[4-(pyrrolidine-1-sulfonyl)piperazin-1-yl]methyl}-4,5,6,7-tetrahydro-1,3-benzothiazole
2-({4-[(benzyloxy)methyl]-1H-1,2,3-triazol-1-yl}methyl)pyridine
methyl[(5-{[(2-methylphenyl)methyl]sulfanyl}-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl)methyl]{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}amine
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-methoxyacetamide
4-[1-(1-methyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]benzoic acid
1-{4-[(3,3-dimethylbutyl)amino]-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
(3R,4R)-4-(hydroxymethyl)-1-(6-phenylpyridazin-3-yl)piperidin-3-ol
ethyl 4-[1-(2-oxo-2-phenylacetyl)piperidin-3-yl]piperazine-1-carboxylate
1-[(2-{[3-chloro-5-(trifluoromethyl)pyridin-2-yl]oxy}phenyl)methyl]-4-methylpiperazine
N-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]-2-(2,5-dioxoimidazolidin-1-yl)acetamide
3-phenyl-4-[2-(propan-2-yl)pyrimidin-4-yl]-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
methyl({[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl})[1-(pyrimidin-4-yl)ethyl]amine
N-(1-{1-[2-(1H-pyrazol-1-yl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopentanecarboxamide
2,8-dimethyl-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}quinoline-4-carboxamide
7-acetamido-2-(2-methoxyphenyl)-1-methyl-N-[2-(pyrazin-2-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide